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1. (WO2007000644) HOMOMORPHOLINE OXAZOLIDINONES AS ANTIBACTERIAL AGENTS
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2007/000644    International Application No.:    PCT/IB2006/001730
Publication Date: 04.01.2007 International Filing Date: 20.06.2006
IPC:
C07D 413/10 (2006.01), C07D 413/14 (2006.01), A61P 31/04 (2006.01), A61K 31/4178 (2006.01)
Applicants: PHARMACIA & UPJOHN COMPANY LLC [US/US]; 7000 Portage Road, Kalamazoo, Michigan 49001-0199 (US) (For All Designated States Except US).
JOSYULA, Vara Prasad Venkata Nagendra [US/US]; (US) (For US Only).
BOYER, Frederick, Earl, Jr. [US/US]; (US) (For US Only).
KIM, Ji-Young [US/US]; (US) (For US Only)
Inventors: JOSYULA, Vara Prasad Venkata Nagendra; (US).
BOYER, Frederick, Earl, Jr.; (US).
KIM, Ji-Young; (US)
Agent: FULLER, Grover, F., Jr.; Pfizer Inc., 150 East 42nd Street, New York, NY 10017-5612 (US)
Priority Data:
60/694,862 29.06.2005 US
Title (EN) HOMOMORPHOLINE OXAZOLIDINONES AS ANTIBACTERIAL AGENTS
(FR) OXAZOLIDINONES D'HOMOMORPHOLINE EN TANT QU'AGENTS ANTIBACTERIENS
Abstract: front page image
(EN)The present invention provides a compound of formula (I) or a pharmaceutically acceptable salt thereof wherein X is -C(=O)NHR4, or CH2-het; R1, R2, R3 are independently H or F; R4 is H, C1-6 alkyl, or OC1-6alkyl; het is a five (5)-membered heterocyclic ring having 1, 2 or 3 heteroatoms selected from the group consisting of non-peroxide oxygen, sulfur, and nitrogen within the ring. The compounds of the present are useful as antibacterial agents.
(FR)La présente invention a trait à un composé de formule (I) dans laquelle: X est -C(=O)NHR4, ou CH2-het; R1, R2, R3 sont indépendamment H ou F; R4 est H, alkyle en C1-C6, ou OC1-6alkyle; het est un noyau hétérocyclique à cinq chaînons ayant 1, 2, 3 hétéroatomes choisis parmi le groupe constitué d'oxygène non peroxyde, de soufre, et d'azote dans le noyau, ou un sel pharmaceutiquement acceptable de celui-ci. Les composés de la présente invention sont utiles en tant qu'agents antibactériens.
Designated States: AE, AG, AL, AM, AT, AU, AZ, BA, BB, BG, BR, BW, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DE, DK, DM, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LV, LY, MA, MD, MG, MK, MN, MW, MX, MZ, NA, NG, NI, NO, NZ, OM, PG, PH, PL, PT, RO, RS, RU, SC, SD, SE, SG, SK, SL, SM, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HU, IE, IS, IT, LT, LU, LV, MC, NL, PL, PT, RO, SE, SI, SK, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: English (EN)
Filing Language: English (EN)