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1. WO2001055107 - AROMATIC AMINES AND AMIDES ACTING ON THE MELANOCORTIN RECEPTORS

Publication Number WO/2001/055107
Publication Date 02.08.2001
International Application No. PCT/GB2001/000356
International Filing Date 29.01.2001
Chapter 2 Demand Filed 21.08.2001
IPC
C07C 233/40 2006.1
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
CACYCLIC OR CARBOCYCLIC COMPOUNDS
233Carboxylic acid amides
01having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
34having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by amino groups
35with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom
40having the carbon atom of the carboxamide group bound to an acyclic carbon atom of a carbon skeleton containing six-membered aromatic rings
C07C 237/06 2006.1
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
CACYCLIC OR CARBOCYCLIC COMPOUNDS
237Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups
02having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton
04the carbon skeleton being acyclic and saturated
06having the nitrogen atoms of the carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
C07C 279/14 2006.1
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
CACYCLIC OR CARBOCYCLIC COMPOUNDS
279Derivatives of guanidine, i.e. compounds containing the group the singly-bound nitrogen atoms not being part of nitro or nitroso groups
04having nitrogen atoms of guanidine groups bound to acyclic carbon atoms of a carbon skeleton
14being further substituted by carboxyl groups
C07D 209/08 2006.1
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
209Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
02condensed with one carbocyclic ring
04Indoles; Hydrogenated indoles
08with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to carbon atoms of the hetero ring
C07D 209/12 2006.1
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
209Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
02condensed with one carbocyclic ring
04Indoles; Hydrogenated indoles
10with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
12Radicals substituted by oxygen atoms
C07D 209/18 2006.1
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
209Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
02condensed with one carbocyclic ring
04Indoles; Hydrogenated indoles
10with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
18Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
CPC
C07C 233/40
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
CACYCLIC OR CARBOCYCLIC COMPOUNDS
233Carboxylic acid amides
01having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
34having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by amino groups
35with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom
40having the carbon atom of the carboxamide group bound to an acyclic carbon atom of a carbon skeleton containing six-membered aromatic rings
C07C 237/06
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
CACYCLIC OR CARBOCYCLIC COMPOUNDS
237Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups
02having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton
04the carbon skeleton being acyclic and saturated
06having the nitrogen atoms of the carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
C07C 2602/10
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
CACYCLIC OR CARBOCYCLIC COMPOUNDS
2602Systems containing two condensed rings
02the rings having only two atoms in common
04One of the condensed rings being a six-membered aromatic ring
10the other ring being six-membered, e.g. tetraline
C07C 279/14
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
CACYCLIC OR CARBOCYCLIC COMPOUNDS
279Derivatives of guanidine, i.e. compounds containing the group , the singly-bound nitrogen atoms not being part of nitro or nitroso groups
04having nitrogen atoms of guanidine groups bound to acyclic carbon atoms of a carbon skeleton
14being further substituted by carboxyl groups
C07D 209/08
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
209Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
02condensed with one carbocyclic ring
04Indoles; Hydrogenated indoles
08with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to carbon atoms of the hetero ring
C07D 209/12
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
209Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
02condensed with one carbocyclic ring
04Indoles; Hydrogenated indoles
10with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
12Radicals substituted by oxygen atoms
Applicants
  • MELACURE THERAPEUTICS AB [SE]/[SE] (AllExceptUS)
  • LUNDSTEDT, Torbjörn [SE]/[SE] (UsOnly)
  • SKOTTNER, Anna [SE]/[SE] (UsOnly)
  • SEIFERT, Elisabeth [SE]/[SE] (UsOnly)
  • ANDERSSON, Per [SE]/[SE] (UsOnly)
  • KAULINA, Larisa [--]/[LV] (UsOnly)
  • DIKOVSKAYA, Klara [LV]/[LV] (UsOnly)
  • MUTULE, Ilze [LV]/[SE] (UsOnly)
  • MUTULIS, Felikss [LV]/[SE] (UsOnly)
  • WIKBERG, Jarl [SE]/[SE] (UsOnly)
  • STARCHENKOV, Igor [--]/[LV] (UsOnly)
  • KREICBERGA, Jana [LV]/[LV] (UsOnly)
Inventors
  • LUNDSTEDT, Torbjörn
  • SKOTTNER, Anna
  • SEIFERT, Elisabeth
  • ANDERSSON, Per
  • KAULINA, Larisa
  • DIKOVSKAYA, Klara
  • MUTULE, Ilze
  • MUTULIS, Felikss
  • WIKBERG, Jarl
  • STARCHENKOV, Igor
  • KREICBERGA, Jana
Agents
  • PETT, Christopher, Phineas
Priority Data
0002056.028.01.2000GB
0002058.628.01.2000GB
Publication Language English (en)
Filing Language English (EN)
Designated States
Title
(EN) AROMATIC AMINES AND AMIDES ACTING ON THE MELANOCORTIN RECEPTORS
(FR) NOUVEAUX AMINES ET AMIDES AROMATIQUES AGISSANT SUR LES RECEPTEURS DE LA MELANOCORTINE
Abstract
(EN) The present invention relates to novel aromatic amines and amides of general formula (I) and to the use of these amines and amides for the treatment of obesity, anorexia, inflammation, mental disorders and other diseases associated with the melanocortin receptors or related systems, e.g. the melanocyte stimulating hormones.
(FR) La présente invention concerne de nouveaux amines et amides aromatiques représentés par la formule générale (I) et l'utilisation des ces amines et amides dans le traitement de l'obésité, de l'anorexie, des inflammations, des troubles mentaux et d'autres maladies associées aux récepteurs de la mélanocortine ou aux systèmes ayant un rapport avec ceux-ci, comme par exemple les hormones stimulatrices des mélanocytes.
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