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1. WO2006094994 - USE OF 4-AMINOPYRIMIDINES FOR THE PREVENTION OF FUNGAL PESTS NOVEL 4-AMINOPYRIMIDINES METHOD FOR PRODUCTION THEREOF AND AGENTS COMPRISING THE SAME

Publication Number WO/2006/094994
Publication Date 14.09.2006
International Application No. PCT/EP2006/060557
International Filing Date 08.03.2006
IPC
A01N 43/54 2006.01
AHUMAN NECESSITIES
01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
43Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
48having rings with two nitrogen atoms as the only ring hetero atoms
541,3-Diazines; Hydrogenated 1,3-diazines
A01P 3/00 2006.01
AHUMAN NECESSITIES
01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
PBIOCIDAL, PEST REPELLANT, PEST ATTRACTANT OR PLANT GROWTH REGULATORY ACTIVITY OF CHEMICAL COMPOUNDS OR PREPARATIONS
3Fungicides
C07D 239/00 2006.01
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
239Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
CPC
A61P 11/00
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
11Drugs for disorders of the respiratory system
A61P 11/06
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
11Drugs for disorders of the respiratory system
06Antiasthmatics
A61P 11/08
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
11Drugs for disorders of the respiratory system
08Bronchodilators
A61P 15/06
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
15Drugs for genital or sexual disorders
06Antiabortive agents; Labour repressants
A61P 17/00
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
17Drugs for dermatological disorders
A61P 17/04
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
17Drugs for dermatological disorders
04Antipruritics
Applicants
  • BASF AKTIENGESELLSCHAFT [DE]/[DE] (AllExceptUS)
  • SCHWÖGLER, Anja [DE]/[DE] (UsOnly)
  • RHEINHEIMER, Joachim [DE]/[DE] (UsOnly)
  • GRAMMENOS, Wassilios [GR]/[DE] (UsOnly)
  • GROTE, Thomas [DE]/[DE] (UsOnly)
  • HÜNGER, Udo [DE]/[DE] (UsOnly)
  • MÜLLER, Bernd [DE]/[DE] (UsOnly)
  • SCHÄFER, Peter [DE]/[DE] (UsOnly)
  • SCHIEWECK, Frank [DE]/[DE] (UsOnly)
Inventors
  • SCHWÖGLER, Anja
  • RHEINHEIMER, Joachim
  • GRAMMENOS, Wassilios
  • GROTE, Thomas
  • HÜNGER, Udo
  • MÜLLER, Bernd
  • SCHÄFER, Peter
  • SCHIEWECK, Frank
Common Representative
  • BASF AKTIENGESELLSCHAFT
Priority Data
10 2005 011 583.710.03.2005DE
Publication Language German (DE)
Filing Language German (DE)
Designated States
Title
(DE) VERWENDUNG VON 4-AMINOPYRIMIDINEN ZUR BEKÄMPFUNG VON SCHADPILZEN, NEUE 4-AMINOPYRIMIDINE, VERFAHREN ZU IHRER HERSTELLUNG SOWIE SIE ENTHALTENDE MITTEL
(EN) USE OF 4-AMINOPYRIMIDINES FOR THE PREVENTION OF FUNGAL PESTS NOVEL 4-AMINOPYRIMIDINES METHOD FOR PRODUCTION THEREOF AND AGENTS COMPRISING THE SAME
(FR) UTILISATION DE 4-AMINOPYRIMIDINES DANS LA LUTTE CONTRE DES CHAMPIGNONS PARASITES, DE NOUVELLES 4-AMINOPYRIMIDINES, DES PROCEDES DE PRODUCTION DESDITS COMPOSES ET DES AGENTS CONTENANT CES DERNIERS
Abstract
(DE)
