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Machine translation
1. (WO2003078419) N-SUBSTITUTED BENZOTHIOPHENESULFONAMIDE DERIVATIVE
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2003/078419    International Application No.:    PCT/JP2003/003023
Publication Date: 25.09.2003 International Filing Date: 13.03.2003
IPC:
C07D 333/62 (2006.01), C07D 413/12 (2006.01), C07D 417/12 (2006.01)
Applicants: TOA EIYO LTD. [JP/JP]; 1-2, Kyobashi 3-chome Chuo-ku, Tokyo 104-0031 (JP)
Inventors: SATO, Shoji; (JP).
MIZUNO, Yusuke; (JP).
MASAKI, Hidekazu; (JP)
Agent: OGURI, Shohei; Eikoh Patent Office 28th Floor, ARK Mori Building 12-32, Akasaka 1-chome Minato-ku, Tokyo 107-6028 (JP)
Priority Data:
2002-072307 15.03.2002 JP
Title (EN) N-SUBSTITUTED BENZOTHIOPHENESULFONAMIDE DERIVATIVE
(FR) DERIVE DU BENZOTHIOPHENESULFONAMIDE SUBSTITUE EN N
Abstract: front page image
(EN)An N-substituted benzothiophenesulfonamide derivative represented by the following formula (I) or pharmaceutically acceptable salt thereof. The compound is excellent in human chymase inhibitory activity and enzyme selectivity. Also provided are a chymase inhibitor and a medicine each containing the derivative or salt. (The substituents are as defined in claim 1.)
(FR)L'invention porte sur un dérivé du benzothiophènesulfonamide substitué en n de formule (I), ou sur un de sels pharmacocompatibles. Ce composé est excellent du point de vue de son activité inhibitrice de la chymase humaine et de sa sélectivité des enzymes. L'invention porte également sur un inhibiteur de la chymase et sur un médicament, contenant tous deux ledit dérivé ou ledit sel. (Les substituants sont définis dans la revendication 1)
Designated States: CA, CN, JP.
European Patent Office (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HU, IE, IT, LU, MC, NL, PT, RO, SE, SI, SK, TR).
Publication Language: Japanese (JA)
Filing Language: Japanese (JA)