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Machine translation
1. (WO2006012395) PEPTIDASE INHIBITORS
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2006/012395    International Application No.:    PCT/US2005/025837
Publication Date: 02.02.2006 International Filing Date: 21.07.2005
IPC:
C07D 207/09 (2006.01), C07D 207/10 (2006.01), A61K 31/4025 (2006.01)
Applicants: ROYALTY, Susan Marie [US/US]; (US).
BURNS, James Ford [US/US]; (US).
SCICINSKI, Jan Jozef [GB/US]; (US).
JAGDMANN, JR., Gunnar Erik [US/US]; (US).
FOGLESONG, Robert James [US/US]; (US).
GRIFFIN, Kellee Renee [US/US]; (US).
DYAKONOV, Tatyana [US/US]; (US).
MIDDLEMISS, David [GB/GB]; (GB)
Inventors: ROYALTY, Susan Marie; (US).
BURNS, James Ford; (US).
SCICINSKI, Jan Jozef; (US).
JAGDMANN, JR., Gunnar Erik; (US).
FOGLESONG, Robert James; (US).
GRIFFIN, Kellee Renee; (US).
DYAKONOV, Tatyana; (US).
MIDDLEMISS, David; (GB)
Agent: MYERS BIGEL SIBLEY & SAJOVEC, P.A.; P.O. Box 37428, Raleigh, North Carolina 27627 (US)
Priority Data:
60/590,541 23.07.2004 US
60/634,362 08.12.2004 US
Title (EN) PEPTIDASE INHIBITORS
(FR) INHIBITEURS DE PEPTIDASE
Abstract: front page image
(EN)The present invention relates to a series of novel compounds having the formula (I) wherein: X is NR3 or O; n is 1 or 2; A is a bicyclic carbocycle and R1 and R2 are as described herein. The compounds are useful as DPP-IV inhibitors, such as for the treatment of diabetes.
(FR)La présente invention concerne une série de nouveaux composés ayant la formule (I) dans laquelle: X représente NR3 ou O; n représente 1 ou 2; A représente un carbocycle bicyclique et R1 ainsi que R2 ont la notation définie dans la description. Les composés sont utiles en tant qu'inhibiteurs de DPP-IV, par exemple dans le traitement du diabète.
Designated States: AE, AG, AL, AM, AT, AU, AZ, BA, BB, BG, BR, BW, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DE, DK, DM, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KP, KR, KZ, LC, LK, LR, LS, LT, LU, LV, MA, MD, MG, MK, MN, MW, MX, MZ, NA, NG, NI, NO, NZ, OM, PG, PH, PL, PT, RO, RU, SC, SD, SE, SG, SK, SL, SM, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, YU, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HU, IE, IS, IT, LT, LU, LV, MC, NL, PL, PT, RO, SE, SI, SK, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: English (EN)
Filing Language: English (EN)