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Machine translation
1. (WO2004094411) PYRAZOLE DERIVATIVES AS PHOSPHODIESTERASE 4 INHIBITORS
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2004/094411    International Application No.:    PCT/US2004/011899
Publication Date: 04.11.2004 International Filing Date: 16.04.2004
IPC:
C07D 231/12 (2006.01), C07D 231/56 (2006.01), C07D 307/20 (2006.01), C07D 405/04 (2006.01), C07D 405/12 (2006.01), C07D 409/12 (2006.01)
Applicants: MEMORY PHARMACEUTICALS CORPORATION [US/US]; 100 Philips Parkway, Montvale, NJ 07645 (US) (For All Designated States Except US).
HOPPER, Allen [US/US]; (US) (For US Only).
KUESTER, Erik [US/US]; (US) (For US Only).
DUNN, Robert [US/US]; (US) (For US Only).
CONTICELLO, Richard [US/US]; (US) (For US Only)
Inventors: HOPPER, Allen; (US).
KUESTER, Erik; (US).
DUNN, Robert; (US).
CONTICELLO, Richard; (US)
Agent: HEANEY, Brion, P.; Millen, White, Zelano and Branigan, Suite 1400, 2200 Clarendon Blvd., Arlington, VA 22201 (US)
Priority Data:
60/463,725 18.04.2003 US
Title (EN) PYRAZOLE DERIVATIVES AS PHOSPHODIESTERASE 4 INHIBITORS
(FR) DERIVES DU PYRAZOLE INHIBITEURS DE LA PHOSPHODIESTERASE 4
Abstract: front page image
(EN)Selective PDE4 inhibition is achieved by aryl and heteroaryl pyrazole compounds. The compounds exhibit improved PDE4 inhibition as compared to compounds such as rolipram and show selectivity with regard to inhibition of other classes of PDEs.
(FR)L'invention porte sur des composés aryle et hétéroaryle de pyrazole inhibiteurs sélectifs de la PDE4 dont l'activité inhibitrice est améliorée par rapport à des composés tels que le rolipram et qui présentent une sélectivité quant à l'inhibition des autres classes de PDEs.
Designated States: AE, AG, AL, AM, AT, AU, AZ, BA, BB, BG, BR, BW, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DE, DK, DM, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, HR, HU, ID, IL, IN, IS, JP, KE, KG, KP, KR, KZ, LC, LK, LR, LS, LT, LU, LV, MA, MD, MG, MK, MN, MW, MX, MZ, NA, NI, NO, NZ, OM, PG, PH, PL, PT, RO, RU, SC, SD, SE, SG, SK, SL, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, YU, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LS, MW, MZ, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HU, IE, IT, LU, MC, NL, PL, PT, RO, SE, SI, SK, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: English (EN)
Filing Language: English (EN)