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1. (WO2005118593) BICYCLIC HETEROCYCLES AS HIV INTEGRASE INHIBITORS
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2005/118593    International Application No.:    PCT/US2005/016473
Publication Date: 15.12.2005 International Filing Date: 12.05.2005
IPC:
C07D 498/04 (2006.01), A61K 31/519 (2006.01), A61P 31/18 (2006.01)
Applicants: BRISTOL-MYERS SQUIBB COMPANY [US/US]; Route 206 and Province Line Road, Princeton, NJ 08543-4000 (US) (For All Designated States Except US).
NAIDU, B., Narasimhulu [IN/US]; (US) (For US Only).
BANVILLE, Jacques [CA/CA]; (CA) (For US Only).
BEAULIEU, Francis [CA/CA]; (CA) (For US Only).
CONNOLLY, Timothy, P. [CA/US]; (US) (For US Only).
KRYSTAL, Mark, R. [US/US]; (US) (For US Only).
MATISKELLA, John, D. [US/US]; (US) (For US Only).
OUELLET, Carl [CA/CA]; (CA) (For US Only).
PLAMONDON, Serge [CA/CA]; (CA) (For US Only).
REMILLARD, Roger [CA/CA]; (CA) (For US Only).
SORENSON, Margaret, E. [US/US]; (US) (For US Only).
UEDA, Yasutsugu [JP/US]; (US) (For US Only).
WALKER, Michael, A. [US/US]; (US) (For US Only)
Inventors: NAIDU, B., Narasimhulu; (US).
BANVILLE, Jacques; (CA).
BEAULIEU, Francis; (CA).
CONNOLLY, Timothy, P.; (US).
KRYSTAL, Mark, R.; (US).
MATISKELLA, John, D.; (US).
OUELLET, Carl; (CA).
PLAMONDON, Serge; (CA).
REMILLARD, Roger; (CA).
SORENSON, Margaret, E.; (US).
UEDA, Yasutsugu; (US).
WALKER, Michael, A.; (US)
Agent: EPPERSON, James; Bristol-Myers Squibb Company, P.O. Box 4000, Princeton, NJ 08543-4000 (US)
Priority Data:
60/575,513 28.05.2004 US
60/603,371 20.08.2004 US
11/126,891 11.05.2005 US
Title (EN) BICYCLIC HETEROCYCLES AS HIV INTEGRASE INHIBITORS
(FR) HETEROCYCLES BICYCLIQUES SERVANT D'INHIBITEURS D'INTEGRASE DU VIH
Abstract: front page image
(EN)The invention encompasses a series cyclic bicyclic pyrimidinone compounds of Formula I which inhibit HIV integrase and prevent viral integration into human DNA. This action makes the compounds useful for treating HIV infection and AIDS. The invention also encompasses pharmaceutical compositions and methods for treating those infected with HIV.
(FR)La présente invention concerne une série de composés de pyrimidinone bicycliques cycliques de formule (I) qui inhibent l'intégrase de VIH et qui empêchent une intégration virale dans l'ADN humain. Ces composés sont par conséquent utilisés pour traiter une infection à VIH et le SIDA. Cette invention concerne également des compositions pharmaceutiques et des procédés pour traiter les personnes infectées par le VIH.
Designated States: AE, AG, AL, AM, AT, AU, AZ, BA, BB, BG, BR, BW, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DE, DK, DM, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KP, KR, KZ, LC, LK, LR, LS, LT, LU, LV, MA, MD, MG, MK, MN, MW, MX, MZ, NA, NG, NI, NO, NZ, OM, PG, PH, PL, PT, RO, RU, SC, SD, SE, SG, SK, SL, SM, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, YU, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HU, IE, IS, IT, LT, LU, MC, NL, PL, PT, RO, SE, SI, SK, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: English (EN)
Filing Language: English (EN)