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1. WO2005095404 - 6-(2-FLUOROPHENYL)-TRIAZOLOPYRIMIDINES, METHOD FOR PRODUCING THEM, THEIR USE FOR CONTROLLING PARASITIC FUNGI AND AGENTS CONTAINING THE SAME

Publication Number WO/2005/095404
Publication Date 13.10.2005
International Application No. PCT/EP2005/003208
International Filing Date 26.03.2005
Chapter 2 Demand Filed 12.04.2006
IPC
C07D 487/04 2006.01
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
487Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/-C07D477/183
02in which the condensed system contains two hetero rings
04Ortho-condensed systems
A01N 43/90 2006.01
AHUMAN NECESSITIES
01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
43Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
90having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
CPC
A01N 43/90
AHUMAN NECESSITIES
01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES, AS HERBICIDES
43Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
90having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
C07D 487/04
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
487Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by C07D451/00 - C07D477/00
02in which the condensed system contains two hetero rings
04Ortho-condensed systems
Applicants
  • BASF AKTIENGESELLSCHAFT [DE]/[DE] (AllExceptUS)
  • BLETTNER, Carsten [DE]/[DE] (UsOnly)
  • GEWEHR, Markus [DE]/[DE] (UsOnly)
  • GRAMMENOS, Wassilios [GR]/[DE] (UsOnly)
  • GROTE, Thomas [DE]/[DE] (UsOnly)
  • HÜNGER, Udo [DE]/[DE] (UsOnly)
  • MÜLLER, Bernd [DE]/[DE] (UsOnly)
  • NIEDENBRÜCK, Matthias [DE]/[DE] (UsOnly)
  • RHEINHEIMER, Joachim [DE]/[DE] (UsOnly)
  • SCHÄFER, Peter [DE]/[DE] (UsOnly)
  • SCHIEWECK, Frank [DE]/[DE] (UsOnly)
  • SCHWÖGLER, Anja [DE]/[DE] (UsOnly)
  • WAGNER, Oliver [DE]/[DE] (UsOnly)
  • RACK, Michael [DE]/[DE] (UsOnly)
  • NAVE, Barbara [AT]/[DE] (UsOnly)
  • SCHERER, Maria [DE]/[DE] (UsOnly)
  • STRATHMANN, Siegfried [DE]/[DE] (UsOnly)
  • SCHÖFL, Ulrich [DE]/[DE] (UsOnly)
  • STIERL, Reinhard [DE]/[DE] (UsOnly)
Inventors
  • BLETTNER, Carsten
  • GEWEHR, Markus
  • GRAMMENOS, Wassilios
  • GROTE, Thomas
  • HÜNGER, Udo
  • MÜLLER, Bernd
  • NIEDENBRÜCK, Matthias
  • RHEINHEIMER, Joachim
  • SCHÄFER, Peter
  • SCHIEWECK, Frank
  • SCHWÖGLER, Anja
  • WAGNER, Oliver
  • RACK, Michael
  • NAVE, Barbara
  • SCHERER, Maria
  • STRATHMANN, Siegfried
  • SCHÖFL, Ulrich
  • STIERL, Reinhard
Common Representative
  • BASF AKTIENGESELLSCHAFT
Priority Data
10 2004 016 082.130.03.2004DE
Publication Language German (DE)
Filing Language German (DE)
Designated States
Title
(DE) 6-(2-FLUORPHENYL)-TRIAZOLOPYRIMIDINE, VERFAHREN ZU IHRER HERSTELLUNG UND IHRE VERWENDUNG ZUR BEKÄMPFUNG VON SCHADPILZEN SOWIE SIE ENTHALTENDE MITTEL
(EN) 6-(2-FLUOROPHENYL)-TRIAZOLOPYRIMIDINES, METHOD FOR PRODUCING THEM, THEIR USE FOR CONTROLLING PARASITIC FUNGI AND AGENTS CONTAINING THE SAME
(FR) 6-(2-FLUOROPHENYL)-TRIAZOLOPYRIMIDINES, PROCEDE DE PRODUCTION DESDITS COMPOSES, LEUR UTILISATION DANS LA LUTTE CONTRE DES CHAMPIGNONS PARASITES ET DES AGENTS CONTENANT LESDITS COMPOSES
Abstract
(DE)
