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1. WO2002032872 - NITROGENOUS AROMATIC RING COMPOUNDS

Publication Number WO/2002/032872
Publication Date 25.04.2002
International Application No. PCT/JP2001/009221
International Filing Date 19.10.2001
Chapter 2 Demand Filed 15.02.2002
IPC
C07D 207/34 2006.1
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
207Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
02with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
30having two double bonds between ring members or between ring members and non-ring members
34with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
C07D 213/26 2006.1
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
213Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
02having three double bonds between ring members or between ring members and non-ring members
04having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
24with substituted hydrocarbon radicals attached to ring carbon atoms
26Radicals substituted by halogen atoms or nitro radicals
C07D 213/68 2006.1
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
213Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
02having three double bonds between ring members or between ring members and non-ring members
04having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
60with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
62Oxygen or sulfur atoms
63One oxygen atom
68attached in position 4
C07D 213/73 2006.1
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
213Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
02having three double bonds between ring members or between ring members and non-ring members
04having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
60with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
72Nitrogen atoms
73Unsubstituted amino or imino radicals
C07D 213/74 2006.1
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
213Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
02having three double bonds between ring members or between ring members and non-ring members
04having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
60with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
72Nitrogen atoms
74Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
C07D 213/75 2006.1
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
213Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
02having three double bonds between ring members or between ring members and non-ring members
04having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
60with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
72Nitrogen atoms
75Amino or imino radicals, acylated by carboxylic or carbonic acids, or by sulfur or nitrogen analogues thereof, e.g. carbamates
CPC
A61K 31/4706
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
33Heterocyclic compounds
395having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
435having six-membered rings with one nitrogen as the only ring hetero atom
47Quinolines; Isoquinolines
47064-Aminoquinolines; 8-Aminoquinolines, e.g. chloroquine, primaquine
A61K 31/4745
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
33Heterocyclic compounds
395having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
435having six-membered rings with one nitrogen as the only ring hetero atom
47Quinolines; Isoquinolines
4738ortho- or peri-condensed with heterocyclic ring systems
4745condensed with ring systems having nitrogen as a ring hetero atom, e.g. phenantrolines
A61K 31/517
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
33Heterocyclic compounds
395having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
495having six-membered rings with two ; or more; nitrogen atoms as the only ring heteroatoms, e.g. piperazine ; or tetrazines
505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
517ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
A61K 31/519
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
33Heterocyclic compounds
395having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
495having six-membered rings with two ; or more; nitrogen atoms as the only ring heteroatoms, e.g. piperazine ; or tetrazines
505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
519ortho- or peri-condensed with heterocyclic rings
A61P 17/06
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
17Drugs for dermatological disorders
06Antipsoriatics
A61P 19/02
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
19Drugs for skeletal disorders
02for joint disorders, e.g. arthritis, arthrosis
Applicants
  • EISAI CO., LTD. [JP]/[JP] (AllExceptUS)
  • FUNAHASHI, Yasuhiro [JP]/[JP] (UsOnly)
  • TSURUOKA, Akihiko [JP]/[JP] (UsOnly)
  • MATSUKURA, Masayuki [JP]/[JP] (UsOnly)
  • HANEDA, Toru [JP]/[JP] (UsOnly)
  • FUKUDA, Yoshio [JP]/[JP] (UsOnly)
  • KAMATA, Junichi [JP]/[JP] (UsOnly)
  • TAKAHASHI, Keiko [JP]/[JP] (UsOnly)
  • MATSUSHIMA, Tomohiro [JP]/[JP] (UsOnly)
  • MIYAZAKI, Kazuki [JP]/[JP] (UsOnly)
  • NOMOTO, Ken-ichi [JP]/[JP] (UsOnly)
  • WATANABE, Tatsuo [JP]/[JP] (UsOnly)
  • OBAISHI, Hiroshi [JP]/[JP] (UsOnly)
  • YAMAGUCHI, Atsumi [JP]/[JP] (UsOnly)
  • SUZUKI, Sachi [JP]/[JP] (UsOnly)
  • NAKAMURA, Katsuji [JP]/[JP] (UsOnly)
  • MIMURA, Fusayo [JP]/[JP] (UsOnly)
  • YAMAMOTO, Yuji [JP]/[JP] (UsOnly)
  • MATSUI, Junji [JP]/[JP] (UsOnly)
  • MATSUI, Kenji [JP]/[JP] (UsOnly)
  • YOSHIBA, Takako [JP]/[JP] (UsOnly)
  • SUZUKI, Yasuyuki [JP]/[JP] (UsOnly)
  • ARIMOTO, Itaru [JP]/[JP] (UsOnly)
Inventors
  • FUNAHASHI, Yasuhiro
  • TSURUOKA, Akihiko
  • MATSUKURA, Masayuki
  • HANEDA, Toru
  • FUKUDA, Yoshio
  • KAMATA, Junichi
  • TAKAHASHI, Keiko
  • MATSUSHIMA, Tomohiro
  • MIYAZAKI, Kazuki
  • NOMOTO, Ken-ichi
  • WATANABE, Tatsuo
  • OBAISHI, Hiroshi
  • YAMAGUCHI, Atsumi
  • SUZUKI, Sachi
  • NAKAMURA, Katsuji
  • MIMURA, Fusayo
  • YAMAMOTO, Yuji
  • MATSUI, Junji
  • MATSUI, Kenji
  • YOSHIBA, Takako
  • SUZUKI, Yasuyuki
  • ARIMOTO, Itaru
Agents
  • HASEGAWA, Yoshiki
Priority Data
2000-32042020.10.2000JP
2000-38619520.12.2000JP
2001-4668522.02.2001JP
Publication Language Japanese (JA)
Filing Language Japanese (JA)
Designated States
Title
(EN) NITROGENOUS AROMATIC RING COMPOUNDS
(FR) COMPOSES A NOYAU AROMATIQUE AZOTE
Abstract
(EN)
Compounds represented by the general formula (|) or salts thereof, or hydrates of both: (|) wherein Ag is an optionally substituted 5- to 14-membered heterocyclic group, or the like; Xg is O-, -S-, or the like; Yg is optionally substituted C6-14 aryl, a 5- to 14-membered heterocyclic group, or the like; and Tg1 is a group of the general formula (||) or the like: (||) [wherein Eg is a single bond, -N(Rg2)-, or the like; Rg1 and Rg2 are each independently hydrogen, optionally substituted C1-6 alkyl, or the like; and Zg is C1-8 alkyl, C3-8 alicyclic hydrocarbyl, C6-14 aryl, or the like].
(FR)
L'invention concerne des composés représentés par la formule générale (I) ou leurs sels, ou leurs hydrates. Dans cette formule, Ag représente un groupe hétérocyclique comprenant entre 5 et 14 éléments, éventuellement substitué, ou analogue ; Xg représente un -O-, un -S-, ou analogue ; Yg représente un aryle en C6 à C14, un groupe hétérocyclique comprenant entre 5 et 14 éléments, ou analogue ; et Tg1 représente un groupe représenté par la formule générale (II) ou analogue [dans laquelle Eg représente une liaison simple, un -N(Rg2)-, ou analogue ; Rg1 et Rg2 représentent chacun indépendamment un hydrogène, un alkyle en C1 à C6 éventuellement substitué, ou analogue ; et Zg représente un alkyle en C1 à C8, un hydrocarbyle alicyclique en C3 à C8, un aryle en C6 à C14, ou analogue].
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