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1. WO2004029049 - NOVEL SALT OF 2-ACYLAMINOTHIAZOLE DERIVATIVE

Publication Number WO/2004/029049
Publication Date 08.04.2004
International Application No. PCT/JP2003/012419
International Filing Date 29.09.2003
Chapter 2 Demand Filed 13.02.2004
IPC
A61K 31/496 2006.1
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
33Heterocyclic compounds
395having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
495having six-membered rings with two nitrogen atoms as the only ring hetero atoms, e.g. piperazine
496Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene
C07D 417/14 2006.1
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
417Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/196
14containing three or more hetero rings
CPC
A61K 31/496
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
33Heterocyclic compounds
395having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
495having six-membered rings with two ; or more; nitrogen atoms as the only ring heteroatoms, e.g. piperazine ; or tetrazines
496Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene
A61P 7/04
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
7Drugs for disorders of the blood or the extracellular fluid
04Antihaemorrhagics; Procoagulants; Haemostatatic agents; Antifibrinolytic agents
C07D 417/14
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
417Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
14containing three or more hetero rings
Applicants
  • YAMANOUCHI PHARMACEUTICAL CO., LTD. [JP]/[JP] (AllExceptUS)
  • SUGASAWA, Keizo [JP]/[JP] (UsOnly)
  • KOGA, Yuji [JP]/[JP] (UsOnly)
  • HIRAYAMA, Fukushi [JP]/[JP] (UsOnly)
  • SUZUKI, Ken-ichi [JP]/[JP] (UsOnly)
  • AWAMURA, Yuuji [JP]/[JP] (UsOnly)
Inventors
  • SUGASAWA, Keizo
  • KOGA, Yuji
  • HIRAYAMA, Fukushi
  • SUZUKI, Ken-ichi
  • AWAMURA, Yuuji
Agents
  • NAGAI, Shozo
Priority Data
2002-28468930.09.2002JP
Publication Language Japanese (ja)
Filing Language Japanese (JA)
Designated States
Title
(EN) NOVEL SALT OF 2-ACYLAMINOTHIAZOLE DERIVATIVE
(FR) NOUVEAU SEL D'UN DERIVE DE 2-ACYLAMINOTHIAZOLE
(JA) 2-アシルアミノチアゾール誘導体の新規な塩
Abstract
(EN) Maleic acid salt of 1-(3-chloro-5-{[4-(4-chlorothiophen-2-yl)-5-(4-cyclohexylpiperazin-1-yl)thiazol-2-yl]carbamoyl}pyridin-2-yl)piperidine-4-carboxylic acid which is useful as a remedy for thrombopenia, and drugs, in particular platelet-increasing agent and/or a remedy for thrombopenia, containing this compound as the active ingredient.
(FR) L'invention se rapporte à un sel d'acide maléique d'acide 1-(3-chloro-5-{[4-(4-chlorothiophén-2-yl)-5-(4-cyclohexylpipérazin-1-yl)thiazol-2-yl]carbamoyl}pyridin-2-yl)pipéridine-4-carboxylique, qui peut être utilisé en tant que remède pour traiter une thrombocytopénie. Cette invention concerne en outre des médicaments, en particulier un agent d'augmentation du nombre de thrombocytes et/ou un remède pour traiter une thrombocytopénie, contenant ledit composé en tant qu'ingrédient actif.
(JA) 血小板減少症治療剤として有用な、1-(3-クロロ-5-{[4-(4-クロロチオフェン-2-イル)-5-(4-シクロヘキシルピペラジン-1-イル)チアゾール-2-イル]カルバモイル}ピリジン-2-イル)ピペリジン-4-カルボン酸マレイン酸塩、及び該化合物を有効成分とする医薬、特に血小板増多剤及び/又は血小板減少症治療剤。
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