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1. (WO2001036371) CARBONIC ACID DERIVATIVES AND THEIR USE AS ECTOPARASITICIDAL COMPOSITION
Latest bibliographic data on file with the International Bureau   

Pub. No.: WO/2001/036371 International Application No.: PCT/EP2000/011470
Publication Date: 25.05.2001 International Filing Date: 17.11.2000
Chapter 2 Demand Filed: 26.05.2001
IPC:
C07C 69/65 (2006.01) ,C07C 69/96 (2006.01) ,C07C 233/20 (2006.01) ,C07C 255/45 (2006.01) ,C07C 255/55 (2006.01) ,C07C 257/08 (2006.01)
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
C
ACYCLIC OR CARBOCYCLIC COMPOUNDS
69
Esters of carboxylic acids; Esters of carbonic or haloformic acids
62
Halogen-containing esters
65
of unsaturated acids
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
C
ACYCLIC OR CARBOCYCLIC COMPOUNDS
69
Esters of carboxylic acids; Esters of carbonic or haloformic acids
96
Esters of carbonic or haloformic acids
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
C
ACYCLIC OR CARBOCYCLIC COMPOUNDS
233
Carboxylic acid amides
01
having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
16
having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms
17
with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom
20
having the carbon atom of the carboxamide group bound to a carbon atom of an acyclic unsaturated carbon skeleton
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
C
ACYCLIC OR CARBOCYCLIC COMPOUNDS
255
Carboxylic acid nitriles
45
having cyano groups bound to carbon atoms of rings other than six-membered aromatic rings
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
C
ACYCLIC OR CARBOCYCLIC COMPOUNDS
255
Carboxylic acid nitriles
49
having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
55
containing cyano groups and esterified hydroxy groups bound to the carbon skeleton
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
C
ACYCLIC OR CARBOCYCLIC COMPOUNDS
257
Compounds containing carboxyl groups, the doubly-bound oxygen atom of a carboxyl group being replaced by a doubly-bound nitrogen atom, this nitrogen atom not being further bound to an oxygen atom, e.g. imino-ethers, amidines
04
without replacement of the other oxygen atom of the carboxyl group, e.g. imino-ethers
08
having carbon atoms of imino-carboxyl groups bound to carbon atoms of six-membered aromatic rings
Applicants:
DUCRAY, Pierre [FR/FR]; FR (UsOnly)
BOUVIER, Jacques [CH/CH]; CH (UsOnly)
KAMINSKY, Roland [DE/CH]; CH (UsOnly)
FROELICH, Olivier [FR/FR]; FR (UsOnly)
NOVARTIS AG [CH/CH]; Lichstrasse 35 CH-4056 Basel, CH (AE, AG, AL, AM, AU, AZ, BA, BB, BE, BF, BG, BJ, BR, BY, BZ, CA, CF, CG, CH, CI, CM, CN, CR, CU, CY, CZ, DE, DK, DM, DZ, EE, ES, FI, FR, GA, GB, GD, GE, GH, GM, GN, GR, GW, HR, HU, ID, IE, IL, IN, IS, IT, JP, KE, KG, KP, KR, KZ, LC, LK, LR, LS, LT, LU, LV, MA, MC, MD, MG, MK, ML, MN, MR, MW, MX, MZ, NE, NL, NO, NZ, PL, PT, RO, RU, SD, SE, SG, SI, SK, SL, SN, SZ, TD, TG, TJ, TM, TR, TT, TZ, UA, UG, UZ, VN, YU, ZA, ZW)
NOVARTIS-ERFINDUNGEN VERWALTUNGSGESELLSCHAFT MBH [AT/AT]; Brunner Strasse 59 A-1230 Vienna, AT (AT)
Inventors:
DUCRAY, Pierre; FR
BOUVIER, Jacques; CH
KAMINSKY, Roland; CH
FROELICH, Olivier; FR
Agent:
BECKER, Konrad; Novartis AG Corporate Intellectual Property Patent & Trademark Dept. CH-4002 Basel, CH
