WIPO logo
Mobile | Deutsch | Español | Français | 日本語 | 한국어 | Português | Русский | 中文 | العربية |
PATENTSCOPE

Search International and National Patent Collections
World Intellectual Property Organization
Search
 
Browse
 
Translate
 
Options
 
News
 
Login
 
Help
 
Machine translation
1. (WO2002030931) AZA- AND POLYAZA-NAPHTHALENYL CARBOXAMIDES USEFUL AS HIV INTEGRASE INHIBITORS
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2002/030931    International Application No.:    PCT/US2001/042564
Publication Date: 18.04.2002 International Filing Date: 09.10.2001
Chapter 2 Demand Filed:    07.05.2002    
IPC:
C07D 471/04 (2006.01)
Applicants: MERCK & CO., INC. [US/US]; 126 East Lincoln Avenue Rahway, NJ 07065-0907 (US) (For All Designated States Except US).
ANTHONY, Neville, J. [GB/US]; (US) (For US Only).
GOMEZ, Robert, P. [US/US]; (US) (For US Only).
YOUNG, Steven, D. [US/US]; (US) (For US Only).
EGBERTSON, Melissa [US/US]; (US) (For US Only).
WAI, John, S. [US/US]; (US) (For US Only).
ZHUANG, Linghang [CN/US]; (US) (For US Only).
EMBREY, Mark [US/US]; (US) (For US Only).
TRAN, Lekhanh [US/US]; (US) (For US Only).
MELAMED, Jeffrey, Y. [US/US]; (US) (For US Only).
LANGFORD, H., Marie [US/US]; (US) (For US Only).
GUARE, James, P. [US/US]; (US) (For US Only).
FISHER, Thorsten, E. [US/US]; (US) (For US Only).
JOLLY, Samson, M. [US/US]; (US) (For US Only).
KUO, Michelle, S. [US/US]; (US) (For US Only).
PERLOW, Debra, S. [US/US]; (US) (For US Only).
BENNETT, Jennifer, J. [US/US]; (US) (For US Only).
FUNK, Timothy, W. [US/US]; (US) (For US Only)
Inventors: ANTHONY, Neville, J.; (US).
GOMEZ, Robert, P.; (US).
YOUNG, Steven, D.; (US).
EGBERTSON, Melissa; (US).
WAI, John, S.; (US).
ZHUANG, Linghang; (US).
EMBREY, Mark; (US).
TRAN, Lekhanh; (US).
MELAMED, Jeffrey, Y.; (US).
LANGFORD, H., Marie; (US).
GUARE, James, P.; (US).
FISHER, Thorsten, E.; (US).
JOLLY, Samson, M.; (US).
KUO, Michelle, S.; (US).
PERLOW, Debra, S.; (US).
BENNETT, Jennifer, J.; (US).
FUNK, Timothy, W.; (US)
Common
Representative:
MERCK & CO., INC.; 126 East Lincoln Avenue Rahway, NJ 07065-0907 (US)
Priority Data:
60/239,707 12.10.2000 US
60/281,656 05.04.2001 US
Title (EN) AZA- AND POLYAZA-NAPHTHALENYL CARBOXAMIDES USEFUL AS HIV INTEGRASE INHIBITORS
(FR) AZA-NAPHTALENYLE CARBOXAMIDES ET POLYAZA-NAPHTALENYLE CARBOXAMIDES UTILES EN TANT QU'INHIBITEURS DE L'INTEGRASE DU VIH
Abstract: front page image
(EN)Aza- and polyaza-naphthalenyl carboxamide derivatives including certain quinoline carboxamide and naphthyridine carboxamide derivatives are described. These compounds are inhibitors of HIV integrase and inhibitors of HIV replication, and are useful in the prevention or treatment of infection by HIV and the treatment of AIDS, as compounds or pharmaceutically acceptable salts, or as ingredients in pharmaceutical compositions, optionally in combination with other antivirals, immunomodulators, antibiotics or vaccines. Methods of preventing, treating or delaying the onset of AIDS and methods of preventing or treating infection by HIV are also described.
(FR)L'invention concerne des dérivés d' aza-naphtalényle carboxamide et de polyaza-naphtalényle carboxamide comprenant certains dérivés de quinoline carboxamide et de naphtyridine carboxamide. Ces composés sont des inhibiteurs de l'intégrase du VIH et des inhibiteurs de réplication du VIH et sont utiles pour la prévention ou le traitement d'infections à VIH et le traitement du SIDA, en tant que composés ou sels pharmaceutiquement acceptables, ou en tant qu'ingrédients dans des compositions pharmaceutiques, éventuellement combinés à d'autres antiviraux, immunomodulateurs, antibiotiques ou vaccins. L'invention concerne également des méthodes permettant de prévenir, de traiter ou de retarder l'apparition du SIDA ainsi que des méthodes permettant de prévenir ou de traiter une infection à VIH.
Designated States: AE, AG, AL, AM, AT, AU, AZ, BA, BB, BG, BR, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DE, DK, DM, DZ, EC, EE, ES, FI, GB, GD, GE, GH, GM, HR, HU, ID, IL, IN, IS, JP, KE, KG, KR, KZ, LC, LK, LR, LS, LT, LU, LV, MA, MD, MG, MK, MN, MW, MX, MZ, NO, NZ, PH, PL, PT, RO, RU, SD, SE, SG, SI, SK, SL, TJ, TM, TR, TT, TZ, UA, UG, US, UZ, VN, YU, ZA, ZW.
African Regional Intellectual Property Organization (GH, GM, KE, LS, MW, MZ, SD, SL, SZ, TZ, UG, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, CH, CY, DE, DK, ES, FI, FR, GB, GR, IE, IT, LU, MC, NL, PT, SE, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: English (EN)
Filing Language: English (EN)