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1. WO1999059591 - PYRAZINONE THROMBIN INHIBITORS

Publication Number WO/1999/059591
Publication Date 25.11.1999
International Application No. PCT/US1999/010730
International Filing Date 14.05.1999
Chapter 2 Demand Filed 01.12.1999
IPC
C07D 241/20 2006.01
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
241Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
02not condensed with other rings
10having three double bonds between ring members or between ring members and non-ring members
14with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
20Nitrogen atoms
C07D 401/12 2006.01
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
401Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
02containing two hetero rings
12linked by a chain containing hetero atoms as chain links
CPC
A61P 43/00
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
43Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
A61P 7/02
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
7Drugs for disorders of the blood or the extracellular fluid
02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
C07D 241/20
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
241Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
02not condensed with other rings
10having three double bonds between ring members or between ring members and non-ring members
14with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
20Nitrogen atoms
C07D 401/12
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
401Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
02containing two hetero rings
12linked by a chain containing hetero atoms as chain links
Applicants
  • MERCK & CO., INC. [US]/[US] (AllExceptUS)
  • SANDERSON, Philip, E. [GB]/[US] (UsOnly)
  • STANTON, Matthew, G. [US]/[US] (UsOnly)
  • BALANI, Suresh, K. [US]/[US] (UsOnly)
Inventors
  • SANDERSON, Philip, E.
  • STANTON, Matthew, G.
  • BALANI, Suresh, K.
Common Representative
  • MERCK & CO., INC.
Priority Data
60/085,98019.05.1998US
9813580.924.06.1998GB
Publication Language English (EN)
Filing Language English (EN)
Designated States
Title
(EN) PYRAZINONE THROMBIN INHIBITORS
(FR) INHIBITEURS DE THROMBINE A BASE DE PYRAZINONE
Abstract
(EN)
Compounds of the invention are useful in inhibiting thrombin and associated thrombotic occlusions having structure (A), wherein (B).
(FR)
L'invention concerne des composés utiles pour inhiber la thrombine et des occlusions thrombotiques associées, qui possèdent la structure (A), notamment (B).
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