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1. (WO2003074479) SEMICARBAZIDE DERIVATIVES AND THEIR USE AS ANTITHROMBOTICS
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2003/074479    International Application No.:    PCT/EP2003/001177
Publication Date: 12.09.2003 International Filing Date: 06.02.2003
Chapter 2 Demand Filed:    27.08.2003    
IPC:
A61K 31/175 (2006.01), A61K 31/18 (2006.01), A61K 31/195 (2006.01), A61K 31/4245 (2006.01), A61P 7/02 (2006.01), A61P 9/08 (2006.01), A61P 9/10 (2006.01), A61P 25/06 (2006.01), A61P 29/00 (2006.01), A61P 35/00 (2006.01), A61P 35/04 (2006.01), A61P 43/00 (2006.01), C07C 281/06 (2006.01), C07C 311/47 (2006.01), C07C 317/40 (2006.01), C07C 317/42 (2006.01), C07D 271/06 (2006.01)
Applicants: MERCK PATENT GMBH [DE/DE]; Frankfurter Strasse 250, 64293 Darmstadt (DE) (For All Designated States Except US).
MEDERSKI, Werner [DE/DE]; (DE) (For US Only).
CEZANNE, Bertram [DE/DE]; (DE) (For US Only).
TSAKLAKIDIS, Christos [GR/DE]; (DE) (For US Only).
DORSCH, Dieter [DE/DE]; (DE) (For US Only).
BARNES, Christopher [GB/DE]; (DE) (For US Only).
GLEITZ, Johannes [DE/DE]; (DE) (For US Only)
Inventors: MEDERSKI, Werner; (DE).
CEZANNE, Bertram; (DE).
TSAKLAKIDIS, Christos; (DE).
DORSCH, Dieter; (DE).
BARNES, Christopher; (DE).
GLEITZ, Johannes; (DE)
Common
Representative:
MERCK PATENT GMBH; Frankfurter Strasse 250, 64293 Darmstadt (DE)
Priority Data:
102 09 211.7 04.03.2002 DE
Title (DE) SEMICARBAZIDDERIVATE UND IHRE VERWENDUNG ALS ANTITHROMBOTIKA
(EN) SEMICARBAZIDE DERIVATIVES AND THEIR USE AS ANTITHROMBOTICS
(FR) DERIVES DE SEMICARBAZIDES ET LEUR UTILISATION EN TANT QU'ANTITHROMBOTIQUES
Abstract: front page image
(DE)Neue Verbindungen der Formel I worin R, R1, R2 und R3 die in Patentanspruch 1 angegebene Bedeutung haben, sind Inhibitoren des Koagulationsfaktors Xa und können zur Prophylaxe und/oder Therapie von thromboembolischen Erkrankungen und zur Behandlung von Tumoren eingesetzt werden.
(EN)The invention relates to the novel compounds of formula (I), wherein R, R1, R2 and R3 are defined as in claim 1. The novel compounds are inhibitors of coagulation factor Xa and are used in the prophylaxis and/or therapy of thromboembolic diseases and in the treatment of tumors.
(FR)L'invention concerne de nouveaux composés de formule (I) dans laquelle R, R1, R2 et R3 ont la signification indiquée dans la première revendication. Ces composés constituent des inhibiteurs du facteur de coagulation Xa et peuvent être utilisés pour prévenir et/ou traiter des maladies thromboemboliques ainsi que pour traiter des tumeurs.
Designated States: AE, AG, AL, AM, AT, AU, AZ, BA, BB, BG, BR, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DE, DK, DM, DZ, EC, EE, ES, FI, GB, GD, GE, GH, GM, HR, HU, ID, IL, IN, IS, JP, KE, KG, KP, KR, KZ, LC, LK, LR, LS, LT, LU, LV, MA, MD, MG, MK, MN, MW, MX, MZ, NO, NZ, OM, PH, PL, PT, RO, RU, SC, SD, SE, SG, SK, SL, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, YU, ZA, ZM, ZW.
African Regional Intellectual Property Organization (GH, GM, KE, LS, MW, MZ, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HU, IE, IT, LU, MC, NL, PT, SE, SI, SK, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: German (DE)
Filing Language: German (DE)