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1. (WO2004099176) DERIVATIVES OF PIPERIDINYL- AND PIPERAZINYL-ALKYL CARBAMATES, PREPARATION METHODS THEREOF AND APPLICATION OF SAME IN THERAPEUTICS
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2004/099176    International Application No.:    PCT/FR2004/001102
Publication Date: 18.11.2004 International Filing Date: 06.05.2004
Chapter 2 Demand Filed:    02.02.2005    
IPC:
C07D 211/26 (2006.01), C07D 213/38 (2006.01), C07D 295/13 (2006.01), C07D 401/04 (2006.01), C07D 401/14 (2006.01), C07D 413/04 (2006.01), C07D 417/04 (2006.01), C07D 471/04 (2006.01), C07D 491/04 (2006.01), C07D 495/04 (2006.01)
Applicants: SANOFI-AVENTIS [FR/FR]; 174, avenue de France, F-75013 Paris (FR) (For All Designated States Except US).
ABOUABDELLAH, Ahmed [FR/FR]; (FR) (For US Only).
BURNIER, Philippe [FR/FR]; (FR) (For US Only).
HOORNAERT, Christian [BE/FR]; (FR) (For US Only).
JEUNESSE, Jean [FR/FR]; (FR) (For US Only).
PUECH, Frédéric [FR/FR]; (FR) (For US Only)
Inventors: ABOUABDELLAH, Ahmed; (FR).
BURNIER, Philippe; (FR).
HOORNAERT, Christian; (FR).
JEUNESSE, Jean; (FR).
PUECH, Frédéric; (FR)
Agent: LUDWIG, Jacques; Sanofi-Aventis, 174, avenue de France, F-75013 Paris (FR)
Priority Data:
03/05540 07.05.2003 FR
Title (EN) DERIVATIVES OF PIPERIDINYL- AND PIPERAZINYL-ALKYL CARBAMATES, PREPARATION METHODS THEREOF AND APPLICATION OF SAME IN THERAPEUTICS
(FR) DERIVES DE PIPERIDINYL- ET PIPERAZINYL-ALKYLCARBAMATES, LEURS PROCEDES DE PREPARATION ET LEUR APPLICATION EN THERAPEUTIQUE
Abstract: front page image
(EN)The invention relates to a compound having general formula (I), wherein: A = N or CR2; R2 = H, F, OH, CN, CF3, C1-6-alkyl, C1-6-alcoxy; n = 2 or 3 and m = 2 when A = N; n = 1, 2 or 3 and m = 1 or 2 when A = CR2; B = covalent bond or C1-8-alkylene; R1 = optionally-substituted heteroaryl; R3 = CHR4CONHR5; R4 = H or C1-6-alkyl; R5 = H, C1-6-alkyl, C3-7-cycloalkyl, C3-7-cycloalkyl-Cl-6-alkylene; the base, the acid addition salt, the hydrate or the solvate thereof. The invention also relates to the application thereof in therapeutics.
(FR)Composé répondant à la formule générale (I) : dans laquelle A = N ou CR2 ; R2 = H, F, OH, CN, CF3, C1-6­-alkyle, C1-6-alcoxy ; n = 2 ou 3 et m = 2 lorsque A = N ; n = 1, 2 ou 3 et m = 1 ou 2 lorsque A = CR2 ; B = liaison covalente ou C1-8-alkylène ; R1 = hétéroaryle éventuellement substitué ; R3 = CHR4CONHR5 ; R4 = H ou C1-6-alkyle ; R5 = H, C1-6-alkyle, C3-7-cycloalkyle, C3-7-cycloalkyle-Cl-6-alkylène ; à l'état de base, de sel d'addition à un acide, d'hydrate ou de solvat. Application en thérapeutique.
Designated States: AE, AG, AL, AM, AT, AU, AZ, BA, BB, BG, BR, BW, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DE, DK, DM, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, HR, HU, ID, IL, IN, IS, JP, KE, KG, KP, KR, KZ, LC, LK, LR, LS, LT, LU, LV, MA, MD, MG, MK, MN, MW, MX, MZ, NA, NI, NO, NZ, OM, PG, PH, PL, PT, RO, RU, SC, SD, SE, SG, SK, SL, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, YU, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HU, IE, IT, LU, MC, NL, PL, PT, RO, SE, SI, SK, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: French (FR)
Filing Language: French (FR)