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Machine translation
1. (WO2001004093) PROCESS FOR PRODUCING PAROXETINE DERIVATIVES BY MITSUNOBU REACTION
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2001/004093    International Application No.:    PCT/GB2000/002698
Publication Date: 18.01.2001 International Filing Date: 13.07.2000
Chapter 2 Demand Filed:    30.01.2001    
IPC:
C07D 211/18 (2006.01), C07D 211/22 (2006.01), C07D 211/24 (2006.01), C07D 405/12 (2006.01)
Applicants: SMITHKLINE BEECHAM PLC [GB/GB]; New Horizons Court, Brentford, Middlesex TW8 9EP (GB) (For All Designated States Except US).
JONES, David, Alan [GB/GB]; (GB) (For US Only)
Inventors: JONES, David, Alan; (GB)
Agent: WEST, Vivien; SmithKline Beecham, Corporate Intellectual Property, Two New Horizons Court, Brentford, Middlesex TW8 9EP (GB).
GIDDINGS, Peter, John; Corporate Intellectual Property, SmithKline Beecham, Two New Horizons Court, Brentford, Middlesex TW8 9EP (GB)
Priority Data:
9916392.5 13.07.1999 GB
Title (EN) PROCESS FOR PRODUCING PAROXETINE DERIVATIVES BY MITSUNOBU REACTION
(FR) NOUVEAU PROCEDE
Abstract: front page image
(EN)A process for manufacturing a compound of structure (1) where Y is substituted phenyl, especially 3,4-methylenedioxy-phenyl, or OY is a sulphonate leaving group; comprises coupling a compound of formula (2) to a phenolic compound such as sesamol or a sulphonic acid using a Mitsunobu reaction.
(FR)L'invention concerne un procédé de production d'un composé de la structure (1) dans laquelle Y est un phényle substitué, en particulier un 3,4-méthylènedioxy-phényle, ou OY est un groupe sulfonate partant. Le procédé consiste à associer un composé de la formule (2) à un composé phénolique, tel que le sésamol ou un acide sulfonique, par une réaction de Mitsunobu.
Designated States: AE, AG, AL, AM, AT, AU, AZ, BA, BB, BG, BR, BY, BZ, CA, CH, CN, CR, CU, CZ, DE, DK, DM, DZ, EE, ES, FI, GB, GD, GE, GH, GM, HR, HU, ID, IL, IN, IS, JP, KE, KG, KP, KR, KZ, LC, LK, LR, LS, LT, LU, LV, MA, MD, MG, MK, MN, MW, MX, MZ, NO, NZ, PL, PT, RO, RU, SD, SE, SG, SI, SK, SL, TJ, TM, TR, TT, TZ, UA, UG, US, UZ, VN, YU, ZA, ZW.
African Regional Intellectual Property Organization (GH, GM, KE, LS, MW, MZ, SD, SL, SZ, TZ, UG, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, CH, CY, DE, DK, ES, FI, FR, GB, GR, IE, IT, LU, MC, NL, PT, SE)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GW, ML, MR, NE, SN, TD, TG).
Publication Language: English (EN)
Filing Language: English (EN)