Verwendung von 4-Aminopyrimidinen der Formel (I), in der die Substituenten folgende Bedeutung haben: R1 Wasserstoff, Halogen, Cyano, Alkyl, Halogenalkyl, Alkenyl, Alkinyl, Cycloalkyl, Alkoxy, Alkoxyalkyl, Benzyloxyalkyl, Alkoxyalkenyl oder Alkoxyalkinyl; R2 Wasserstoff, Halogen, Cyano, Alkyl, Halogenalkyl, Alkenyl, Alkinyl, Cycloalkyl, Alkoxy, Alkoxyalkyl und Alkylthioalkyl, wobei die Kohlenstoffketten in R1 und/oder R2 gemäß der Beschreibung substituiert sein können, R1 und R2 können gemeinsam mit den Kohlenstoffatomen, an die sie gebunden sind, einen fünf- bis siebengliederigen Ring bilden, der ein bis drei gleiche oder verschiedene Heteroatome aus der Gruppe O, N oder S enthalten kann; R3 Wasserstoff, Halogen, Cyano, Hydroxy, Mercapto, Azido, Alkyl, Alkenyl, Alkinyl, Halogenalkyl, -O-D, -S(O)m-D, ON=CRaRb, CRc=NORa, NRcN=CRaRb, NRaRb, NRcNRaRb, NORa, NRcC(=NRc')NRaRb, NRcC(=O)NRaRb, NRaCN,-NRaC(=O)Rc, NRaC(=NORc)Rc', OC(=O)Ra, C(=NORc)NRaRb, CRc(=NNRaRb), C(=O)NRaRb , C(=O)Ra, CO2Ra, C(=O)NRzRb, C(=O)-N-ORb, C(=S)-NRzRb, C(=NORa)NRzRb, C(=NRa)NRzRb, C(=O)NRa-NRzRb, C(=N-NRzRc)NRaRb, C(=NORb)Ra, C(=N-NRzRb)Ra, CRaRb-ORz, CRaRb-NRzRc, ON(=CRaRb), NRa(C(=O)Rb), NRa(C(=O)ORb), NRa(C(=O)-NRzRb), NRa(C(=NRc)Rb), NRa(N=CRcRb), NRa-NRzRb, -NRz-ORa, NRa(C(=NRc)-NRzRb), NRa(C(=NORc)Rb), D Alkyl, Alkenyl, Alkinyl, Halogenalkyl, Cyclalkyl; fünf- oder sechsgliedriger gesättigter, partiell ungesättigter oder aromatischer mono- oder bicyclischer Heterocyclus, enthaltend ein bis vier Heteroatome aus der Gruppe O, N oder S, eine der Gruppen G1 oder G2, wobei m, x, Ra, Rb, Rc, Rd, Re, Rz, Y, Z gemäß der Beschreibung definiert sind und die aliphatischen, alicyclischen oder aromatischen Gruppen R3, Ra,Rb,Rc, Rd oder Re gemäß der Beschreibung substituiert sein können; zur Bekämpfung von Schadpilzen, neue 4-Aminopyridine, Verfahren zur Herstellung dieser Verbindungen sowie sie enthaltende Mittel.
(EN)
The invention relates to the use of 4-aminopyrimidines of formula (I), in which R1 = H, halogen, cyano, alkyl, alkylhalide, alkenyl, alkinyl, cycloalkyl, alkoxy, alkoxyalkyl, benzyloxyalkyl, alkoxyalkenyl or alkoxyalkinyl, R2 = H, halogen, cyano, alkyl, alkylhalide, alkenyl, alkinyl, cycloalkyl, alkoxy, alkoxyalkyl and alkylthioalkyl, whereby the hydrocarbon chain in R1 and/or R2 can be substituted as given in the description, R1 and R2 can form, together with the carbon atom to which they are bonded, a 5-7-membered ring which can contain one to three same or different heteroatoms selected from the group O, N or S, R3 = H, halogen, cyano, hydroxy, mercapto, azido, alkyl, alkenyl, alkinyl, alkylhalide, -O-D, -S(O)m-D, ON=CRaRb, CRc=NORa, NRcN=CRaRb, NRaRb, NRcNRaRb, NORa, NRcC(=NRc')NRaRb, NRcC(=O)NRaRb, NRaCN,-NRaC(=O)Rc, NRaC(=NORc)Rc', OC(=O)Ra, C(=NORc)NRaRb, CRc(=NNRaRb), C(=O)NRaRb, C(=O)Ra, CO2Ra, C(=O)NRzRb, C(=O)-N-ORb, C(=S)-NRzRb, C(=NORa)NRzRb, C(=NRa)NRzRb, C(=O)NRa-NRzRb, C(=N-NRzRc)NRaRb, C(=NORb)Ra, C(=N-NRzRb)Ra, CRaRb-ORz, CRaRb-NRzRc, ON(=CRaRb), NRa(C(=O)Rb), NRa(C(=O)ORb), NRa(C(=O)-NRzRb), NRa(C(=NRc)Rb), NRa(N=CRcRb), NRa-NRzRb, -NRz-ORa, NRa(C(=NRc)-NRzRb), NRa(C(=NORc)Rb), D = alkyl, alkenyl, alkinyl, alkylhalide, cycloalkyl, five- or six-membered saturated, partly-unsaturated or aromatic mono- or bi-cyclic heterocycles, containing one to four heteroatoms from the group O, N or S, one of the groups G1 or G2, whereby m, x, Ra, Rb, Rc, Rd, Re, Rz, Y, Z are as defined in the description and the aliphatic, alicyclic or aromatic groups R3, Ra, Rb, Rc, Rd or Re can be substituted as given in the description for the prevention of fungal pests, novel 4-aminopyridines, method for production of said compounds and agents comprising the same.
