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1. (WO2003059335) PHENYL SULFOXIDES AND PHENYL SULFONES
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2003/059335    International Application No.:    PCT/EP2003/000052
Publication Date: 24.07.2003 International Filing Date: 07.01.2003
Chapter 2 Demand Filed:    18.07.2003    
IPC:
C07C 317/18 (2006.01), C07D 207/06 (2006.01), C07D 207/46 (2006.01), C07D 211/22 (2006.01), C07D 211/46 (2006.01), C07D 211/52 (2006.01), C07D 213/74 (2006.01), C07D 239/42 (2006.01), C07D 241/08 (2006.01), C07D 295/205 (2006.01), C07D 491/10 (2006.01)
Applicants: BAYER HEALTHCARE AG [DE/DE]; 51368 Leverkusen (DE) (For All Designated States Except US).
HENDRIX, Martin [DE/DE]; (DE) (For US Only).
BAUMANN, Karlheinz [DE/DE]; (DE) (For US Only).
GROSSER, Rolf [DE/DE]; (DE) (For US Only).
KÖNIG, Gerhard [DE/DE]; (DE) (For US Only).
DÜSTERHUS, Vera [DE/DE]; (DE) (For US Only).
KRÜGER, Joachim [DE/DE]; (DE) (For US Only)
Inventors: HENDRIX, Martin; (DE).
BAUMANN, Karlheinz; (DE).
GROSSER, Rolf; (DE).
KÖNIG, Gerhard; (DE).
DÜSTERHUS, Vera; (DE).
KRÜGER, Joachim; (DE)
Common
Representative:
BAYER HEALTHCARE AG; 51368 Leverkusen (DE)
Priority Data:
102 01 392.6 16.01.2002 DE
Title (DE) PHENYLSULFOXIDE UND -SULFONE
(EN) PHENYL SULFOXIDES AND PHENYL SULFONES
(FR) OXYDES SULFONIQUES DE PHENYLE ET SULFONES DE PHENYLE
Abstract: front page image
(DE)Die Erfindung betrifft Phenylsulfoxide und -sulfone der Formel (I) und Verfahren zu ihrer Herstellung sowie ihre Verwendung zur Herstellung von Arzneimitteln zur Behandlung und/oder Prophylaxe von Krankheiten, insbesondere der Alzheimerschen Krankheit. Die erfindungsgemässen Verbindungen inhibieren ϝ-Sekretase. (Formel I).
(EN)The invention relates to the phenyl sulfoxides and phenyl sulfones of formula (I) and to methods for producing the same as well as to their use in the production of drugs for the treatment and/or prophylaxis of diseases, especially Alzheimer's disease. The inventive compounds inhibit $g(g) secretase.
(FR)L'invention concerne de l'oxyde sulfonique de phényle ou des sulfones de phényle de formule (I), leur procédé de production et leur utilisation dans la production de médicaments pour le traitement et/ou la prophylaxie de maladies, en particulier la maladie d'Alzheimer. Lesdits composés de l'invention inhibent la $g(g)-sécrétase.
Designated States: AE, AG, AL, AM, AT, AU, AZ, BA, BB, BG, BR, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DE, DK, DM, DZ, EC, EE, ES, FI, GB, GD, GE, GH, GM, HR, HU, ID, IL, IN, IS, JP, KE, KG, KP, KR, KZ, LC, LK, LR, LS, LT, LU, LV, MA, MD, MG, MK, MN, MW, MX, MZ, NI, NO, NZ, OM, PH, PL, PT, RO, RU, SC, SD, SE, SG, SK, SL, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, YU, ZA, ZM, ZW.
African Regional Intellectual Property Organization (GH, GM, KE, LS, MW, MZ, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HU, IE, IT, LU, MC, NL, PT, SE, SI, SK, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: German (DE)
Filing Language: German (DE)