WIPO logo
Mobile | Deutsch | Español | Français | 日本語 | 한국어 | Português | Русский | 中文 | العربية |
PATENTSCOPE

Search International and National Patent Collections
World Intellectual Property Organization
Search
 
Browse
 
Translate
 
Options
 
News
 
Login
 
Help
 
Machine translation
1. (WO2005113576) AMINOSULPHONYL- OR AMINOSULPHONYLAMINO-SUBSTITUTED PHENYL ESTERS AS ESTRIOL AND ESTETROL PRODRUGS
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2005/113576    International Application No.:    PCT/EP2005/005258
Publication Date: 01.12.2005 International Filing Date: 10.05.2005
IPC:
C07J 41/00 (2006.01), A61K 31/565 (2006.01), A61P 5/30 (2006.01)
Applicants: SCHERING AKTIENGESELLSCHAFT [DE/DE]; Müllerstrasse 178, 13353 Berlin (DE) (For All Designated States Except US).
WYRWA, Ralf [DE/DE]; (DE) (For US Only).
DROESCHER, Peter [DE/DE]; (DE) (For US Only).
RING, Sven [DE/DE]; (DE) (For US Only).
ELGER, Walter [DE/DE]; (DE) (For US Only).
SCHNEIDER, Birgitt [DE/DE]; (DE) (For US Only).
HILLISCH, Alexander [AT/DE]; (DE) (For US Only).
REDDERSEN, Gudrun [DE/DE]; (DE) (For US Only)
Inventors: WYRWA, Ralf; (DE).
DROESCHER, Peter; (DE).
RING, Sven; (DE).
ELGER, Walter; (DE).
SCHNEIDER, Birgitt; (DE).
HILLISCH, Alexander; (DE).
REDDERSEN, Gudrun; (DE)
Priority Data:
10 2004 025 985.2 21.05.2004 DE
Title (DE) AMINOSULFONYL- ODER AMINOSULFONYLAMINO-SUBSTITUIERTE PHENYL-ESTER ALS ESTRIOL-UND ESTETROL-PRODRUGS
(EN) AMINOSULPHONYL- OR AMINOSULPHONYLAMINO-SUBSTITUTED PHENYL ESTERS AS ESTRIOL AND ESTETROL PRODRUGS
(FR) PHENYLESTER SUBSTITUE PAR AMINOSULFONYLE OU AMINOSULFONYLAMINO COMME PROMEDICAMENTS A BASE D'OESTRIOL ET D'OESTETROL
Abstract: front page image
(DE)Die vorliegende Erfindung stellt Estriol- und Estetrol-Prodrugs der allgemeinen Formel (I) bereit, in denen die Gruppe Y an das Steroid gebunden ist, Verfahren zu deren Herstellung, pharmazeutische Zusammensetzungen, die diese Verbindungen enthalten, sowie deren Verwendung zur Herstellung von Arzneimitteln mit estrogener Wirkung.
(EN)The invention relates to estriol and estetrol prodrugs of general formula (I), in which group Y is bonded to the steroid, the method for production thereof, pharmaceutical compositions comprising said compounds and the use thereof for production of medicaments with estrogenic effect.
(FR)La présente invention concerne des promédicaments à base d'oestriol et d'oestétrol de formule générale (I), dans lesquels le groupe Y est lié au stéroïde, un procédé de production desdits promédicaments, des compositions pharmaceutiques contenant ces composés ainsi que leur utilisation dans la production de médicaments à effet oestrogène.
Designated States: AE, AG, AL, AM, AT, AU, AZ, BA, BB, BG, BR, BW, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DK, DM, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KP, KR, KZ, LC, LK, LR, LS, LT, LU, LV, MA, MD, MG, MK, MN, MW, MX, MZ, NA, NG, NI, NO, NZ, OM, PG, PH, PL, PT, RO, RU, SC, SD, SE, SG, SK, SL, SM, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, YU, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HU, IE, IS, IT, LT, LU, MC, NL, PL, PT, RO, SE, SI, SK, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: German (DE)
Filing Language: German (DE)