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1. (WO2007009689) 4,5-DIHYDR0-1H-PYRAZOLE DERIVATIVES, THEIR PREPARATION AND USE AS MEDICAMENTS
Latest bibliographic data on file with the International Bureau

Pub. No.: WO/2007/009689 International Application No.: PCT/EP2006/006963
Publication Date: 25.01.2007 International Filing Date: 15.07.2006
IPC:
C07D 231/06 (2006.01) ,C07D 403/12 (2006.01) ,C07D 409/04 (2006.01) ,A61K 31/4155 (2006.01) ,A61K 31/415 (2006.01) ,A61P 3/04 (2006.01) ,A61P 25/30 (2006.01) ,A61P 35/00 (2006.01)
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
231
Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
02
not condensed with other rings
06
having one double bond between ring members or between a ring member and a non-ring member
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
403
Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/167
02
containing two hetero rings
12
linked by a chain containing hetero atoms as chain links
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
409
Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
02
containing two hetero rings
04
directly linked by a ring-member-to-ring- member bond
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
33
Heterocyclic compounds
395
having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
41
having five-membered rings with two or more ring hetero atoms, at least one of which is nitrogen, e.g. tetrazole
415
1,2-Diazoles
4155
not condensed and containing further heterocyclic rings
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
33
Heterocyclic compounds
395
having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
41
having five-membered rings with two or more ring hetero atoms, at least one of which is nitrogen, e.g. tetrazole
415
1,2-Diazoles
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
P
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
3
Drugs for disorders of the metabolism
04
Anorexiants; Antiobesity agents
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
P
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
25
Drugs for disorders of the nervous system
30
for treating abuse or dependence
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
P
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
35
Antineoplastic agents
Applicants:
LABORATORIOS DEL DR.ESTEVE, S.A. [ES/ES]; Avda Mare de Deu de Montserrat 221 E-08041 Barcelona, ES (AllExceptUS)
BUSCHMANN, Helmut [DE/ES]; ES (UsOnly)
TORRENS JOVER, Antonio [ES/ES]; ES (UsOnly)
MAS PRIO, Jose [ES/ES]; ES (UsOnly)
QUINTANA RUIZ, Jordi, Ramon [ES/ES]; ES (UsOnly)
YENES MINGUEZ, Susana [ES/ES]; ES (UsOnly)
Inventors:
BUSCHMANN, Helmut; ES
TORRENS JOVER, Antonio; ES
MAS PRIO, Jose; ES
QUINTANA RUIZ, Jordi, Ramon; ES
YENES MINGUEZ, Susana; ES
Agent:
HAJO, Peters; Bosch, Graf von Stosch, Jehle Patentanwaltsgesells chaft mbH Flüggenstrasse 13 80639 München, DE
Priority Data:
05384029.415.07.2005EP
60/705,43205.08.2005US
Title (EN) 4,5-DIHYDR0-1H-PYRAZOLE DERIVATIVES, THEIR PREPARATION AND USE AS MEDICAMENTS
(FR) DERIVES DE 4, 5-DIHYDR0-1H-PYRAZOLE, PREPARATION ET UTILISATION DE CEUX-CI COMME MEDICAMENTS
Abstract:
(EN) The present invention relates to 4-substituted pyrazoline compounds of formula (I), methods for their preparation, medicaments comprising these compounds as well as their use for the preparation of a medicament for the treatment of humans and animals.
(FR) L'invention concerne des composés de pyrazoline 4 substituée de formule I, des procédés de préparation de ceux-ci, des médicaments comprenant ces composés, ainsi que l'utilisation de ceux-ci dans la préparation d'un médicament destiné au traitement d'êtres humains et d'animaux.
Designated States: AE, AG, AL, AM, AT, AU, AZ, BA, BB, BG, BR, BW, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DE, DK, DM, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LV, LY, MA, MD, MG, MK, MN, MW, MX, MZ, NA, NG, NI, NO, NZ, OM, PG, PH, PL, PT, RO, RS, RU, SC, SD, SE, SG, SK, SL, SM, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW
African Regional Intellectual Property Organization (ARIPO) (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HU, IE, IS, IT, LT, LU, LV, MC, NL, PL, PT, RO, SE, SI, SK, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG)
Publication Language: English (EN)
Filing Language: English (EN)
Also published as:
MXMX/a/2008/000736KR1020080032157EP1917247BRPI0613057-7JP2009501181CN101263120
CA2612468AU2006271994IN10113/DELNP/2007