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1. (WO2004103954) AMIDE DERIVATIVE
Latest bibliographic data on file with the International Bureau   

Pub. No.: WO/2004/103954 International Application No.: PCT/JP2004/007221
Publication Date: 02.12.2004 International Filing Date: 20.05.2004
IPC:
C07C 237/04 (2006.01) ,C07D 401/04 (2006.01) ,C07D 401/14 (2006.01)
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
C
ACYCLIC OR CARBOCYCLIC COMPOUNDS
237
Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups
02
having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton
04
the carbon skeleton being acyclic and saturated
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
401
Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
02
containing two hetero rings
04
directly linked by a ring-member-to-ring- member bond
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
401
Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
14
containing three or more hetero rings
Applicants:
中川 忠清 NAKAGAWA, Tadakiyo [JP/JP]; JP (UsOnly)
鈴木 保 SUZUKI, Tamotsu [JP/JP]; JP (UsOnly)
竹中 薫 TAKENAKA, Kaoru [JP/JP]; JP (UsOnly)
藤田 真一 FUJITA, Shinichi [JP/JP]; JP (UsOnly)
山多 洋司 YAMADA, Youji [JP/JP]; JP (UsOnly)
島 洋一郎 SHIMA, Yoichiro [JP/JP]; JP (UsOnly)
奥住 竜哉 OKUZUMI, Tatsuya [JP/JP]; JP (UsOnly)
吉村 敏彦 YOSHIMURA, Toshihiko [JP/JP]; JP (UsOnly)
吉田 正尚 YOSHIDA, Masanao [JP/JP]; JP (UsOnly)
村田 正弘 MURATA, Masahiro [JP/JP]; JP (UsOnly)
味の素株式会社 AJINOMOTO CO., INC. [JP/JP]; 〒1048315 東京都中央区京橋1丁目15番1号 Tokyo 15-1, Kyobashi 1-chome, Chuo-ku, Tokyo 1048315, JP (AllExceptUS)
Inventors:
中川 忠清 NAKAGAWA, Tadakiyo; JP
鈴木 保 SUZUKI, Tamotsu; JP
竹中 薫 TAKENAKA, Kaoru; JP
藤田 真一 FUJITA, Shinichi; JP
山多 洋司 YAMADA, Youji; JP
島 洋一郎 SHIMA, Yoichiro; JP
奥住 竜哉 OKUZUMI, Tatsuya; JP
吉村 敏彦 YOSHIMURA, Toshihiko; JP
吉田 正尚 YOSHIDA, Masanao; JP
村田 正弘 MURATA, Masahiro; JP
Agent:
高島 一 TAKASHIMA, Hajime; 〒5410044 大阪府大阪市中央区伏見町四丁目2番14号 藤村大和生命ビル Osaka Meiji Yasuda Seimei Osaka Midosuji Bldg., 1-1, Fushimimachi 4-chome, Chuo-ku, Osaka-shi, Osaka 541-0044, JP
Priority Data:
2003-14268120.05.2003JP
Title (EN) AMIDE DERIVATIVE
(FR) DERIVE D'AMIDE
(JA) アミド誘導体
Abstract:
(EN) An amide derivative represented by the formula (I): [wherein A represents cycloalkyl, aryl, or heteroaryl; X represents nitrogen or CR17; Y represents NRa, -(CRbRb')m-, etc.; m is 0 to 4; R1 to R17 may be the same or different and each represents hydrogen, halogeno, cyano, nitro, carboxy, formyl, hydroxy, ammonium, optionally substituted alkyl, ZR18, etc.; Z represents -O-, -S(O)p-, -S(O)pO-, -NH-, -NR19-, etc.; and R1 may be bonded to R2 to form a ring] or a pharmaceutically acceptable salt, hydrate, or solvate of the derivative. They are used in medical applications such as anti-inflammation and analgesia.
(FR) L'invention concerne un dérivé d'amide représenté par la formule (I) [dans laquelle A représente cycloalkyle, aryle ou hétéroaryle; X représente de l'azote ou CR17; Y représente NRa, -(CRbRb')m-, etc.; m varie entre 0 et 4; R1 à R17 peuvent être identiques ou différents et chacun représente hydrogène, halogéno, cyano, nitro, carboxy, formyle, hydroxy, ammonium, un alkyle éventuellement substitué, ZR18, etc.; Z représente -O-, -S(O)p-, -S(O)pO-, -NH-, -NR19-, etc.; et R1 peut être lié à R2 pour former un noyau], ou un sel, un hydrate ou un solvate acceptable d'un point de vue pharmaceutique du dérivé. Ceux-ci peuvent être utilisés dans des applications médicales telles que des médicaments anti-inflammatoires ou analgésiques.
(JA) not available
front page image
Designated States: AE, AG, AL, AM, AT, AU, AZ, BA, BB, BG, BR, BW, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DE, DK, DM, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, HR, HU, ID, IL, IN, IS, JP, KE, KG, KP, KR, KZ, LC, LK, LR, LS, LT, LU, LV, MA, MD, MG, MK, MN, MW, MX, MZ, NA, NI, NO, NZ, OM, PG, PH, PL, PT, RO, RU, SC, SD, SE, SG, SK, SL, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, YU, ZA, ZM, ZW
African Regional Intellectual Property Organization (ARIPO) (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Office (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (EPO) (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HU, IE, IT, LU, MC, NL, PL, PT, RO, SE, SI, SK, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG)
Publication Language: Japanese (JA)
Filing Language: Japanese (JA)