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1. (WO2006106440) MACROLIDE COMPOUNDS CONTAINING BIOTIN AND PHOTO-AFFINITY GROUP FOR MACROLIDE TARGET IDENTIFICATION
Latest bibliographic data on file with the International Bureau   

Pub. No.: WO/2006/106440 International Application No.: PCT/IB2006/001484
Publication Date: 12.10.2006 International Filing Date: 13.01.2006
Chapter 2 Demand Filed: 06.12.2006
IPC:
C07H 17/08 (2006.01)
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
H
SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
17
Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
04
Heterocyclic radicals containing only oxygen as ring hetero atoms
08
Hetero rings containing eight or more ring members, e.g. erythromycins
Applicants:
CULIC, Ognjen [HR/HR]; HR (UsOnly)
BOSNAR, Martina [HR/HR]; HR (UsOnly)
MARJANOVIC, Nikola [HR/HR]; HR (UsOnly)
MILDNER, Boris [HR/HR]; HR (UsOnly)
TOMASKOVIC, Linda [HR/HR]; HR (UsOnly)
ALIHODZIC, Sulejman [HR/HR]; HR (UsOnly)
GLAXOSMITHKLINE ISTRAZIVACKI CENTAR ZAGREB D.O.O. [HR/HR]; Prilaz Baruna Filipovica 29 10000 Zagreb, HR (AllExceptUS)
Inventors:
CULIC, Ognjen; HR
BOSNAR, Martina; HR
MARJANOVIC, Nikola; HR
MILDNER, Boris; HR
TOMASKOVIC, Linda; HR
ALIHODZIC, Sulejman; HR
Agent:
CRAWLEY, Karen; GlaxoSmithKline Corporate Intellectual Property CN925.1 980 Great West Road Brentford Middlesex TW8 9GS, GB
Priority Data:
60/644,33314.01.2005US
Title (EN) MACROLIDE COMPOUNDS CONTAINING BIOTIN AND PHOTO-AFFINITY GROUP FOR MACROLIDE TARGET IDENTIFICATION
(FR) COMPOSES MACROLIDE CONTENANT DE LA BIOTINE ET UN GROUPE A PHOTO-AFFINITE POUR L'IDENTIFICATION CIBLE DE MACROLIDE
Abstract:
(EN) The present invention relates to new macrolide compounds represented by the general structure I, wherein M is a macrolide, P is a photo-affinity group bearing subunit containing biotin, and L is a linking molecule, and to their pharmaceutically acceptable salts and solvates, to processes and intermediates for their preparation and to the use of these compounds for Hie macrolide target identification.
(FR) L'invention concerne de nouveaux composés macrolide représentés par la structure générale (I) dans laquelle M désigne un macrolide, P désigne un groupe à photo-affinité portant une sous-unité contenant de la biotine, et L désigne une molécule de liaison. L'invention concerne en outre les sels pharmaceutiquement acceptables et les solvates de ces composés, ainsi que des procédés et des produits intermédiaires pour leur préparation. Elle concerne également l'utilisation de ces composés pour l'identification cible de macrolide Hie.
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Designated States: AE, AG, AL, AM, AT, AU, AZ, BA, BB, BG, BR, BW, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DE, DK, DM, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LC, LK, LR, LS, LT, LU, LV, LY, MA, MD, MG, MK, MN, MW, MX, MZ, NA, NG, NI, NO, NZ, OM, PG, PH, PL, PT, RO, RU, SC, SD, SE, SG, SK, SL, SM, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, YU, ZA, ZM, ZW
African Regional Intellectual Property Organization (ARIPO) (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Office (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (EPO) (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HU, IE, IS, IT, LT, LU, LV, MC, NL, PL, PT, RO, SE, SI, SK, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG)
Publication Language: English (EN)
Filing Language: English (EN)