Search International and National Patent Collections

1. (WO1999005140) INDOLE AND 2,3-DIHYDROINDOLE DERIVATIVES, THEIR PREPARATION AND USE

Pub. No.:    WO/1999/005140    International Application No.:    PCT/DK1998/000336
Publication Date: Fri Feb 05 00:59:59 CET 1999 International Filing Date: Tue Jul 21 01:59:59 CEST 1998
IPC: C07D 405/12
C07D 405/14
C07D 409/12
Applicants: H. LUNDBECK A/S
MOLTZEN, Ejner, Knud
PERREGAARD, Jens, Kristian
MIKKELSEN, Ivan
SMITH, Garrick, Paul
Inventors: MOLTZEN, Ejner, Knud
PERREGAARD, Jens, Kristian
MIKKELSEN, Ivan
SMITH, Garrick, Paul
Title: INDOLE AND 2,3-DIHYDROINDOLE DERIVATIVES, THEIR PREPARATION AND USE
Abstract:
The present invention relates to indole and 2,3-dihydroindole derivatives having formula (I) any of its enantiometers or any mixture thereof, or an acid addition salt thereof, wherein A, R?1, R2, R3¿, W, X, Y and Z are as described in the description. The compounds are potent serotonin reuptake inhibitors and have 5-HT¿1A? receptor antagonistic activity.