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Machine translation
1. (WO2005121096) A MULTICORE INDAZOLINONE LIBRARY
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2005/121096    International Application No.:    PCT/GB2005/002230
Publication Date: 22.12.2005 International Filing Date: 08.06.2005
IPC:
C07D 231/00 (2006.01)
Applicants: THE UNIVERSITY COURT OF THE UNIVERSITY OF ST ANDREWS [GB/GB]; College Gate, North Street, St Andrews, Fife KY16 9AJ (GB) (For All Designated States Except US).
WESTWOOD, Nicholas, James [GB/GB]; (GB) (For US Only).
ISAMBERT, Nicolas, Stanislas, Jean [FR/GB]; (GB) (For US Only)
Inventors: WESTWOOD, Nicholas, James; (GB).
ISAMBERT, Nicolas, Stanislas, Jean; (GB)
Agent: MURGITROYD & COMPANY; Scotland House, 165-169 Scotland Street, Glasgow G5 8PL (GB)
Priority Data:
0412741.1 08.06.2004 GB
Title (EN) A MULTICORE INDAZOLINONE LIBRARY
(FR) BANQUE DE COMPOSES CHIMIQUES A NOYAUX MULTIPLES
Abstract: front page image
(EN)There is provided a method to convert O-functionalized indazolinone-derivatives to the corresponding N2-functinoalised indazolinone derivatives, by use of microwave energy or a transition metal catalyst. A preferred catalyst is palladium tetrakis. The method described allows the creation of a library of chemical compounds which can be screened for biological activity.
(FR)L'invention concerne un procédé qui permet de convertir des dérivés d'indazolinone O-fonctionalisés en dérivés d'indazolinone N2-fonctionalisés correspondants, au moyen d'énergie produite par des micro-ondes ou d'un catalyseur métallique de transition. A titre de catalyseur préféré, on peut citer le tétrakis palladium. Ledit procédé permet de créer une banque de composés chimiques qui peuvent être criblés pour leur activité biologique.
Designated States: AE, AG, AL, AM, AT, AU, AZ, BA, BB, BG, BR, BW, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DE, DK, DM, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KP, KR, KZ, LC, LK, LR, LS, LT, LU, LV, MA, MD, MG, MK, MN, MW, MX, MZ, NA, NG, NI, NO, NZ, OM, PG, PH, PL, PT, RO, RU, SC, SD, SE, SG, SK, SL, SM, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, YU, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HU, IE, IS, IT, LT, LU, MC, NL, PL, PT, RO, SE, SI, SK, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: English (EN)
Filing Language: English (EN)