(FR)
L'invention concerne l'utilisation de 4-aminopyrimidines de formule (I), dans laquelle les substituants ont la signification suivante : R1 = hydrogène, halogène, cyano, alkyle, halogénoalkyle, alcényle, alcinyle, cycloalkyle, alcoxy, alcoxyalkyle, benzyloxyalkyle, alcoxyalcényle ou alcoxyalcinyle ; R2 = hydrogène, halogène, cyano, alkyle, halogénoalkyle, alcényle, alcinyle, cycloalkyle, alcoxy, alcoxyalkyle et alkylthioalkyle, les chaînes carbonées dans R1 et/ou R2 selon la description pouvant être substituées, R1 et R2 pouvant être former conjointement avec les atomes de carbone, auxquels ces éléments sont liés, un cycle de cinq à sept chaînons pouvant contenir un à trois hétéroatomes identiques ou différents du groupe O, N ou S ; R3 = hydrogène, halogène, cyano, hydroxy, mercapto, azido, alkyle, alcényle, alcinyle, halogénoalkyle, -O-D, -S(O)m-D, ON=CRaRb, CRc=NORa, NRcN=CRaRb, NRaRb, NRcNRaRb, NORa, NRcC(=NRc')NRaRb, NRcC(=O)NRaRb, NRaCN,-NRaC(=O)Rc, NRaC(=NORc)Rc', OC(=O)Ra, C(=NORc)NRaRb, CRc(=NNRaRb), C(=O)NRaRb, C(=O)Ra, CO2Ra, C(=O)NRzRb, C(=O)-N-ORb, C(=S)-NRzRb, C(=NORa)NRzRb, C(=NRa)NRzRb, C(=O)NRa-NRzRb, C(=N-NRzRc)NRaRb, C(=NORb)Ra, C(=N-NRzRb)Ra, CRaRb-ORz, CRaRb-NRzRc, ON(=CRaRb), NRa(C(=O)Rb), NRa(C(=O)ORb), NRa(C(=O)-NRzRb), NRa(C(=NRc)Rb), NRa(N=CRcRb), NRa-NRzRb, -NRz-ORa, NRa(C(=NRc)-NRzRb), NRa(C(=NORc)Rb), D alkyle, alcényle, alcinyle, halogénoalkyle, cyclalkyle, des hétérocycles mono ou bicycliques de cinq à six chaînons saturés, partiellement insaturés ou aromatiques, contenant un à quatre hétéroatomes du groupe O, N ou S, un des groupes G1 ou G2, m, x, Ra, Rb, Rc, Rd, Re, Rz, Y, Z étant définis dans la description et les groupes aliphatiques, alicycliques ou aromatiques R3, Ra,Rb,Rc, Rd ou Re selon la description pouvant être substitués, dans la lutte contre les champignons parasites, de nouvelles 4-aminopyridines, des procédés de production desdits composés ainsi que des agents contenant ces dernier.
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