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1. (WO2007008317) PROCESS FOR PREPARATION OF SERTRALINE HYDROCHLORIDE FORM I
Latest bibliographic data on file with the International Bureau

Pub. No.: WO/2007/008317 International Application No.: PCT/US2006/022500
Publication Date: 18.01.2007 International Filing Date: 09.06.2006
IPC:
C07C 211/42 (2006.01) ,A61K 31/137 (2006.01) ,A61P 25/22 (2006.01) ,A61P 25/24 (2006.01)
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
C
ACYCLIC OR CARBOCYCLIC COMPOUNDS
211
Compounds containing amino groups bound to a carbon skeleton
33
having amino groups bound to carbon atoms of rings other than six-membered aromatic rings
39
of an unsaturated carbon skeleton
41
containing condensed ring systems
42
with six-membered aromatic rings being part of the condensed ring systems
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
13
Amines, e.g. amantadine
135
having aromatic rings, e.g. methadone
137
Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
P
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
25
Drugs for disorders of the nervous system
22
Anxiolytics
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
P
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
25
Drugs for disorders of the nervous system
24
Antidepressants
Applicants:
TEVA PHARMACEUTICAL INDUSTRIES LTD. [IL/IL]; 5 BASEL STREET P.o. Box 3190 49131 Petah Tiqva, IL (AE, AG, AL, AM, AT, AU, AZ, BA, BE, BF, BG, BJ, BR, BW, BY, BZ, CA, CF, CG, CH, CI, CM, CN, CO, CR, CU, CY, CZ, DE, DK, DM, DZ, EC, EE, EG, ES, FI, FR, GA, GB, GD, GE, GH, GM, GN, GQ, GR, GW, HR, HU, ID, IE, IL, IN, IS, IT, JP, KE, KG, KM, KN, KP, KR, KZ, LC, LK, LR, LS, LT, LU, LV, LY, MA, MC, MD, MG, MK, ML, MN, MR, MW, MX, MZ, NA, NE, NG, NI, NL, NO, NZ, OM, PG, PH, PL, PT, RO, RS, RU, SC, SD, SE, SG, SI, SK, SL, SM, SN, SY, SZ, TD, TG, TJ, TM, TN, TR, TT, TZ, UA, UG, UZ, VC, VN, ZA, ZM, ZW)
TEVA PHARMACEUTICALS USA, INC. [US/US]; 1090 HORSHAM ROAD P.o. Box 1090 North Wales, PA 19454-1090, US (BB)
BOROCHOVITZ, Ronen [IL/IL]; IL (UsOnly)
SHABAT, Shalom [IL/IL]; IL (UsOnly)
Inventors:
BOROCHOVITZ, Ronen; IL
SHABAT, Shalom; IL
Agent:
BIRDE, Patrick, J. ; KENYON & KENYON LLP One Broadway New York, NY 10004-1050, US
Priority Data:
60/689,77709.06.2005US
Title (EN) PROCESS FOR PREPARATION OF SERTRALINE HYDROCHLORIDE FORM I
(FR) PROCEDE DE PREPARATION DE LA FORME I DE CHLORHYDRATE DE SERTRALINE
Abstract:
(EN) Provided is a process for preparation of sertraline HCl Form I on an industrial scale comprising steps of : a) heating sertraline HCI in n-butanol to a temperature of about 400 C to about reflux temperature, and b) crystallizing sertraline HCI
(FR) L'invention concerne un procédé de préparation de la forme I de HCl de sertraline à l'échelle industrielle.
Designated States: AE, AG, AL, AM, AT, AU, AZ, BA, BB, BG, BR, BW, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DE, DK, DM, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LC, LK, LR, LS, LT, LU, LV, LY, MA, MD, MG, MK, MN, MW, MX, MZ, NA, NG, NI, NO, NZ, OM, PG, PH, PL, PT, RO, RS, RU, SC, SD, SE, SG, SK, SL, SM, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW
African Regional Intellectual Property Organization (ARIPO) (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HU, IE, IS, IT, LT, LU, LV, MC, NL, PL, PT, RO, SE, SI, SK, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG)
Publication Language: English (EN)
Filing Language: English (EN)
Also published as:
IL185730EP1893559