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Machine translation
1. (WO2004002491) MORPHOLINE AND TETRAHYDROPYRAN DRIVATIVES AND THEIR USE AS CATHEPSIN INHIBITORS
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2004/002491    International Application No.:    PCT/US2003/019960
Publication Date: 08.01.2004 International Filing Date: 25.06.2003
Chapter 2 Demand Filed:    02.12.2003    
IPC:
A61K 31/4245 (2006.01), A61K 31/5375 (2006.01), A61K 31/5377 (2006.01), C07D 213/40 (2006.01), C07D 263/32 (2006.01), C07D 263/56 (2006.01), C07D 271/06 (2006.01), C07D 295/185 (2006.01), C07D 498/04 (2006.01)
Applicants: AVENTIS PHARMACEUTICALS INC. [US/US]; 300 Somerset Corporate Boulevard, Bridgewater, NJ 08807-2854 (US) (For All Designated States Except US).
AXYS PHARMACEUTICALS, INC. [US/US]; 180 Kimball Way, South San Francisco, CA 94080 (US) (For All Designated States Except US).
GRAUPE, Michael [AT/US]; (US) (For US Only).
PALMER, James, T. [US/US]; (US) (For US Only).
PATTERSON, John, W. [US/US]; (US) (For US Only).
PICKETT, Stephen, D. [GB/GB]; (GB) (For US Only).
ALDOUS, David, J. [US/US]; (US) (For US Only).
THURAIRATNAM, Sukanthini [GB/US]; (US) (For US Only).
TIMM, Andreas, P. [DE/US]; (US) (For US Only).
HALLEY, Frank [FR/FR]; (FR) (For US Only).
LAI, Justine [SG/GB]; (GB) (For US Only).
LINK, John [US/US]; (US) (For US Only).
LI, Jiayao [CN/US]; (US) (For US Only)
Inventors: GRAUPE, Michael; (US).
PALMER, James, T.; (US).
PATTERSON, John, W.; (US).
PICKETT, Stephen, D.; (GB).
ALDOUS, David, J.; (US).
THURAIRATNAM, Sukanthini; (US).
TIMM, Andreas, P.; (US).
HALLEY, Frank; (FR).
LAI, Justine; (GB).
LINK, John; (US).
LI, Jiayao; (US)
Agent: WANG, George, G.; AVENTIS PHARMACEUTICALS INC., P. O. Box 6800, Route 202-206, Bridgewater, NJ 08807-0800 (US)
Priority Data:
10/183,128 26.06.2002 US
Title (EN) MORPHOLINE AND TETRAHYDROPYRAN DRIVATIVES AND THEIR USE AS CATHEPSIN INHIBITORS
(FR) DERIVES DE MORPHOLINE ET DE TETRAHYDROPYRANE ET LEUR UTILISATION EN TANT QU'INHIBITEURS DE CATHEPSINE
Abstract: front page image
(EN)The present invention relates to novel cathepsin S inhibitors, the pharmaceutically acceptable salts and N-oxides thereof, their uses as therapeutic agents and the methods of their making.
(FR)La présente invention concerne de nouveaux inhibiteurs de cathepsine S, leurs sels et N-oxydes pharmaceutiquement acceptables, leurs utilisations en tant qu'agents thérapeutiques et leurs procédés de production.
Designated States: AE, AG, AL, AM, AT, AU, AZ, BA, BB, BG, BR, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DE, DK, DM, DZ, EC, EE, ES, FI, GB, GD, GE, GH, GM, HR, HU, ID, IL, IN, IS, JP, KE, KG, KP, KR, KZ, LC, LK, LR, LS, LT, LU, LV, MA, MD, MG, MK, MN, MW, MX, MZ, NI, NO, NZ, OM, PH, PL, PT, RO, RU, SC, SD, SE, SG, SK, SL, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, YU, ZA, ZM, ZW.
African Regional Intellectual Property Organization (GH, GM, KE, LS, MW, MZ, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HU, IE, IT, LU, MC, NL, PT, RO, SE, SI, SK, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: English (EN)
Filing Language: English (EN)