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1. WO2005100302 - SOLID STATE FORMS OF (-)-(1R,2S)-2-AMINO-4-METHYLENE-CYCLOPENTANECARBOXYLIC ACID

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Publication Number WO/2005/100302
Publication Date 27.10.2005
International Application No. PCT/IB2005/000971
International Filing Date 13.04.2005
IPC
C07C 227/42 2006.1
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
CACYCLIC OR CARBOCYCLIC COMPOUNDS
227Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
38Separation; Purification; Stabilisation; Use of additives
40Separation; Purification
42Crystallisation
C07C 229/48 2006.1
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
CACYCLIC OR CARBOCYCLIC COMPOUNDS
229Compounds containing amino and carboxyl groups bound to the same carbon skeleton
46having amino or carboxyl groups bound to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton
48with amino groups and carboxyl groups bound to carbon atoms of the same non-condensed ring
CPC
A61P 31/10
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
31Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
10Antimycotics
C07C 227/42
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
CACYCLIC OR CARBOCYCLIC COMPOUNDS
227Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
38Separation; Purification; Stabilisation; Use of additives
40Separation; Purification
42Crystallisation
C07C 229/48
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
CACYCLIC OR CARBOCYCLIC COMPOUNDS
229Compounds containing amino and carboxyl groups bound to the same carbon skeleton
46having amino or carboxyl groups bound to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton
48with amino groups and carboxyl groups bound to carbon atoms of the same non-condensed ring
C07C 2601/08
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
CACYCLIC OR CARBOCYCLIC COMPOUNDS
2601Systems containing only non-condensed rings
06with a five-membered ring
08the ring being saturated
Applicants
  • GLAXOSMITHKLINE ISTRAZIVACKI CENTAR ZAGREB D.O.O. [HR]/[HR] (AllExceptUS)
  • BAYER HEALTHCARE AG [DE]/[DE] (AllExceptUS)
  • ZEGARAC, Miroslav [HR]/[HR] (UsOnly)
  • MESTROVIC, Ernest [HR]/[HR] (UsOnly)
  • HULITA, Nada, Kosutic [HR]/[HR] (UsOnly)
  • FILIC, Darko [HR]/[HR] (UsOnly)
  • DUMIC, Miljenko [HR]/[HR] (UsOnly)
  • GRUNENBERG, Alfons [DE]/[DE] (UsOnly)
  • KEIL, Brigit [DE]/[DE] (UsOnly)
  • CERIC, Helena [HR]/[HR] (UsOnly)
Inventors
  • ZEGARAC, Miroslav
  • MESTROVIC, Ernest
  • HULITA, Nada, Kosutic
  • FILIC, Darko
  • DUMIC, Miljenko
  • GRUNENBERG, Alfons
  • KEIL, Brigit
  • CERIC, Helena
Priority Data
60/563,26516.04.2004US
60/608,17607.09.2004US
Publication Language English (en)
Filing Language English (EN)
Designated States
Title
(EN) SOLID STATE FORMS OF (-)-(1R,2S)-2-AMINO-4-METHYLENE-CYCLOPENTANECARBOXYLIC ACID
(FR) FORMES A L'ETAT SOLIDE D'ACIDE (-)-(1R,1S)-2-AMINO-4-METHYLENE-CYCLOPENTANECARBOXYLIQUE
Abstract
(EN) The present invention relates to the solid state forms &agr;, &bgr;, &dgr;, ϵ, and &zgr; of (-)-(1R,1S)-2-amino-4-methylene-cyclopentanecarboxylic acid, to the processes for their preparation, to pharmaceutical compositions containing the said solid state forms of (-)-(1R,1S)-2-amino-methylene-cyclopentanecarboxylic acid as the active ingredients as well as to a method of treatment using the same.
(FR) L'invention concerne des formes à l'état solide ?, ?, ?, e, et ? d'acide (-)-(1R,1S)-2-amino-4-méthylène-cyclopentanecarboxylique, leurs procédés de préparation, des compositions pharmaceutiques contenant les formes à l'état solide d'acide (-)-(1R,1S)-2-amino-méthylène-cyclopentanecarboxylique en tant que principes actifs ainsi qu'une méthode de traitement utilisant lesdites formes à l'état solide.
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