Die vorliegende Anmeldung offenbart 6-(2-Fluorphenyl)-triazolopyrimidine der Formel I in der die Substituenten folgende Bedeutung haben: R1C4-C8-Alkyl, C4-C8-Halogenalkyl, substituiertes C3-C8-Cycloalkyl, C3-C8- Halogencycloalkyl, C5-C8-Alkenyl, C2-C8-Halogenalkenyl, C3-C6-Cycloalkenyl, C3-C6-Halogencyclo­alkenyl, C2-C8-Alkinyl, C2-C8-Halogenalkinyl oder Phenyl, Naphthyl, oder ein fünf­oder sechsgliedriger gesättigter, partiell ungesättigter oder aromatischer Hetero­cyclus, enthaltend ein bis vier Heteroatome aus der Gruppe O, N oder S, R2 Wasserstoff, C1-C3-Alkyl oder eine der bei R1 genannten Gruppen, R1 und R2 können auch zusammen mit dem Stickstoffatom, an das sie gebunden sind, ein fünf- oder sechsgliedriges Heterocyclyl oder Heteroaryl bilden, welches über N gebunden ist und ein bis drei weitere Heteroatome aus der Gruppe O, N und S als Ringglied enthalten,wobei ggf. durch Methyigruppen substituiertes Piperidin-1-yl ausgenommen blei­bt; R1 und/oder R2 können gemäß der Beschreibung substituiert sein; L1 Chlor oder Fluor; L2 Wasserstoff,wenn L1 Fluor bedeutet, zusätzlich Fluor, X Alkyl. Desweiteren werden Verfahren zu ihrer Herstellung und ihre Verwendung zur Bekämpfung von Schadpilzen sowie die enthaltende Mittel offenbart.
(EN)
The invention relates to the 6-(2-fluorophenyl)-triazolopyrimidines of formula (I), wherein the substituents are defined as follows: R1 represents C4-C8 alkyl, C4-C8 halogen alkyl, substituted C3-C8 cycloalkyl, C3-C8 halogen cycloalkyl, C5-C8 alkenyl, C2-C8 halogen alkenyl, C3-C6 cycloalkenyl, C3-C6 halogen cycloalkenyl, C2-C8 alkinyl, C2-C8 halogen alkinyl or phenyl, naphthyl, or a five-membered or six-membered saturated, partially unsaturated or aromatic heterocycle comprising one to four heteroatoms from the group including O, N or S; R2 represents hydrogen, C1-C3 alkyl or one of the groups mentioned for R1, R1 and R2, together with the nitrogen atom to which they are bound, may form a five-membered or six-membered heterocyclyl or heteroaryl which is bound via N, and may contain one to three additional heteroatoms from the group including O, N and S as a ring member, whereby piperidino-1-yl which is optionally substituted by methyl groups is exempt; R1 and/or R2 may be substituted according to the description; L1 represents chlorine or fluorine; L2 represents hydrogen, if L1 represents fluorine, L2 additionally represents fluorine; X represents alkyl. The invention also relates to a method for producing the aforementioned compounds, to agents containing them and to their use for controlling phytopathogenic parasitic fungi.
(FR)
L'invention concerne des 6-(2-fluorophényl)-triazolopyrimidines de formule (I), dans laquelle les substituants ont la signification suivante : R1 = alkyle en C4-C8, halogénoalkyle en C4-C8, cycloalkyle en C3-C8 substitué, halogénocycloalkyle en C3-C8, alcényle en C5-C8, halogénoalcényle en C2-C8, cycloalcényle en C3-C6, halogénocycloalcényle en C3-C6, alcinyle en C2-C8, halogénoalcinyle en C2-C8 ou phényle, naphthyle ou un hétérocycle saturé, partiellement insaturé ou aromatique à cinq ou six chaînons, contenant un à quatre hétéroatomes du groupe O, N ou S ; R2 = hydrogène, alkyle en C1-C3 ou un des groupes mentionnés pour R1, R1 et R2 pouvant également former, conjointement avec l'atome d'azote auquel ces derniers sont liés, un hétéroaryle ou hétérocyclyle à cinq ou six chaînons, lié par l'intermédiaire de N et contenant un à trois autres hétéroatomes du groupe O, N et S comme chaînon cyclique, à l'exception de pipéridin-1-yle éventuellement substitué par des groupes méthyle, et R1 et/ou R2 pouvant être substitués selon la description ; L1 = chlore ou fluor ; L2 = hydrogène, si L1 signifie fluor, et fluor ; X = alkyle. Ladite invention concerne également un procédé pour produire ces composés, des agents contenant ces derniers ainsi que leur utilisation dans la lutte contre les champignons phytopathogènes.
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