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1. (WO2005021545) IMIDAZO[1,5-a]PYRIDINE OR IMIDAZO[1,5-a]PIPERIDINE DERIVATIVES AND THEIR USE FOR THE PREPARATION OF MEDICAMENT AGAINST 5-HT2A RECEPTOR-RELATED DISORDERS
Latest bibliographic data on file with the International Bureau   

Pub. No.: WO/2005/021545 International Application No.: PCT/SE2004/001235
Publication Date: 10.03.2005 International Filing Date: 27.08.2004
Chapter 2 Demand Filed: 24.03.2005
IPC:
C07D 471/04 (2006.01) ,C07D 487/04 (2006.01)
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
471
Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/-C07D463/251
02
in which the condensed system contains two hetero rings
04
Ortho-condensed systems
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
487
Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/-C07D477/183
02
in which the condensed system contains two hetero rings
04
Ortho-condensed systems
Applicants:
BERTHOLD, Malin [SE/SE]; SE (UsOnly)
CROSSLEY, Roger [GB/GB]; GB (UsOnly)
WARD, Terry [GB/GB]; GB (UsOnly)
GALAPAGOS NV; Gen. De Wittelaan L11 A3 2800 Mechelen, BE (AllExceptUS)
Inventors:
BERTHOLD, Malin; SE
CROSSLEY, Roger; GB
WARD, Terry; GB
Agent:
BAKER-MUNTON, Nicola; Stratagem IPM Ltd. Fosters Wing, Anstey Hall Maris Lane, Trumpington Cambridge CB2 2LG, GB
Priority Data:
0302368-603.09.2003SE
60/505,33723.09.2003US
Title (EN) IMIDAZO[1,5-a]PYRIDINE OR IMIDAZO[1,5-a]PIPERIDINE DERIVATIVES AND THEIR USE FOR THE PREPARATION OF MEDICAMENT AGAINST 5-HT2A RECEPTOR-RELATED DISORDERS
(FR) DERIVES D'IMIDAZO[1,5-A]PYRIDINE OU D'IMIDAZO[1,5-A]PIPERIDINE ET LEUR UTILISATION DANS LA PREPARATION D'UN MEDICAMENT DIRIGE CONTRE LES TROUBLES LIES AU RECEPTEUR 5-HT2A
Abstract:
(EN) The present invention relates to compounds of Formula (I): wherein X, Y, Z, and R1 are as described herein, processes for preparing the compounds, pharmaceutical compositions comprising the compounds, and use of the compounds and compositions in the prophylaxis or treatment of a 5-HT2A receptor-related disorder.
(FR) La présente invention concerne des composés correspondant à la formule (I): dans laquelle X, Y, Z, et R1 sont décrits dans l'invention, des procédés de préparation de ces composés, des compositions pharmaceutiques les contenant et l'utilisation de ces composés et compositions dans la prévention ou le traitement des troubles liés au récepteur de 5-HT2A.
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Designated States: AE, AG, AL, AM, AT, AU, AZ, BA, BB, BG, BR, BW, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DE, DK, DM, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, HR, HU, ID, IL, IN, IS, JP, KE, KG, KP, KR, KZ, LC, LK, LR, LS, LT, LU, LV, MA, MD, MG, MK, MN, MW, MX, MZ, NA, NI, NO, NZ, OM, PG, PH, PL, PT, RO, RU, SC, SD, SE, SG, SK, SL, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, YU, ZA, ZM, ZW
African Regional Intellectual Property Organization (ARIPO) (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Office (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (EPO) (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HU, IE, IT, LU, MC, NL, PL, PT, RO, SE, SI, SK, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG)
Publication Language: English (EN)
Filing Language: English (EN)