WO2005021545 IMIDAZO[1,5-a]PYRIDINE OR IMIDAZO[1,5-a]PIPERIDINE DERIVATIVES AND THEIR USE FOR THE PREPARATION OF MEDICAMENT AGAINST 5-HT2A RECEPTOR-RELATED DISORDERS

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Publication Number WO/2005/021545

Publication Date 10.03.2005

International Application No. PCT/SE2004/001235

International Filing Date 27.08.2004

Chapter 2 Demand Filed 24.03.2005

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CPC

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Applicants

GALAPAGOS NV (AllExceptUS)
BERTHOLD, Malin [SE]/[SE] (UsOnly)
CROSSLEY, Roger [GB]/[GB] (UsOnly)
WARD, Terry [GB]/[GB] (UsOnly)

Inventors

BERTHOLD, Malin
CROSSLEY, Roger
WARD, Terry

Agents

BAKER-MUNTON, Nicola

Priority Data

0302368-6		03.09.2003		SE
60/505,337		23.09.2003		US

Publication Language English (en)

Filing Language English (EN)

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Title

(EN) IMIDAZO[1,5-a]PYRIDINE OR IMIDAZO[1,5-a]PIPERIDINE DERIVATIVES AND THEIR USE FOR THE PREPARATION OF MEDICAMENT AGAINST 5-HT2A RECEPTOR-RELATED DISORDERS

(FR) DERIVES D'IMIDAZO[1,5-A]PYRIDINE OU D'IMIDAZO[1,5-A]PIPERIDINE ET LEUR UTILISATION DANS LA PREPARATION D'UN MEDICAMENT DIRIGE CONTRE LES TROUBLES LIES AU RECEPTEUR 5-HT2A

Abstract

(EN) The present invention relates to compounds of Formula (I): wherein X, Y, Z, and R¹ are as described herein, processes for preparing the compounds, pharmaceutical compositions comprising the compounds, and use of the compounds and compositions in the prophylaxis or treatment of a 5-HT2A receptor-related disorder.

(FR) La présente invention concerne des composés correspondant à la formule (I): dans laquelle X, Y, Z, et R¹ sont décrits dans l'invention, des procédés de préparation de ces composés, des compositions pharmaceutiques les contenant et l'utilisation de ces composés et compositions dans la prévention ou le traitement des troubles liés au récepteur de 5-HT2A.

C	CHEMISTRY; METALLURGY
07	ORGANIC CHEMISTRY
D	HETEROCYCLIC COMPOUNDS
471	Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/-C07D463/251
02	in which the condensed system contains two hetero rings
04	Ortho-condensed systems

C	CHEMISTRY; METALLURGY
07	ORGANIC CHEMISTRY
D	HETEROCYCLIC COMPOUNDS
487	Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/-C07D477/183
02	in which the condensed system contains two hetero rings
04	Ortho-condensed systems

C	CHEMISTRY; METALLURGY
07	ORGANIC CHEMISTRY
D	HETEROCYCLIC COMPOUNDS
471	Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/-C07D463/251
02	in which the condensed system contains two hetero rings
04	Ortho-condensed systems

C	CHEMISTRY; METALLURGY
07	ORGANIC CHEMISTRY
D	HETEROCYCLIC COMPOUNDS
487	Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/-C07D477/183
02	in which the condensed system contains two hetero rings
04	Ortho-condensed systems

A	HUMAN NECESSITIES
61	MEDICAL OR VETERINARY SCIENCE; HYGIENE
P	SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
1	Drugs for disorders of the alimentary tract or the digestive system
14	Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents

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1. WO2005021545 - IMIDAZO[1,5-a]PYRIDINE OR IMIDAZO[1,5-a]PIPERIDINE DERIVATIVES AND THEIR USE FOR THE PREPARATION OF MEDICAMENT AGAINST 5-HT2A RECEPTOR-RELATED DISORDERS