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1. (WO2005030706) AMIDE TYPE CARBOXAMIDE DERIVATIVE
Latest bibliographic data on file with the International Bureau   

Pub. No.: WO/2005/030706 International Application No.: PCT/JP2004/013892
Publication Date: 07.04.2005 International Filing Date: 24.09.2004
Chapter 2 Demand Filed: 30.09.2004
IPC:
C07C 237/42 (2006.01) ,C07D 409/12 (2006.01)
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
C
ACYCLIC OR CARBOCYCLIC COMPOUNDS
237
Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups
28
having the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a non-condensed six-membered aromatic ring of the carbon skeleton
42
having nitrogen atoms of amino groups bound to the carbon skeleton of the acid part, further acylated
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
409
Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
02
containing two hetero rings
12
linked by a chain containing hetero atoms as chain links
Applicants: KAWAGUCHI, Takayuki[JP/JP]; JP (UsOnly)
AKATSUKA, Hidenori[JP/JP]; JP (UsOnly)
MORIMOTO, Masamichi[JP/JP]; JP (UsOnly)
WATANABE, Tatsuya[JP/JP]; JP (UsOnly)
IIJIMA, Toru[JP/JP]; JP (UsOnly)
MURAKAMI, Jun[JP/JP]; JP (UsOnly)
TANABE SEIYAKU CO., LTD.[JP/JP]; 2-10, Dosho-machi 3-chome, Chuo-ku Osaka-shi, Osaka 5418505, JP (AllExceptUS)
Inventors: KAWAGUCHI, Takayuki; JP
AKATSUKA, Hidenori; JP
MORIMOTO, Masamichi; JP
WATANABE, Tatsuya; JP
IIJIMA, Toru; JP
MURAKAMI, Jun; JP
Agent: KAWAMIYA, Osamu; Aoyama & Partners IMP Building 3-7, Shiromi 1-chome, Chuo-ku Osaka-shi, Osaka 5400001, JP
Priority Data:
2003-33459526.09.2003JP
Title (EN) AMIDE TYPE CARBOXAMIDE DERIVATIVE
(FR) DERIVE CARBOXAMIDE DU TYPE AMIDE
(JA) アミド型カルボキサミド誘導体
Abstract:
(EN) An amide type carboxamide derivative represented by the general formula [1]: [Chemical formula 1] (wherein X represents -N= or -CH=; R1 represents halogeno, lower alkyl, etc.; R2 represents, e.g., [Chemical formula 2] Y1 and Y2 are the same or different and each represents halogeno or a group selected among lower alkyls, lower alkoxys, etc.; and ring A represents phenyl, etc.) or a pharmacologically acceptable salt of the derivative. The derivative and salt are useful as a medicine, especially an FXa inhibitor.
(FR) L'invention concerne un dérivé carboxamide du type amide représenté par la formule (1) dans laquelle X représente N= ou CH=; R1 représente, entre autres, halogéno, alkyle inférieur; R2 représente par exemple (2), (Y1 et Y2 étant identiques ou différents et chacun représentant halogéno ou un groupe choisi parmi, entre autres, alkyles inférieurs, alcoxys inférieurs; et le cycle A représente, entre autres, phényle) ou un sel acceptable au plan pharmacologique dudit dérivé. Le dérivé et le sel de l'invention sont utiles en médecine, notamment en tant qu'inhibiteur du FXa.
(JA) not available
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Designated States: AE, AG, AL, AM, AT, AU, AZ, BA, BB, BG, BR, BW, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DE, DK, DM, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, HR, HU, ID, IL, IN, IS, JP, KE, KG, KP, KR, KZ, LC, LK, LR, LS, LT, LU, LV, MA, MD, MG, MK, MN, MW, MX, MZ, NA, NI, NO, NZ, OM, PG, PH, PL, PT, RO, RU, SC, SD, SE, SG, SK, SL, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, YU, ZA, ZM, ZW
African Regional Intellectual Property Organization (ARIPO) (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Office (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (EPO) (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HU, IE, IT, LU, MC, NL, PL, PT, RO, SE, SI, SK, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG)
Publication Language: Japanese (JA)
Filing Language: Japanese (JA)