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Machine translation
1. (WO2005121152) SUBSTITUTED TRIAZOLE DERIVATIVES AS OXYTOCIN ANTAGONISTS
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2005/121152    International Application No.:    PCT/IB2005/001541
Publication Date: 22.12.2005 International Filing Date: 27.05.2005
Chapter 2 Demand Filed:    01.09.2005    
IPC:
C07D 498/04 (2006.01), C07D 498/14 (2006.01), C07D 471/14 (2006.01), A61K 31/551 (2006.01), A61K 31/553 (2006.01), A61P 15/00 (2006.01)
Applicants: PFIZER LIMITED [GB/GB]; Ramsgate Road, Sandwich, Kent CT13 9NJ (GB) (GB only).
BROWN, Alan, Daniel [GB/GB]; (GB) (For US Only).
CALABRESE, Andrew, Antony [GB/GB]; (GB) (For US Only).
ELLIS, David [GB/GB]; (GB) (For US Only).
WATSON, Lesa [GB/GB]; (GB) (For US Only).
PFIZER INC. [US/US]; 235 East 42nd Street, New York, NY 10017 (US) (AE, AG, AL, AM, AT, AU, AZ, BA, BB, BE, BF, BG, BJ, BR, BW, BY, BZ, CA, CF, CG, CH, CI, CM, CN, CO, CR, CU, CY, CZ, DE, DK, DM, DZ, EC, EE, EG, ES, FI, FR, GA, GD, GE, GH, GM, GN, GQ, GR, GW, HR, HU, ID, IE, IL, IN, IS, IT, JP, KE, KG, KM, KP, KR, KZ, LC, LK, LR, LS, LT, LU, LV, MA, MC, MD, MG, MK, ML, MN, MR, MW, MX, MZ, NA, NE, NG, NI, NL, NO, NZ, OM, PG, PH, PL, PT, RO, RU, SC, SD, SE, SG, SI, SK, SL, SM, SN, SY, SZ, TD, TG, TJ, TM, TN, TR, TT, TZ, UA, UG, UZ, VC, VN, YU, ZA, ZM, ZW only)
Inventors: BROWN, Alan, Daniel; (GB).
CALABRESE, Andrew, Antony; (GB).
ELLIS, David; (GB).
WATSON, Lesa; (GB)
Agent: RUDDOCK, Keith, S.; Pfizer Research and Development, Ramsgate Road, Sandwich, Kent CT13 9NJ (GB)
Priority Data:
0412874.0 09.06.2004 GB
60/588,170 14.07.2004 US
Title (EN) SUBSTITUTED TRIAZOLE DERIVATIVES AS OXYTOCIN ANTAGONISTS
(FR) DERIVES TRIAZOLE SUBSTITUES UTILISES EN TANT QU'ANTAGONISTES DE L'OXYTOCINE
Abstract: front page image
(EN)This invention relates to compounds of formula (I) with activity as oxytocin antagonists, uses thereof, processes for the preparation thereof and compositions containing said inhibitors. These inhibitors have utility in a variety of therapeutic areas including sexual dysfunction, particularly premature ejaculation (P.E.).
(FR)La présente invention concerne des composés représentés par la formule (I) qui sont actifs en tant qu'antagonistes de l'oxytocine, les utilisations de ces derniers et des procédés de préparation de ces composés ainsi que des compositions contenant lesdits inhibiteurs. Ces inhibiteurs sont utiles dans divers domaines thérapeutiques tels que la dysfonction sexuelle, notamment l'éjaculation prématurée (EP). Formule (I)
Designated States: AE, AG, AL, AM, AT, AU, AZ, BA, BB, BG, BR, BW, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DE, DK, DM, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KP, KR, KZ, LC, LK, LR, LS, LT, LU, LV, MA, MD, MG, MK, MN, MW, MX, MZ, NA, NG, NI, NO, NZ, OM, PG, PH, PL, PT, RO, RU, SC, SD, SE, SG, SK, SL, SM, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, YU, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HU, IE, IS, IT, LT, LU, MC, NL, PL, PT, RO, SE, SI, SK, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: English (EN)
Filing Language: English (EN)