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1. (WO2006012502) FORMULATION OF INSOLUBLE SMALL MOLECULE THERAPEUTICS IN LIPID-BASED CARRIERS
Latest bibliographic data on file with the International Bureau   

Pub. No.: WO/2006/012502 International Application No.: PCT/US2005/026020
Publication Date: 02.02.2006 International Filing Date: 22.07.2005
IPC:
A61K 31/506 (2006.01) ,A61P 35/00 (2006.01)
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
33
Heterocyclic compounds
395
having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
495
having six-membered rings with two nitrogen atoms as the only ring hetero atoms, e.g. piperazine
505
Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
506
not condensed and containing further heterocyclic rings
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
P
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
35
Antineoplastic agents
Applicants: PARMAR, Manjeet[CA/US]; US (UsOnly)
RIGEL PHARMACEUTICALS, INC.[US/US]; 1180 Veterans. Blvd. South San Francsico, CA 94080, US (AllExceptUS)
Inventors: PARMAR, Manjeet; US
Agent: PEASE, Ann, M., Caviani; Dechert LLP P.O. Box 10004 Palo Alto, CA 94303-0961, US
Priority Data:
60/590,78923.07.2004US
Title (EN) FORMULATION OF INSOLUBLE SMALL MOLECULE THERAPEUTICS IN LIPID-BASED CARRIERS
(FR) PREPARATION D'AGENTS THERAPEUTIQUES A PETITES MOLECULES INSOLUBLES DANS DES EXCIPIENTS LIPIDIQUES
Abstract:
(EN) The present invention provides formulations containing at least one unsaturated amphiphilic lipid and an amphipathic or hydrophobic drug and methods of making these formulations. In particular, the present invention provides formulations of least one unsaturated phospholipid and an amphipathic or hydrophobic pyrimidine drug, methods of making these formulations and the use of such formulations in a variety of contexts, including, for example, the treatment of proliferative disorders, such as tumors and cancers.
(FR) La présente invention concerne des préparations contenant au moins un lipide amphiphile insaturé et une substance thérapeutique amphipathique ou hydrophobe, ainsi que des méthodes destinées à la fabrication de ces préparations. La présente invention concerne plus précisément des préparations contenant au moins un phospholipide insaturé et une substance thérapeutique pyrimidique amphipathique ou hydrophobe, ainsi que des méthodes destinées à la fabrication de ces préparations et à leur utilisation dans divers contextes, y compris, sans en exclure d'autres, dans le traitement des tumeurs et des maladies évolutives, telles que les cancers.
Designated States: AE, AG, AL, AM, AT, AU, AZ, BA, BB, BG, BR, BW, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DE, DK, DM, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KP, KR, KZ, LC, LK, LR, LS, LT, LU, LV, MA, MD, MG, MK, MN, MW, MX, MZ, NA, NG, NI, NO, NZ, OM, PG, PH, PL, PT, RO, RU, SC, SD, SE, SG, SK, SL, SM, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, YU, ZA, ZM, ZW
African Regional Intellectual Property Organization (ARIPO) (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Office (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (EPO) (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HU, IE, IS, IT, LT, LU, LV, MC, NL, PL, PT, RO, SE, SI, SK, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG)
Publication Language: English (EN)
Filing Language: English (EN)