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1. WO2000040599 - POLYOL COMPOUNDS, THEIR PRODUCTION AND USE

Publication Number WO/2000/040599
Publication Date 13.07.2000
International Application No. PCT/JP2000/000023
International Filing Date 06.01.2000
Chapter 2 Demand Filed 21.07.2000
IPC
A61K 38/00 2006.01
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
38Medicinal preparations containing peptides
C07K 5/02 2006.01
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
KPEPTIDES
5Peptides having up to four amino acids in a fully defined sequence; Derivatives thereof
02containing at least one abnormal peptide link
CPC
A61K 38/00
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
38Medicinal preparations containing peptides
C07K 5/0207
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
KPEPTIDES
5Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
02containing at least one abnormal peptide link
0207containing the structure -NH-(X)4-C(=0), e.g. 'isosters', replacing two amino acids
Applicants
  • TAKEDA CHEMICAL INDUSTRIES, LTD. [JP/JP]; 1-1, Doshomachi 4-chome Chuo-ku Osaka-shi Osaka 541-0045, JP (AllExceptUS)
  • KAMIYAMA, Keiji [JP/JP]; JP (UsOnly)
  • NISHIKIMI, Yuji [JP/JP]; JP (UsOnly)
  • HASUOKA, Atsushi [JP/JP]; JP (UsOnly)
  • NAKAO, Masafumi [JP/JP]; JP (UsOnly)
  • MIYAGAWA, Ken-ichiro [JP/JP]; JP (UsOnly)
  • AKIYAMA, Yohko [JP/JP]; JP (UsOnly)
Inventors
  • KAMIYAMA, Keiji; JP
  • NISHIKIMI, Yuji; JP
  • HASUOKA, Atsushi; JP
  • NAKAO, Masafumi; JP
  • MIYAGAWA, Ken-ichiro; JP
  • AKIYAMA, Yohko; JP
Agents
  • TAKAHASHI, Shuichi ; Osaka Plant of Takeda Chemical Industries, Ltd. 17-85, Jusohonmachi 2-chome Yodogawa-ku Osaka-shi Osaka 532-0024, JP
  • ELKINGTON AND FIFE; Prospect House 8 Pembroke Road Sevenoaks Kent TN13 1XR, GB
Priority Data
11/189807.01.1999JP
Publication Language English (EN)
Filing Language English (EN)
Designated States
Title
(EN) POLYOL COMPOUNDS, THEIR PRODUCTION AND USE
(FR) COMPOSES DE POLYOL, PRODUCTION ET UTILISATION DE CES DERNIERS
Abstract
(EN)
A compound of formula (I) wherein X is L-serine residue, L-asparagine residue or (S)-2-aminobutyric acid residue and Y is $g(a)-L-amino acid residue, its salt or its pro-drug has remarkable antibacterial activity against $i(Helicobacter) bacteria.
(FR)
L'invention a pour objet un composé selon la formule (I). Dans cette dernière, X est un résidu de L-sérine, L-asparagine ou d'acide (S)-2-aminobutyrique et Y représente un résidu d'acide $g(a)-L-amine, son sel ou son promédicament . Ce composé présente une excellente activité antibactérienne contre les bactérie de $i(Helicobacter) .
Also published as
US09857887
Latest bibliographic data on file with the International Bureau