WIPO logo
Mobile | Deutsch | Español | Français | 日本語 | 한국어 | Português | Русский | 中文 | العربية |
PATENTSCOPE

Search International and National Patent Collections
World Intellectual Property Organization
Search
 
Browse
 
Translate
 
Options
 
News
 
Login
 
Help
 
Machine translation
1. (WO2002030930) AZA- AND POLYAZA-NAPHTHALENYL CARBOXAMIDES USEFUL AS HIV INTEGRASE INHIBITORS
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2002/030930    International Application No.:    PCT/US2001/031456
Publication Date: 18.04.2002 International Filing Date: 09.10.2001
Chapter 2 Demand Filed:    07.05.2002    
IPC:
C07D 471/04 (2006.01)
Applicants: MERCK & CO., INC. [US/US]; 126 East Lincoln Avenue Rahway, NJ 07065-0907 (US) (For All Designated States Except US).
ANTHONY, Neville, J. [GB/US]; (US) (For US Only).
GOMEZ, Robert, P. [US/US]; (US) (For US Only).
YOUNG, Steven, D. [US/US]; (US) (For US Only).
EGBERTSON, Melissa [US/US]; (US) (For US Only).
WAI, John, S. [US/US]; (US) (For US Only).
ZHUANG, Linghang [CN/US]; (US) (For US Only).
EMBREY, Mark [US/US]; (US) (For US Only).
TRAN, Lekhanh [US/US]; (US) (For US Only).
MELAMED, Jeffrey, Y. [US/US]; (US) (For US Only).
LANGFORD, H., Marie [US/US]; (US) (For US Only).
GUARE, James, P. [US/US]; (US) (For US Only).
FISHER, Thorsten, E. [US/US]; (US) (For US Only).
JOLLY, Samson, M. [US/US]; (US) (For US Only).
KUO, Michelle, S. [US/US]; (US) (For US Only).
PERLOW, Debra, S. [US/US]; (US) (For US Only).
BENNETT, Jennifer, J. [US/US]; (US) (For US Only).
FUNK, Timothy, W. [US/US]; (US) (For US Only)
Inventors: ANTHONY, Neville, J.; (US).
GOMEZ, Robert, P.; (US).
YOUNG, Steven, D.; (US).
EGBERTSON, Melissa; (US).
WAI, John, S.; (US).
ZHUANG, Linghang; (US).
EMBREY, Mark; (US).
TRAN, Lekhanh; (US).
MELAMED, Jeffrey, Y.; (US).
LANGFORD, H., Marie; (US).
GUARE, James, P.; (US).
FISHER, Thorsten, E.; (US).
JOLLY, Samson, M.; (US).
KUO, Michelle, S.; (US).
PERLOW, Debra, S.; (US).
BENNETT, Jennifer, J.; (US).
FUNK, Timothy, W.; (US)
Common
Representative:
MERCK & CO., INC.; 126 East Lincoln Avenue Rahway, NJ 07065-0907 (US)
Priority Data:
60/239,707 12.10.2000 US
60/281,656 05.04.2001 US
Title (EN) AZA- AND POLYAZA-NAPHTHALENYL CARBOXAMIDES USEFUL AS HIV INTEGRASE INHIBITORS
(FR) AZA- ET POLYAZA-NAPHTHALENYL CARBOXAMIDES UTILES COMME INHIBITEURS DE L'INTEGRASE DU VIH
Abstract: front page image
(EN)Aza- and polyaza-naphthalenyl carboxamide derivatives including certain quinoline carboxamide and naphthyridine carboxamide derivatives are described. These compounds are inhibitors of HIV integrase and inhibitors of HIV replication, and are useful in the prevention or treatment of infection by HIV and the treatment of AIDS, as compounds or pharmaceutically acceptable salts, or as ingredients in pharmaceutical compositions, optionally in combination with other antivirals, immunomodulators, antibiotics or vaccines. Methods of preventing, treating or delaying the onset of AIDS and methods of preventing or treating infection by HIV are also described.
(FR)L'invention concerne des dérivés d'aza- et de polyaza-nathtalenyl carboxamides, y compris certains dérivés de quinoline carboxamide et naphtyridine carboxamide. Ces composés sont des inhibiteurs de l'intégrase du VIH et des inhibiteurs de la réplication du VIH, et sont utiles dans la prévention et le traitement d'une infection par le VIH et le traitement du SIDA, comme composés ou sels pharmaceutiquement acceptables ou comme ingrédients dans des compositions pharmaceutiques, éventuellement combinés avec d'autres antiviraux, immunomodulateurs, antibiotiques ou vaccins. L'invention concerne également des méthodes destinées à prévenir, traiter ou à retarder l'apparition des premiers signes du SIDA ainsi que des méthodes de prévention ou de traitement d'une infection par le VIH.
Designated States: AE, AG, AL, AM, AT, AU, AZ, BA, BB, BG, BR, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DE, DK, DM, DZ, EC, EE, ES, FI, GB, GD, GE, GH, GM, HR, HU, ID, IL, IN, IS, JP, KE, KG, KR, KZ, LC, LK, LR, LS, LT, LU, LV, MA, MD, MG, MK, MN, MW, MX, MZ, NO, NZ, PH, PL, PT, RO, RU, SD, SE, SG, SI, SK, SL, TJ, TM, TR, TT, TZ, UA, UG, US, UZ, VN, YU, ZA, ZW.
African Regional Intellectual Property Organization (GH, GM, KE, LS, MW, MZ, SD, SL, SZ, TZ, UG, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, CH, CY, DE, DK, ES, FI, FR, GB, GR, IE, IT, LU, MC, NL, PT, SE, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: English (EN)
Filing Language: English (EN)