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Machine translation
1. (WO2007009705) (RAC)-N-PIPERIDINYL-5-(4-CHLOROPHENYL)-1-(2,4-DICHLOROPHENYL)-4,5-DIHYDR0-1H-PYRAZOLE-3-CARBOXAMIDE HYDRATES
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2007/009705    International Application No.:    PCT/EP2006/006979
Publication Date: 25.01.2007 International Filing Date: 15.07.2006
IPC:
C07D 231/06 (2006.01), A61K 31/4155 (2006.01), A61P 3/04 (2006.01), A61P 25/30 (2006.01), A61P 35/00 (2006.01)
Applicants: LABORATORIOS DEL DR. ESTEVE, S.A. [ES/ES]; Avenida Mare de Deu de Montserrat, 221, E-08041 Barcelona (ES) (For All Designated States Except US).
BUSCHMANN, Helmut, H. [DE/ES]; (ES) (For US Only).
TORRENS JOVER, Antonio [ES/ES]; (ES) (For US Only).
SOLA, Lluis [ES/ES]; (ES) (For US Only).
BENET BUCHHOLZ, Jordi [ES/ES]; (ES) (For US Only)
Inventors: BUSCHMANN, Helmut, H.; (ES).
TORRENS JOVER, Antonio; (ES).
SOLA, Lluis; (ES).
BENET BUCHHOLZ, Jordi; (ES)
Agent: PETERS, Hajo; Bosch, Graf von Stosch, Jehle Patentanwaltsgesells, chaft mbH, Flüggenstrasse 13, 80639 München (DE)
Priority Data:
05384011.2 15.07.2005 EP
60/705,472 05.08.2005 US
Title (EN) (RAC)-N-PIPERIDINYL-5-(4-CHLOROPHENYL)-1-(2,4-DICHLOROPHENYL)-4,5-DIHYDR0-1H-PYRAZOLE-3-CARBOXAMIDE HYDRATES
(FR) HYDRATES DE (RAC) -N-PIPERIDINYL-5- (4-CHLOROPHENYL) -1- (2, 4-DICHLOROPHENYL) -4, 5-DIHYDR0-1H-PYR AZOLE-3 -CARBOXAMIDE
Abstract: front page image
(EN)The present invention relates to (rac)-N-piperidinyl-5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4,5-dihydro-1H- pyrazole-3-carboxamide • X H2O, with X between 0.7 and 0.3. Especially preferred is (rac)-N-piperidinyl-5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4,5-dihydro-1H- pyrazole-3-carboxamide • monohydrate. Methods for their preparation, and their use as modulators of the cannabinoid receptor are also disclosed.
(FR)L'invention concerne un (rac)-N-pipéridinyl-5-(4-chlorophényl)-1-(2,4-dichlorophényl)-4,5-dihydro-1H- pyrazole-3-carboxamide X H2O, X étant compris entre 0,7 et 0,3. L'invention concerne de préférence (rac)-N-pipéridinyl-5-(4-chlorophényl)-1-(2,4-dichlorophényl)-4,5-dihydro-1H- pyrazole-3-carboxamide monohydrate. L'invention concerne également leurs procédés de préparation et leur utilisation comme modulateurs du récepteur cannabinoïde.
Designated States: AE, AG, AL, AM, AT, AU, AZ, BA, BB, BG, BR, BW, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DE, DK, DM, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LV, LY, MA, MD, MG, MK, MN, MW, MX, MZ, NA, NG, NI, NO, NZ, OM, PG, PH, PL, PT, RO, RS, RU, SC, SD, SE, SG, SK, SL, SM, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HU, IE, IS, IT, LT, LU, LV, MC, NL, PL, PT, RO, SE, SI, SK, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: English (EN)
Filing Language: English (EN)