WO2006050843 AMINOQUINAZOLINES COMPOUNDS

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Publication Number WO/2006/050843

Publication Date 18.05.2006

International Application No. PCT/EP2005/011682

International Filing Date 02.11.2005

Chapter 2 Demand Filed 28.04.2006

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Applicants

F. HOFFMANN-LA ROCHE AG [CH]/[CH] (AllExceptUS)
BERTHEL, Steven, Joseph [US]/[US] (UsOnly)
CHEUNG, Adrian, Wai-Hing [CN]/[US] (UsOnly)
THAKKAR, Kshitij, Chhabilbhai [IN]/[US] (UsOnly)
YUN, Weiya [CN]/[US] (UsOnly)

Inventors

BERTHEL, Steven, Joseph
CHEUNG, Adrian, Wai-Hing
THAKKAR, Kshitij, Chhabilbhai
YUN, Weiya

Agents

SALUD, Carlos

Priority Data

60/626,288		09.11.2004		US
60/715,260		08.09.2005		US

Publication Language English (en)

Filing Language English (EN)

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Title

(EN) AMINOQUINAZOLINES COMPOUNDS

(FR) COMPOSES AMINOQUINAZOLINES

Abstract

(EN) The present invention is concerned with compounds of formula (1), wherein R¹, R²and X are as defined in the description and claims. The compounds of the present invention are PTP-1B inhibitors and can be used as medicaments.

(FR) La présente invention concerne des composés de formule (1), dans laquelle R¹, R²et X sont tels que définis dans le descriptif et les revendications. Les composés de l'invention sont des inhibiteurs de PTP-1B et peuvent être utilisés comme médicaments.

C	CHEMISTRY; METALLURGY
07	ORGANIC CHEMISTRY
D	HETEROCYCLIC COMPOUNDS
239	Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
02	not condensed with other rings
24	having three or more double bonds between ring members or between ring members and non-ring members
28	with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
32	One oxygen, sulfur or nitrogen atom
42	One nitrogen atom

A	HUMAN NECESSITIES
61	MEDICAL OR VETERINARY SCIENCE; HYGIENE
K	PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31	Medicinal preparations containing organic active ingredients
33	Heterocyclic compounds
395	having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
495	having six-membered rings with two nitrogen atoms as the only ring hetero atoms, e.g. piperazine
505	Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
517	ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine

C	CHEMISTRY; METALLURGY
07	ORGANIC CHEMISTRY
D	HETEROCYCLIC COMPOUNDS
239	Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
02	not condensed with other rings
24	having three or more double bonds between ring members or between ring members and non-ring members
28	with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
32	One oxygen, sulfur or nitrogen atom
42	One nitrogen atom

A	HUMAN NECESSITIES
61	MEDICAL OR VETERINARY SCIENCE; HYGIENE
K	PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31	Medicinal preparations containing organic active ingredients
33	Heterocyclic compounds
395	having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
495	having six-membered rings with two nitrogen atoms as the only ring hetero atoms, e.g. piperazine
505	Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
517	ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine

A	HUMAN NECESSITIES
61	MEDICAL OR VETERINARY SCIENCE; HYGIENE
P	SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
3	Drugs for disorders of the metabolism
04	Anorexiants; Antiobesity agents

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1. WO2006050843 - AMINOQUINAZOLINES COMPOUNDS