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1. (WO2006120541) ETHER LINKED MACROLIDES USEFUL FOR THE TREATMENT OF MICROBIAL INFECTIONS
Latest bibliographic data on file with the International Bureau   

Pub. No.: WO/2006/120541 International Application No.: PCT/IB2006/001194
Publication Date: 16.11.2006 International Filing Date: 09.05.2006
Chapter 2 Demand Filed: 01.03.2007
IPC:
C07H 17/08 (2006.01) ,A61K 31/7048 (2006.01)
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
H
SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
17
Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
04
Heterocyclic radicals containing only oxygen as ring hetero atoms
08
Hetero rings containing eight or more ring members, e.g. erythromycins
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
70
Carbohydrates; Sugars; Derivatives thereof
7042
Compounds having saccharide radicals and heterocyclic rings
7048
having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin
Applicants:
ALIHODZIC, Sulejman [HR/HR]; HR (UsOnly)
PAVLOVIC, Drazen [HR/HR]; HR (UsOnly)
HUNT, Eric [GB/GB]; GB (UsOnly)
FORREST, Andrew, Keith [GB/GB]; GB (UsOnly)
PALEJ, Ivana [HR/HR]; HR (UsOnly)
KAPIC, Samra [HR/HR]; HR (UsOnly)
STIMAC, Vlado [HR/HR]; HR (UsOnly)
GLAXOSMITHKLINE ISTRAZIVACKI CENTAR ZAGREB D.O.O. [HR/HR]; Prilaz baruna Filipovica 29 10000 Zagreb, HR (AllExceptUS)
GLAXO GROUP LTD. [GB/GB]; Glaxo Wellcome House Berkeley Avenue Greenford UB6 0NN, GB (AllExceptUS)
Inventors:
ALIHODZIC, Sulejman; HR
PAVLOVIC, Drazen; HR
HUNT, Eric; GB
FORREST, Andrew, Keith; GB
PALEJ, Ivana; HR
KAPIC, Samra; HR
STIMAC, Vlado; HR
Agent:
CRAWLEY, Karen; GlaxoSmithKline CIP (CN925.1) 980 Great West Road, Brentford Middlesex TW8 9GS, GB
Priority Data:
60/679,77910.05.2005US
Title (EN) ETHER LINKED MACROLIDES USEFUL FOR THE TREATMENT OF MICROBIAL INFECTIONS
(FR) MACROLIDES A LIAISON ETHER CONVENANT POUR LE TRAITEMENT DES INFECTIONS MICROBIENNES
Abstract:
(EN) The present invention relates to 14- or 15-membered macrolides substituted at the 4' position of formula (I) in which R1 is a ether moiety and pharmaceutically acceptable derivatives thereof, to processes for their preparation and their use in therapy or prophylaxis of systemic or topical microbial infections in a human or animal body.
(FR) L'invention concerne des macrolides à 14 ou 15 chaînons substitués en position- 4', représentés par la formule (I), et des dérivés pharmaceutiquement acceptables de ceux-ci, ainsi que des procédés permettant de préparer ces composés, et leur utilisation pour le traitement ou la prévention des infections microbiennes systémiques ou topiques chez l'homme ou chez l'animal.
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Designated States: AE, AG, AL, AM, AT, AU, AZ, BA, BB, BG, BR, BW, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DE, DK, DM, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LC, LK, LR, LS, LT, LU, LV, LY, MA, MD, MG, MK, MN, MW, MX, MZ, NA, NG, NI, NO, NZ, OM, PG, PH, PL, PT, RO, RU, SC, SD, SE, SG, SK, SL, SM, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, YU, ZA, ZM, ZW
African Regional Intellectual Property Organization (ARIPO) (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Office (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (EPO) (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HU, IE, IS, IT, LT, LU, LV, MC, NL, PL, PT, RO, SE, SI, SK, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG)
Publication Language: English (EN)
Filing Language: English (EN)