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Machine translation
1. (WO2003002530) PYRROLIDINES AS DIPEPTIDYL PEPTIDASE INHIBITORS
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2003/002530    International Application No.:    PCT/US2002/020466
Publication Date: 09.01.2003 International Filing Date: 26.06.2002
Chapter 2 Demand Filed:    13.12.2002    
IPC:
C07D 207/16 (2006.01), C07D 207/273 (2006.01), C07D 207/48 (2006.01), C07D 277/06 (2006.01), C07D 401/06 (2006.01), C07D 401/12 (2006.01), C07D 401/14 (2006.01), C07D 403/12 (2006.01), C07D 409/12 (2006.01), C07D 413/12 (2006.01), C07D 413/14 (2006.01), C07D 451/04 (2006.01)
Applicants: SMITHKLINE BEECHAM CORPORATION [US/US]; One Franklin Plaza, Philadelphia, PA 19101 (US) (For All Designated States Except US).
HAFFNER, Curt, Dale [US/US]; (US) (For US Only).
MCDOUGALD, Darryl, Lynn [US/US]; (US) (For US Only).
RANDHAWA, Amarjit, Sab [CA/US]; (US) (For US Only).
REISTER, Steven, Michael [US/US]; (US) (For US Only).
DEATON, David, N. [US/US]; (US) (For US Only).
LENHARD, James, Martin [US/US]; (US) (For US Only)
Inventors: HAFFNER, Curt, Dale; (US).
MCDOUGALD, Darryl, Lynn; (US).
RANDHAWA, Amarjit, Sab; (US).
REISTER, Steven, Michael; (US).
DEATON, David, N.; (US).
LENHARD, James, Martin; (US)
Agent: LEVY, David, J; GlaxoSmtihKline, Five Moore Drive, PO Box 13398, Research Triangle Park, NC 27709 (US)
Priority Data:
60/301,333 27.06.2001 US
60/387,011 06.06.2002 US
Title (EN) PYRROLIDINES AS DIPEPTIDYL PEPTIDASE INHIBITORS
(FR) PYRROLIDINES SERVANT D'INHIBITEURS DE DIPEPTIDYL PEPTIDASE
Abstract: front page image
(EN)The present invention relates to novel compounds of formula (I):, their use for inhibiting serine proteases, such as dipeptidyl peptidases, such as dipeptidyl peptidase IV (DPP-IV) and to methods for their production and their therapeutic utility.
(FR)La présente invention concerne de nouveaux composés, leur utilisation dans l'inhibition de sérine protéases telles que des dipeptidyl peptidases, par exemple dipeptidyl peptidase IV (DPP-IV), des procédés de fabrication de ces composés ainsi que leur utilisation en thérapie.
Designated States: AE, AG, AL, AM, AT, AU, AZ, BA, BB, BG, BR, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DE, DK, DM, DZ, EC, EE, ES, FI, GB, GD, GE, GH, GM, HR, HU, ID, IL, IN, IS, JP, KE, KG, KP, KR, KZ, LC, LK, LR, LS, LT, LU, LV, MA, MD, MG, MK, MN, MW, MX, MZ, NO, NZ, OM, PH, PL, PT, RO, RU, SD, SE, SG, SI, SK, SL, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VN, YU, ZA, ZM, ZW.
African Regional Intellectual Property Organization (GH, GM, KE, LS, MW, MZ, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, CH, CY, DE, DK, ES, FI, FR, GB, GR, IE, IT, LU, MC, NL, PT, SE, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: English (EN)
Filing Language: English (EN)