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1. (WO2001032629) 1-BENZYLPYRAZOLES-3-CARBOXYLIC ACID TRICYCLIC DERIVATIVES AS CANNABINOID RECEPTOR ANTAGONISTS

Pub. No.:    WO/2001/032629    International Application No.:    PCT/FR2000/003047
Publication Date: Fri May 11 01:59:59 CEST 2001 International Filing Date: Fri Nov 03 00:59:59 CET 2000
IPC: C07D 231/54
Applicants: SANOFI-SYNTHELABO
BARTH, Francis
MILLAN, Joseph
OUSTRIC, Didier
RINALDI, Murielle
VERNHET, Martine
Inventors: BARTH, Francis
MILLAN, Joseph
OUSTRIC, Didier
RINALDI, Murielle
VERNHET, Martine
Title: 1-BENZYLPYRAZOLES-3-CARBOXYLIC ACID TRICYCLIC DERIVATIVES AS CANNABINOID RECEPTOR ANTAGONISTS
Abstract:
The invention concerns 1-benzylpyrazole-3-carboxylic acid tricyclic derivatives of formula W4 wherein: X represents a (CH2)n- group and R1 represents a non-aromatic C3-C15 carbocyclic radical. The invention also concerns the method for preparing said derivatives and medicines containing them. The compounds of formula (I) have an activity towards cannabinoid CB2 receptors.