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1. (WO2005100302) SOLID STATE FORMS OF (-)-(1R,2S)-2-AMINO-4-METHYLENE-CYCLOPENTANECARBOXYLIC ACID
Latest bibliographic data on file with the International Bureau   
Pub. No.: WO/2005/100302 International Application No.: PCT/IB2005/000971
Publication Date: 27.10.2005 International Filing Date: 13.04.2005
IPC:
C07C 227/42 (2006.01) ,C07C 229/48 (2006.01)
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
C
ACYCLIC OR CARBOCYCLIC COMPOUNDS
227
Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
38
Separation; Purification; Stabilisation; Use of additives
40
Separation; Purification
42
Crystallisation
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
C
ACYCLIC OR CARBOCYCLIC COMPOUNDS
229
Compounds containing amino and carboxyl groups bound to the same carbon skeleton
46
having amino or carboxyl groups bound to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton
48
with amino groups and carboxyl groups bound to carbon atoms of the same non-condensed ring
Applicants:
ZEGARAC, Miroslav [HR/HR]; HR (UsOnly)
MESTROVIC, Ernest [HR/HR]; HR (UsOnly)
HULITA, Nada, Kosutic [HR/HR]; HR (UsOnly)
FILIC, Darko [HR/HR]; HR (UsOnly)
DUMIC, Miljenko [HR/HR]; HR (UsOnly)
GRUNENBERG, Alfons [DE/DE]; DE (UsOnly)
KEIL, Brigit [DE/DE]; DE (UsOnly)
CERIC, Helena [HR/HR]; HR (UsOnly)
GLAXOSMITHKLINE ISTRAZIVACKI CENTAR ZAGREB D.O.O. [HR/HR]; Prilaz baruna Filipovica 29 10000 Zagreb, HR (AllExceptUS)
BAYER HEALTHCARE AG [DE/DE]; 51368 Leverkusen, DE (AllExceptUS)
Inventors:
ZEGARAC, Miroslav; HR
MESTROVIC, Ernest; HR
HULITA, Nada, Kosutic; HR
FILIC, Darko; HR
DUMIC, Miljenko; HR
GRUNENBERG, Alfons; DE
KEIL, Brigit; DE
CERIC, Helena; HR
Priority Data:
60/563,26516.04.2004US
60/608,17607.09.2004US
Title (EN) SOLID STATE FORMS OF (-)-(1R,2S)-2-AMINO-4-METHYLENE-CYCLOPENTANECARBOXYLIC ACID
(FR) FORMES A L'ETAT SOLIDE D'ACIDE (-)-(1R,1S)-2-AMINO-4-METHYLENE-CYCLOPENTANECARBOXYLIQUE
Abstract:
(EN) The present invention relates to the solid state forms &agr;, &bgr;, &dgr;, ϵ, and &zgr; of (-)-(1R,1S)-2-amino-4-methylene-cyclopentanecarboxylic acid, to the processes for their preparation, to pharmaceutical compositions containing the said solid state forms of (-)-(1R,1S)-2-amino-methylene-cyclopentanecarboxylic acid as the active ingredients as well as to a method of treatment using the same.
(FR) L'invention concerne des formes à l'état solide ?, ?, ?, e, et ? d'acide (-)-(1R,1S)-2-amino-4-méthylène-cyclopentanecarboxylique, leurs procédés de préparation, des compositions pharmaceutiques contenant les formes à l'état solide d'acide (-)-(1R,1S)-2-amino-méthylène-cyclopentanecarboxylique en tant que principes actifs ainsi qu'une méthode de traitement utilisant lesdites formes à l'état solide.
Designated States: AE, AG, AL, AM, AT, AU, AZ, BA, BB, BG, BR, BW, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DE, DK, DM, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KP, KR, KZ, LC, LK, LR, LS, LT, LU, LV, MA, MD, MG, MK, MN, MW, MX, MZ, NA, NI, NO, NZ, OM, PG, PH, PL, PT, RO, RU, SC, SD, SE, SG, SK, SL, SM, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, YU, ZA, ZM, ZW
African Regional Intellectual Property Organization (ARIPO) (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Office (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (EPO) (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HU, IE, IS, IT, LT, LU, MC, NL, PL, PT, RO, SE, SI, SK, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG)
Publication Language: English (EN)
Filing Language: English (EN)