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1. (WO2007003422) CRYSTALLINE FORMS OF MACROLIDE COMPOUNDS ENDOWED WITH ANTIINFLAMMATORY ACTIVITY
Latest bibliographic data on file with the International Bureau

Pub. No.: WO/2007/003422 International Application No.: PCT/EP2006/006541
Publication Date: 11.01.2007 International Filing Date: 05.07.2006
IPC:
C07H 17/08 (2006.01) ,A61K 31/7048 (2006.01) ,A61P 29/00 (2006.01)
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
H
SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
17
Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
04
Heterocyclic radicals containing only oxygen as ring hetero atoms
08
Hetero rings containing eight or more ring members, e.g. erythromycins
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
70
Carbohydrates; Sugars; Derivatives thereof
7042
Compounds having saccharide radicals and heterocyclic rings
7048
having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
P
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
29
Non-central analgesic, antipyretic or antiinflammatory agents, e.g antirheumatic agents; Non-steroidal antiinflammatory drugs (NSAIDs)
Applicants:
ZAMBON S.P.A. [IT/IT]; Via Lillo del Duca, 10 I-20091 Bresso, IT (AllExceptUS)
MARAGNI, Paolo [IT/IT]; IT (UsOnly)
BRAGA, Dario [IT/IT]; IT (UsOnly)
BRESCELLO, Roberto [IT/IT]; IT (UsOnly)
COTARCA, Livius [RO/IT]; IT (UsOnly)
DI MARIA, Alessandro [IT/IT]; IT (UsOnly)
MASSACCESI, Franco [IT/IT]; IT (UsOnly)
MELOTTO, Elisa [IT/IT]; IT (UsOnly)
MICHIELETTO, Ivan [IT/IT]; IT (UsOnly)
MORAZZONI, Gabriele [IT/IT]; IT (UsOnly)
NAPOLETANO, Mauro [IT/IT]; IT (UsOnly)
PELLACINI, Franco [IT/IT]; IT (UsOnly)
RESTELLI, Angelo [IT/IT]; IT (UsOnly)
VERZINI, Massimo [IT/IT]; IT (UsOnly)
Inventors:
MARAGNI, Paolo; IT
BRAGA, Dario; IT
BRESCELLO, Roberto; IT
COTARCA, Livius; IT
DI MARIA, Alessandro; IT
MASSACCESI, Franco; IT
MELOTTO, Elisa; IT
MICHIELETTO, Ivan; IT
MORAZZONI, Gabriele; IT
NAPOLETANO, Mauro; IT
PELLACINI, Franco; IT
RESTELLI, Angelo; IT
VERZINI, Massimo; IT
Agent:
MORELLI, Roberta; Zambon S.p.A. Patent Office Via Lillo del Duca, 10 I-20091 Bresso, IT
Priority Data:
05106123.206.07.2005EP
Title (EN) CRYSTALLINE FORMS OF MACROLIDE COMPOUNDS ENDOWED WITH ANTIINFLAMMATORY ACTIVITY
(FR) FORMES CRISTALLINES DE COMPOSES MACROLIDES DOTES D'UNE ACTIVITE ANTI-INFLAMMATOIRE
Abstract:
(EN) The present invention relates to macrolide compounds endowed with antiinflammatory activity and more particularly relates to new stable crystalline forms of a macrolide derivative with antiinflammatory activity, processes for the preparation of such forms, pharmaceutical compositions containing them as active ingredient and the use of said crystalline Forms for the treatment of inflammatory diseases.
(FR) L'invention concerne des composés macrolides dotés d'une activité anti-inflammatoire et, pus précisément, des formes cristallines stables d'un dérivé de macrolide possédant une activité anti-inflammatoire, des procédés de préparation de telles formes, des compositions pharmaceutiques renfermant celles-ci comme principe actif et l'utilisation des formes cristallines dans le traitement de maladies inflammatoires.
Designated States: AE, AG, AL, AM, AT, AU, AZ, BA, BB, BG, BR, BW, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DE, DK, DM, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LV, LY, MA, MD, MG, MK, MN, MW, MX, MZ, NA, NG, NI, NO, NZ, OM, PG, PH, PL, PT, RO, RS, RU, SC, SD, SE, SG, SK, SL, SM, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW
African Regional Intellectual Property Organization (ARIPO) (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HU, IE, IS, IT, LT, LU, LV, MC, NL, PL, PT, RO, SE, SI, SK, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG)
Publication Language: English (EN)
Filing Language: English (EN)
Also published as:
RSP-2010/0268MXMX/a/2008/000279IL188400EP1907406BRPI0612598-0ZA2008/00414
JP2008544970ES2343748US20090018089CN101291947CN102295671CA2613911
EA200800266PT1907406AU2006265277DK1907406IN620/CHENP/2008