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Machine translation
1. (WO1999041244) SUBSTITUTED AMINOPHENYL ISOXAZOLINE DERIVATIVES USEFUL AS ANTIMICROBIALS
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/1999/041244    International Application No.:    PCT/US1999/001854
Publication Date: 19.08.1999 International Filing Date: 03.02.1999
Chapter 2 Demand Filed:    21.07.1999    
IPC:
C07D 261/04 (2006.01), C07D 413/10 (2006.01), C07D 413/12 (2006.01), C07D 417/10 (2006.01), C07D 521/00 (2006.01)
Applicants: PHARMACIA & UPJOHN COMPANY [US/US]; 301 Henrietta Street Kalamazoo, MI 49001 (US) (For All Designated States Except US).
BARBACHYN, Michael, R. [US/US]; (US) (For US Only).
MORRIS, Joel [US/US]; (US) (For US Only).
WISHKA, Donn, G. [US/US]; (US) (For US Only).
THOMAS, Richard, C. [US/US]; (US) (For US Only).
CLEEK, Gary, J. [US/US]; (US) (For US Only)
Inventors: BARBACHYN, Michael, R.; (US).
MORRIS, Joel; (US).
WISHKA, Donn, G.; (US).
THOMAS, Richard, C.; (US).
CLEEK, Gary, J.; (US)
Agent: YANG, Lucy, X.; Intellectual Property Legal Services Pharmacia & Upjohn Company 301 Henrietta Street Kalamazoo, MI 49001 (US).
PERRY Robert Edward Gill Jennings & Every; Gill Jenings & Every Broadgate House 7 Eldon Street London EC2M 7LH (GB)
Priority Data:
60/075,126 13.02.1998 US
Title (EN) SUBSTITUTED AMINOPHENYL ISOXAZOLINE DERIVATIVES USEFUL AS ANTIMICROBIALS
(FR) DERIVES D'ISOXAZOLINE AMINOPHENYLE SUBSTITUES UTILISES COMME AGENTS ANTIMICROBIENS
Abstract: front page image
(EN)The present invention provides novel substituted aminophenyl isoxazoline derivatives of formula (I), wherein R¿1? is H, alkyl, cycloalkyl, alkoxy, amino, or alkylamino; X and Y are the same and different and are H, F, or CH¿3?; W is O, or S; Q is a 4-, 5-, 6-, 7-, or 9-membered heterocyclic moiety containing one or more nitrogen, sulfur and/or oxygen. The compounds of the invention are useful as antimicrobial agents for preventing and treating infectious diseases.
(FR)La présente invention porte sur de nouveaux dérivés d'isoxazoline aminophényle substitués de la formule (I) dans laquelle R¿1? représente H, alkyle, cycloalkyle, amino ou alkylamino; X et Y sont identiques et différents et représentent H, F ou CH¿3?; W représente O, S; Q représente une fraction hétérocyclique à 4, 5, 6, 7 ou 9 éléments et contenant au moins un azote, soufre et/ou oxygène. Les composés de cette invention sont utiles comme agents antimicrobiens dans la prévention et le traitement de maladies infectieuses.
Designated States: AL, AM, AT, AU, AZ, BA, BB, BG, BR, BY, CA, CH, CN, CU, CZ, DE, DK, EE, ES, FI, GB, GD, GE, GH, GM, HR, HU, ID, IL, IN, IS, JP, KE, KG, KP, KR, KZ, LC, LK, LR, LS, LT, LU, LV, MD, MG, MK, MN, MW, MX, NO, NZ, PL, PT, RO, RU, SD, SE, SG, SI, SK, SL, TJ, TM, TR, TT, UA, UG, US, UZ, VN, YU, ZW.
African Regional Intellectual Property Organization (GH, GM, KE, LS, MW, SD, SZ, UG, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, CH, CY, DE, DK, ES, FI, FR, GB, GR, IE, IT, LU, MC, NL, PT, SE)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GW, ML, MR, NE, SN, TD, TG).
Publication Language: English (EN)
Filing Language: English (EN)