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1. (WO2001000210) REVERSE-TURN MIMETICS AND METHODS RELATING THERETO
Latest bibliographic data on file with the International Bureau   

Pub. No.: WO/2001/000210 International Application No.: PCT/US2000/017053
Publication Date: 04.01.2001 International Filing Date: 20.06.2000
Chapter 2 Demand Filed: 25.01.2001
IPC:
A61K 31/4985 (2006.01) ,A61K 31/519 (2006.01) ,A61K 31/551 (2006.01) ,A61K 38/00 (2006.01) ,C07B 61/00 (2006.01) ,C07D 487/04 (2006.01) ,C07K 5/02 (2006.01)
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
33
Heterocyclic compounds
395
having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
495
having six-membered rings with two nitrogen atoms as the only ring hetero atoms, e.g. piperazine
4985
Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
33
Heterocyclic compounds
395
having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
495
having six-membered rings with two nitrogen atoms as the only ring hetero atoms, e.g. piperazine
505
Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
519
ortho- or peri-condensed with heterocyclic rings
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
33
Heterocyclic compounds
395
having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
55
having seven-membered rings, e.g. azelastine, pentylenetetrazole
551
having two nitrogens as ring hetero atoms, e.g. clozapine, dilazep
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
38
Medicinal preparations containing peptides
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
B
GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
61
Other general methods
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
487
Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/-C07D477/183
02
in which the condensed system contains two hetero rings
04
Ortho-condensed systems
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
K
PEPTIDES
5
Peptides having up to four amino acids in a fully defined sequence; Derivatives thereof
02
containing at least one abnormal peptide link
Applicants: KAHN, Michael[US/US]; US (UsOnly)
EGUCHI, Masakatsu[JP/US]; US (UsOnly)
KIM, Hwa-Ok[US/US]; US (UsOnly)
STASIAK, Marcin[PL/US]; US (UsOnly)
MOLECUMETICS LTD.[US/US]; Suite 400 2023 120th Avenue Northeast Bellevue, WA 98005, US (AllExceptUS)
Inventors: KAHN, Michael; US
EGUCHI, Masakatsu; US
KIM, Hwa-Ok; US
STASIAK, Marcin; US
Agent: HERMANNS, Karl, R. ; Seed Intellectual Property Law Group PLLC Suite 6300 701 Fifth Avenue Seattle, WA 98104-7092, US
GOWSHALL, Jon V., FORREST & BOEHMERT,; Franz-Joseph-Str. 38, D-80801 Munchen, DE
Priority Data:
09/344,22125.06.1999US
Title (EN) REVERSE-TURN MIMETICS AND METHODS RELATING THERETO
(FR) MIMETIQUES DE COUDES INVERSES ET METHODES ASSOCIEES
Abstract:
(EN) Conformationally constrained compounds which mimic the secondary structure of reverse-turn regions of biologically active peptides and proteins are disclosed. Such reverse-turn mimetics have utility in the treatment of cell adhesion-indicated diseases, such as multiple sclerosis, atherosclerosis, asthma and inflammatory bowel disease.
(FR) L'invention concerne des composés conformationnellement contraints qui imitent la structure secondaire de régions à coudes inverses de peptides et de protéines biologiquement actifs. Lesdits mimétiques de coudes inverses sont utiles pour le traitement de pathologies induites par l'adhésion de cellules, telles que la sclérose en plaques, l'athérosclérose, l'asthme ou les affections intestinales inflammatoires.
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Designated States: AE, AG, AL, AM, AT, AU, AZ, BA, BB, BG, BR, BY, BZ, CA, CH, CN, CR, CU, CZ, DE, DK, DM, DZ, EE, ES, FI, GB, GD, GE, GH, GM, HR, HU, ID, IL, IN, IS, JP, KE, KG, KP, KR, KZ, LC, LK, LR, LS, LT, LU, LV, MA, MD, MG, MK, MN, MW, MX, MZ, NO, NZ, PL, PT, RO, RU, SD, SE, SG, SI, SK, SL, TJ, TM, TR, TT, TZ, UA, UG, US, UZ, VN, YU, ZA, ZW
African Regional Intellectual Property Organization (ARIPO) (GH, GM, KE, LS, MW, MZ, SD, SL, SZ, TZ, UG, ZW)
Eurasian Patent Office (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (EPO) (AT, BE, CH, CY, DE, DK, ES, FI, FR, GB, GR, IE, IT, LU, MC, NL, PT, SE)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GW, ML, MR, NE, SN, TD, TG)
Publication Language: English (EN)
Filing Language: English (EN)