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1. (WO2003008395) SUBSTITUTED ISOXAZOLES AND THE USE THEREOF AS ANTIBIOTICS
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2003/008395    International Application No.:    PCT/ES2002/000358
Publication Date: 30.01.2003 International Filing Date: 17.07.2002
Chapter 2 Demand Filed:    30.01.2003    
IPC:
C07D 261/08 (2006.01), C07D 413/12 (2006.01), C07D 413/14 (2006.01), C07D 417/14 (2006.01)
Applicants: LABORATORIOS S.A.L.V.A.T., S.A. [ES/ES]; Calle Gall, 30-36, E-08950 Esplugues de Llobregat (ES) (For All Designated States Except US).
FARRERONS GALLEMI, Carles [ES/ES]; (ES) (For US Only).
LAGUNAS ARNAL, Carmen [ES/ES]; (ES) (For US Only).
FERNANDEZ SERRAT, Anna [ES/ES]; (ES) (For US Only).
CATENA RUIZ, Juan Lorenzo [ES/ES]; (ES) (For US Only).
MIQUEL BONO, Ignacio José [ES/ES]; (ES) (For US Only).
BALSA LOPEZ, Dolors [ES/ES]; (ES) (For US Only).
SALCEDO ROCA, Carolina [ES/ES]; (ES) (For US Only).
TOLEDO MESA, Natividad [ES/ES]; (ES) (For US Only).
FERNANDEZ GARCIA, Andrés [ES/ES]; (ES) (For US Only)
Inventors: FARRERONS GALLEMI, Carles; (ES).
LAGUNAS ARNAL, Carmen; (ES).
FERNANDEZ SERRAT, Anna; (ES).
CATENA RUIZ, Juan Lorenzo; (ES).
MIQUEL BONO, Ignacio José; (ES).
BALSA LOPEZ, Dolors; (ES).
SALCEDO ROCA, Carolina; (ES).
TOLEDO MESA, Natividad; (ES).
FERNANDEZ GARCIA, Andrés; (ES)
Agent: SUGRAÑES MOLINE, Pedro; Calle Provenza, 304, E-08008 Barcelona (ES).
SUGRANES-VERDONCES-FERREGÜELA; 304, Calle Provenza_(Association NO.121), E-08008 Barcelona (ES)
Priority Data:
P 200101793 20.07.2001 ES
Title (EN) SUBSTITUTED ISOXAZOLES AND THE USE THEREOF AS ANTIBIOTICS
(ES) ISOXAZOLES SUSTITUIDOS Y SU UTILIZACION COMO ANTIBIOTICOS
(FR) ISOXAZOLES SUBSTITUES ET UTILISATION COMME ANTIBIOTIQUES
Abstract: front page image
(EN)The invention relates to compounds having formula (I), wherein X is O, S, NH, OCO, NH-CO, NH-COO, NH-CO-NH, NH-CS or NH-CS-NH; R4 is H, (C1-C3)-alkyl which is optionally substituted with halogen or a heterocyclic carbon radical which is selected from various possibilities; R1 and R3 are H or F; and R2 is a heterocyclic nitrogen or carbon radical. Said compounds can be used to treat microbial infections in the human or animal body.
(ES)Los compuestos de fórmula (I), donde X es O, S, NH, OCO, NH-CO, NH-COO, NH-CO-NH, NH-CS o NH-CS-NH; R4 es H, (C1-C3)-alquilo opcionalmente sustituido por halógeno, o un radical heterocíclico de carbono seleccionado entre varias posibilidades; R1 y R3 son H o F; y R2 es un radical heterocíclico de nitrógeno o carbono, son útiles para el tratamiento de infecciones microbianas en el cuerpo humano o animal.
(FR)L'invention concerne des composés représentés par la formule (I), dans laquelle X est O, S, NH, OCO, NH-CO, NH-COO, NH-CO-NH, NH-CS ou NH-CS-NH; R4 est H, (C1-C3)-alkyle éventuellement substitué par halogène, ou un radical hétérocyclique de carbone sélectionné parmi diverses possibilités; R1 et R3 sont H ou F; et R2 est un radical hétérocyclique d'azote ou de carbone. Lesdits composés sont utilisés dans le traitement d'infections microbiennes dans le corps humain ou animal.
Designated States: AE, AG, AL, AM, AT, AU, AZ, BA, BB, BG, BR, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DE, DK, DM, DZ, EC, EE, ES, FI, GB, GD, GE, GH, GM, HR, HU, ID, IL, IN, IS, JP, KE, KG, KP, KR, KZ, LC, LK, LR, LS, LT, LU, LV, MA, MD, MG, MK, MN, MW, MX, MZ, NO, NZ, OM, PH, PL, PT, RO, RU, SD, SE, SG, SI, SK, SL, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VN, YU, ZA, ZM, ZW.
African Regional Intellectual Property Organization (GH, GM, KE, LS, MW, MZ, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, IE, IT, LU, MC, NL, PT, SE, SK, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: Spanish (ES)
Filing Language: Spanish (ES)