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1. (WO2003076421) AMINOCARBONYL-DERIVATIVES AS NOVEL INHIBITORS OF HISTONE DEACETYLASE
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2003/076421    International Application No.:    PCT/EP2003/002511
Publication Date: 18.09.2003 International Filing Date: 11.03.2003
Chapter 2 Demand Filed:    02.09.2003    
IPC:
C07D 207/09 (2006.01), C07D 207/14 (2006.01), C07D 211/58 (2006.01), C07D 213/78 (2006.01), C07D 217/02 (2006.01), C07D 239/42 (2006.01), C07D 295/155 (2006.01), C07D 295/26 (2006.01), C07D 307/68 (2006.01), C07D 401/04 (2006.01), C07D 401/12 (2006.01), C07D 403/04 (2006.01), C07D 409/12 (2006.01), C07D 413/04 (2006.01), C07D 471/10 (2006.01), C12Q 1/48 (2006.01)
Applicants: JANSSEN PHARMACEUTICA N.V. [BE/BE]; Turnhoutseweg 30, B-2340 Beerse (BE) (For All Designated States Except US).
VAN EMELEN, Kristof [BE/BE]; (BE) (For US Only).
DE WINTER, Hans, Louis, Jos [BE/BE]; (BE) (For US Only).
DYATKIN, Alexey, Borisovich [RU/US]; (US) (For US Only).
VERDONCK, Marc, Gustaaf, Celine [BE/BE]; (BE) (For US Only).
MEERPOEL, Lieven [BE/BE]; (BE) (For US Only)
Inventors: VAN EMELEN, Kristof; (BE).
DE WINTER, Hans, Louis, Jos; (BE).
DYATKIN, Alexey, Borisovich; (US).
VERDONCK, Marc, Gustaaf, Celine; (BE).
MEERPOEL, Lieven; (BE)
Common
Representative:
JANSSEN PHARMACEUTICA N.V.; Karen Vermuyten GA4736, J & J Patent Law Department, Turnhoutseweg 30, B-2340 Beerse (BE)
Priority Data:
60/363,799 13.03.2002 US
Title (EN) AMINOCARBONYL-DERIVATIVES AS NOVEL INHIBITORS OF HISTONE DEACETYLASE
(FR) DERIVES AMINOCARBONYL UTILISES EN TANT QUE NOUVEAUX INHIBITEURS D'HISTONE DEACETYLASE
Abstract: front page image
(EN)This invention comprises the novel compounds of formula (I)wherein n, R1, R2, R3, R4, L, Q, X, Y, Z and have defined meanings, having histone deacetylase inhibiting enzymatic activity; their preparation, compositions containing them and their use as a medicine.
(FR)L'invention concerne des nouveaux composés de formule générale (I) dans laquelle n, R1, R2, R3, R4, L, Q, X, Y, Z et a) ont la signification indiquée dans la description, qui présentent une activité enzymatique inhibant l'histone déacetylase. L'invention concerne également leur préparation, des compositions les contenant ainsi que leur utilisation en tant que médicament.
Designated States: AE, AG, AL, AM, AT, AU, AZ, BA, BB, BG, BR, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DE, DK, DM, DZ, EC, EE, ES, FI, GB, GD, GE, GH, GM, HR, HU, ID, IL, IN, IS, JP, KE, KG, KP, KR, KZ, LC, LK, LR, LS, LT, LU, LV, MA, MD, MG, MK, MN, MW, MX, MZ, NI, NO, NZ, OM, PH, PL, PT, RO, RU, SC, SD, SE, SG, SK, SL, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, YU, ZA, ZM, ZW.
African Regional Intellectual Property Organization (GH, GM, KE, LS, MW, MZ, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HU, IE, IT, LU, MC, NL, PT, SE, SI, SK, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: English (EN)
Filing Language: English (EN)