Priority Data:
2115/9919.11.1999CH
Title (EN) CARBONIC ACID DERIVATIVES AND THEIR USE AS ECTOPARASITICIDAL COMPOSITION
(FR) DERIVES D'ACIDE CARBONIQUE ET UTILISATION EN TANT QUE COMPOSITION ECTOPARASITICIDE
Abstract:
(EN) There are described new compounds of formula (I) wherein, when n is 0, at least one of the two phenyl rings is substituted; R1 and R2 are each independently of the other hydrogen, halogen, cyano, nitro, C1-4alkyl, C1-4haloalkyl, C1-4alkoxy, C1-4 haloalkoxy or benzyl; A is oxygen, sulfur or -N(R6)-, wherein R6 is C1-4alkyl, phenylthio or tolylthio; B is -C(O)-, -O-C(O)- or -C(N-R6)-, wherein n is 0 or 1 and R6 is hydrogen of C1-4alkyl; p is an integer from 1 to 10; R3, R4 and R5 are each independently of the others hydrogen, halogen, cyano, nitro, C1-4alkyl, C1-4haloalkyl, C1-4alkoxy or C1-4haloalkoxy; or R3 and R4 are adjacent to one another and together with the phenyl ring to which they are bonded form a naphthyl group; m is 0, 1, 2 or 3; and Z is C1-6 alkyl, phenyl or halogen; in free form or in the form of physiologically tolerable salts. Also described is the preparation of those substances and their use in controlling ectoparasites on domestic animals, productive livestock and pets, as well as ectoparasiticidal compositions for use on such animals.
(FR) L'invention concerne des composés de formule (I) dans laquelle n est 0, au moins un des deux cycles phényle est substitué, R1 et R2 sont tous deux indépendants de l'autre hydrogène, halogène, cyano, nitro, C1-4alkyle, C1-4haloalkyle, C1-4alkoxy, C1-4haloalkoxy ou benzyle; A est de l'oxygène, du soufre ou -N(R6)-, R6 étant du C1-4alkyle, phénylthio ou tolylthio; B est -C(O)-, -O-C(O)- ou -C(N-R6)-, n étant 0 ou 1, et R6 est de l'hydrogène de C1-4alkyle; p est un entier de 1 à 10; R3, R4 et R5 sont tous indépendants des autres hydrogène, halogène, cyano, nitro, C1-4alkyle, C1-4haloalkyle, C1-4alkoxy ou C1-4haloalkoxy; ou R3 et R4 sont adjacents et forment un groupe naphtyle avec le cycle phényle auquel ils sont liés ; m est 0, 1, 2 ou 3; et Z est du C1-6alkyle, phényl ou halogène, sous forme libre ou sous forme de sels physiologiquement acceptables. L'invention concerne également la préparation de ces substances et leur utilisation dans le contrôle des ectoparasites sur des animaux domestiques, et sur le bétail et les animaux producteurs, ainsi que des compositions ectoparasiticides destinées à une utilisation sur de tels animaux.
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Designated States: AE, AG, AL, AM, AT, AU, AZ, BA, BB, BG, BR, BY, BZ, CA, CH, CN, CR, CU, CZ, DE, DK, DM, DZ, EE, ES, FI, GB, GD, GE, GH, GM, HR, HU, ID, IL, IN, IS, JP, KE, KG, KP, KR, KZ, LC, LK, LR, LS, LT, LU, LV, MA, MD, MG, MK, MN, MW, MX, MZ, NO, NZ, PL, PT, RO, RU, SD, SE, SG, SI, SK, SL, TJ, TM, TR, TT, TZ, UA, UG, US, UZ, VN, YU, ZA, ZW
African Regional Intellectual Property Organization (ARIPO) (GH, GM, KE, LS, MW, MZ, SD, SL, SZ, TZ, UG, ZW)
Eurasian Patent Office (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (EPO) (AT, BE, CH, CY, DE, DK, ES, FI, FR, GB, GR, IE, IT, LU, MC, NL, PT, SE, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GW, ML, MR, NE, SN, TD, TG)
Publication Language: English (EN)
Filing Language: English (EN)