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1. (WO2007002308) PROCESS FOR PREPARING TRIAZOLE SUBSTITUTED AZAINDOLEOXOACETIC PIPERAZINE DERIVATIVES AND NOVEL SALT FORMS PRODUCED THEREIN
Latest bibliographic data on file with the International Bureau

Pub. No.: WO/2007/002308 International Application No.: PCT/US2006/024335
Publication Date: 04.01.2007 International Filing Date: 21.06.2006
IPC:
C07D 471/04 (2006.01) ,A61K 31/4745 (2006.01) ,A61P 31/12 (2006.01)
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
471
Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/-C07D463/251
02
in which the condensed system contains two hetero rings
04
Ortho-condensed systems
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
33
Heterocyclic compounds
395
having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
435
having six-membered rings with one nitrogen as the only ring hetero atom
47
Quinolines; Isoquinolines
4738
ortho- or peri-condensed with heterocyclic ring systems
4745
condensed with ring systems having nitrogen as a ring hetero atom, e.g. phenanthrolines
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
P
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
31
Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
12
Antivirals
Applicants:
BRISTOL-MYERS SQUIBB COMPANY [US/US]; P.O. Box 4000 Route 206 And Provinceline Road Princeton, New Jersey 08543-4000, US (AllExceptUS)
SOUNDARARAJAN, Nachimuthu [US/US]; US (UsOnly)
QIU, Yuping [CN/US]; US (UsOnly)
HU, Wenhao [CN/US]; US (UsOnly)
KRONENTHAL, David, R. [US/US]; US (UsOnly)
SIRARD, Pierre [CA/CA]; CA (UsOnly)
LAJEUNESSE, Jean [CA/CA]; CA (UsOnly)
DROGHINI, Roberto [CA/CA]; CA (UsOnly)
CHIDAMBARAM, Ramakrishnan [US/US]; US (UsOnly)
QIAN, Xinhua [US/US]; US (UsOnly)
NATALIE, JR., Kenneth, J. [US/US]; US (UsOnly)
PACK, Shawn, K. [US/US]; US (UsOnly)
REISING, Nathan [US/US]; US (UsOnly)
TANG, Erqing [US/US]; US (UsOnly)
FAKES, Michael, G. [US/US]; US (UsOnly)
GAO, Qi [US/US]; US (UsOnly)
QIAN, Feng [CN/US]; US (UsOnly)
VAKKALAGADDA, Blisse, J. [IN/US]; US (UsOnly)
LAI, Chiajen [CN/US]; US (UsOnly)
KUANG, Shan-Ming [CN/US]; US (UsOnly)
Inventors:
SOUNDARARAJAN, Nachimuthu; US
QIU, Yuping; US
HU, Wenhao; US
KRONENTHAL, David, R.; US
SIRARD, Pierre; CA
LAJEUNESSE, Jean; CA
DROGHINI, Roberto; CA
CHIDAMBARAM, Ramakrishnan; US
QIAN, Xinhua; US
NATALIE, JR., Kenneth, J.; US
PACK, Shawn, K.; US
REISING, Nathan; US
TANG, Erqing; US
FAKES, Michael, G.; US
GAO, Qi; US
QIAN, Feng; US
VAKKALAGADDA, Blisse, J.; US
LAI, Chiajen; US
KUANG, Shan-Ming; US
Agent:
RODNEY, Burton ; Bristol-Myers Squibb Company P.o. Box 4000 Princeton, New Jersey 08543-4000, US
Priority Data:
60/693,00422.06.2005US
Title (EN) PROCESS FOR PREPARING TRIAZOLE SUBSTITUTED AZAINDOLEOXOACETIC PIPERAZINE DERIVATIVES AND NOVEL SALT FORMS PRODUCED THEREIN
(FR) PROCEDE DE PREPARATION DE DERIVES DE PIPERAZINE AZAINDOLEOXOACETIQUE A SUBSTITUTION TRIAZOLE ET NOUVELLES FORMES DE SELS OBTENUES SELON CE PROCEDE
Abstract:
(EN) A process is provided for preparing triazole substituted azaindoleoxoacetic piperazine derivative. Novel intermediates produced in the above process, and novel N-1 and amorphous forms of a 1,2,3-triazole substituted azaindoloxoacetic piperazine derivatives and processes for producing such novel forms are also provided.
(FR) L'invention concerne un procédé de préparation de dérivés de pipérazine azaindoléoxoacétique à substitution triazole. L'invention concerne également de nouveaux intermédiaires produits selon ledit procédé, et de nouvelles formes N-1 et amorphes de dérivés de pipérazine azaindoléoxoacétique 1,2,3-triazole substitués ainsi que des procédés de production de ces nouvelles formes.
front page image
Designated States: AE, AG, AL, AM, AT, AU, AZ, BA, BB, BG, BR, BW, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DE, DK, DM, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LV, LY, MA, MD, MG, MK, MN, MW, MX, MZ, NA, NG, NI, NO, NZ, OM, PG, PH, PL, PT, RO, RS, RU, SC, SD, SE, SG, SK, SL, SM, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW
African Regional Intellectual Property Organization (ARIPO) (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HU, IE, IS, IT, LT, LU, LV, MC, NL, PL, PT, RO, SE, SI, SK, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG)
Publication Language: English (EN)
Filing Language: English (EN)
Also published as:
NO20076575PE2007-0122EP1907389JP2008546795ES2368788CN101243085
IN75/DELNP/2008