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Machine translation
1. (WO2004099136) PROCESS FOR PRODUCING PYRROLIDINE DERIVATIVE
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2004/099136    International Application No.:    PCT/JP2004/006471
Publication Date: 18.11.2004 International Filing Date: 07.05.2004
Chapter 2 Demand Filed:    02.03.2005    
IPC:
C07D 207/12 (2006.01)
Applicants: DAIICHI PHARMACEUTICAL CO., LTD. [JP/JP]; 14-10, Nihonbashi 3-chome, Chuo-ku, Tokyo 1038234 (JP) (For All Designated States Except US).
NAKAYAMA, Atsushi [JP/JP]; (JP) (For US Only).
MACHINAGA, Nobuo [JP/JP]; (JP) (For US Only).
YONEDA, Yoshiyuki [JP/JP]; (JP) (For US Only).
SETOGUCHI, Masaki [JP/JP]; (JP) (For US Only)
Inventors: NAKAYAMA, Atsushi; (JP).
MACHINAGA, Nobuo; (JP).
YONEDA, Yoshiyuki; (JP).
SETOGUCHI, Masaki; (JP)
Agent: THE PATENT CORPORATE BODY ARUGA PATENT OFFICE; Kyodo Bldg. 3-6, Nihonbashiningyocho 1-chome Chuo-ku, Tokyo 1030013 (JP)
Priority Data:
2003-131978 09.05.2003 JP
2003-144430 22.05.2003 JP
2003-209579 29.08.2003 JP
Title (EN) PROCESS FOR PRODUCING PYRROLIDINE DERIVATIVE
(FR) PROCEDE DE PRODUCTION DE DERIVES DE PYRROLIDINE
(JA) ピロリジン誘導体の製造方法
Abstract: front page image
(EN)A process for industrially advantageously producing a 1,4-trans-cyclohexanecarboxylic acid derivative (1) which has excellent VLA-4 inhibitory activity and is safe; and an intermediate advantageous for the production process. The process comprises converting a compound represented by the formula (I) into a compound represented by the formula (VI) according to the following scheme.
(FR)L'invention concerne un procédé de production industrielle, avantageuse, d'un dérivé d'acide 1,4-trans-cyclohexanecarboxylique (1) qui présente une excellente activité inhibitrice de VLA-4 et qui est sûr ; ainsi qu'un intermédiaire avantageux pour le procédé de production. Ledit procédé consiste à convertir un composé représenté par la formule (I) en un composé représenté par la formule (VI) selon le schéma suivant. (Voir schéma)
(JA)not available
Designated States: AE, AG, AL, AM, AT, AU, AZ, BA, BB, BG, BR, BW, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DE, DK, DM, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, HR, HU, ID, IL, IN, IS, JP, KE, KG, KP, KR, KZ, LC, LK, LR, LS, LT, LU, LV, MA, MD, MG, MK, MN, MW, MX, MZ, NA, NI, NO, NZ, OM, PG, PH, PL, PT, RO, RU, SC, SD, SE, SG, SK, SL, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, YU, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HU, IE, IT, LU, MC, NL, PL, PT, RO, SE, SI, SK, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: Japanese (JA)
Filing Language: Japanese (JA)