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1. (WO2005012283) SUBSTITUTED BENZOTHIOPHENE COMPOUNDS AND USES THEREOF
Latest bibliographic data on file with the International Bureau

Pub. No.: WO/2005/012283 International Application No.: PCT/US2004/024545
Publication Date: 10.02.2005 International Filing Date: 29.07.2004
IPC:
A61K 31/38 (2006.01) ,C07D 333/70 (2006.01) ,C07D 409/04 (2006.01) ,C07D 409/14 (2006.01)
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
33
Heterocyclic compounds
38
having sulfur as a ring hetero atom
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
333
Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
50
condensed with carbocyclic rings or ring systems
52
Benzo [b] thiophenes; Hydrogenated benzo [b] thiophenes
62
with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
68
Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
70
attached in position 2
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
409
Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
02
containing two hetero rings
04
directly linked by a ring-member-to-ring- member bond
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
409
Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
14
containing three or more hetero rings
Applicants:
BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. [US/US]; 900 Ridgebury Road P.O. Box 368 Ridgefield, Connecticut 06877-0368, US (AllExceptUS)
CHEN, Zhidong [US/US]; US (UsOnly)
GINN, John, David [US/US]; US (UsOnly)
HICKEY, Eugene, Richard [US/US]; US (UsOnly)
LIU, Weimin [CN/US]; US (UsOnly)
MAO, Can [CN/US]; US (UsOnly)
MORWICK, Tina, Marie [US/US]; US (UsOnly)
NEMOTO, Peter, Allen [US/US]; US (UsOnly)
SPERO, Denice [US/US]; US (UsOnly)
SUN, Sanxing [CN/US]; US (UsOnly)
Inventors:
CHEN, Zhidong; US
GINN, John, David; US
HICKEY, Eugene, Richard; US
LIU, Weimin; US
MAO, Can; US
MORWICK, Tina, Marie; US
NEMOTO, Peter, Allen; US
SPERO, Denice; US
SUN, Sanxing; US
Agent:
RAYMOND, Robert, P. ; Boehringer Ingelheim Corporation 900 Ridgebury Road P.O. Box 368 Ridgefield, Connecticut 06877-0368, US
Priority Data:
60/491,57531.07.2003US
Title (EN) SUBSTITUTED BENZOTHIOPHENE COMPOUNDS AND USES THEREOF
(FR) COMPOSES DE BENZOTHIOPHENE SUBSTITUES ET UTILISATIONS
Abstract:
(EN) Disclosed are compounds of the formula (I), wherein R1, R2, R3 and R4 are described herein, which are active as anti-inflammatory agents. Also disclosed are methods of using and making such compounds.
(FR) L'invention concerne des composés de formule (I). R1, R2, R3 et R4 sont tels que spécifiés dans la description. Ces composés sont actifs comme agents anti-inflammatoires. L'invention concerne également des procédés relatifs à l'utilisation et à l'élaboration des composés en question.
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Designated States: AE, AG, AL, AM, AT, AU, AZ, BA, BB, BG, BR, BW, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DE, DK, DM, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, HR, HU, ID, IL, IN, IS, JP, KE, KG, KP, KR, KZ, LC, LK, LR, LS, LT, LU, LV, MA, MD, MG, MK, MN, MW, MX, MZ, NA, NI, NO, NZ, OM, PG, PH, PL, PT, RO, RU, SC, SD, SE, SG, SK, SL, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, YU, ZA, ZM, ZW
African Regional Intellectual Property Organization (ARIPO) (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HU, IE, IT, LU, MC, NL, PL, PT, RO, SE, SI, SK, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG)
Publication Language: English (EN)
Filing Language: English (EN)
Also published as:
EP1651629JP2007533602CA2534127