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1. (WO2007005174) 4- (3 -HYDROXY- AND 3-AMINOMETHYL-CYCLOHEXEN-3-YLMETHYL) 1, 3-DIHYDROIMDAZOLE-2-THIONE DERIVATIVES AS ALPHA-2 ADRENERGIC AGONISTS
Latest bibliographic data on file with the International Bureau

Pub. No.: WO/2007/005174 International Application No.: PCT/US2006/021866
Publication Date: 11.01.2007 International Filing Date: 06.06.2006
IPC:
C07D 233/84 (2006.01) ,A61K 31/4164 (2006.01) ,A61P 5/24 (2006.01) ,A61P 9/12 (2006.01) ,A61P 25/24 (2006.01) ,A61P 27/06 (2006.01) ,A61P 29/00 (2006.01)
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
233
Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
54
having two double bonds between ring members or between ring members and non-ring members
66
with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
84
Sulfur atoms
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
33
Heterocyclic compounds
395
having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
41
having five-membered rings with two or more ring hetero atoms, at least one of which is nitrogen, e.g. tetrazole
4164
1,3-Diazoles
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
P
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
5
Drugs for disorders of the endocrine system
24
of the sex hormones
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
P
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
9
Drugs for disorders of the cardiovascular system
12
Antihypertensives
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
P
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
25
Drugs for disorders of the nervous system
24
Antidepressants
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
P
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
27
Drugs for disorders of the senses
02
Ophthalmic agents
06
Antiglaucoma agents or miotics
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
P
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
29
Non-central analgesic, antipyretic or antiinflammatory agents, e.g antirheumatic agents; Non-steroidal antiinflammatory drugs (NSAIDs)
Applicants:
ALLERGAN, INC. [US/US]; 2525 Dupont Drive Irvine, CA 92612, US (AllExceptUS)
CHOW, Ken [US/US]; US (UsOnly)
HEIDELBAUGH, Todd, M. [US/US]; US (UsOnly)
NGUYEN, Phong, X. [US/US]; US (UsOnly)
Inventors:
CHOW, Ken; US
HEIDELBAUGH, Todd, M.; US
NGUYEN, Phong, X.; US
Agent:
JOHNSON, Brent, A. ; Allergan, Inc. 2525 Dupont Drive Irvine, CA 92612, US
Priority Data:
11/172,22929.06.2005US
Title (EN) 4- (3 -HYDROXY- AND 3-AMINOMETHYL-CYCLOHEXEN-3-YLMETHYL) 1, 3-DIHYDROIMDAZOLE-2-THIONE DERIVATIVES AS ALPHA-2 ADRENERGIC AGONISTS
(FR) AGONISTES ADRENERGIQUES ALPHA-2
Abstract:
(EN) A compound is disclosed herein comprising Formulat (I); or a pharmaceutically acceptable salt or a prodrug thereof; wherein R is OH or NH2- Methods, compositions, and medicaments related thereto are also disclosed.
(FR) L'invention concerne un composé de formule (I); ou un sel pharmaceutiquement acceptable ou un promédicament de celui-ci. Dans la formule (I), R désigne OH ou NH2-. L'invention concerne également des méthodes, des compositions, et des médicaments associés à ce composé.
front page image
Designated States: AE, AG, AL, AM, AT, AU, AZ, BA, BB, BG, BR, BW, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DE, DK, DM, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LC, LK, LR, LS, LT, LU, LV, LY, MA, MD, MG, MK, MN, MW, MX, MZ, NA, NG, NI, NO, NZ, OM, PG, PH, PL, PT, RO, RS, RU, SC, SD, SE, SG, SK, SL, SM, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW
African Regional Intellectual Property Organization (ARIPO) (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HU, IE, IS, IT, LT, LU, LV, MC, NL, PL, PT, RO, SE, SI, SK, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG)
Publication Language: English (EN)
Filing Language: English (EN)