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1. (WO1998031704) TACHYKININ ANTAGONISTS
Latest bibliographic data on file with the International Bureau   

Pub. No.: WO/1998/031704 International Application No.: PCT/EP1997/007307
Publication Date: 23.07.1998 International Filing Date: 29.12.1997
Chapter 2 Demand Filed: 20.07.1998
IPC:
A61K 38/00 (2006.01) ,C07K 5/078 (2006.01) ,C07K 7/22 (2006.01)
Applicants: WALPOLE, Christopher, Simon, John[GB/CA]; CA (UsOnly)
PRASHAD, Mahavir[IN/US]; US (UsOnly)
HAR, Denis[US/US]; US (UsOnly)
NOVARTIS AG[CH/CH]; Schwarzwaldallee 215 CH-4058 Basel, CH (AL, AM, AT, AU, AZ, BA, BB, BE, BF, BG, BJ, BR, BY, CA, CF, CG, CH, CI, CM, CN, CU, CZ, DE, DK, EE, ES, FI, FR, GA, GB, GE, GH, GM, GN, GR, GW, HU, ID, IE, IL, IS, IT, JP, KE, KG, KP, KR, KZ, LC, LK, LR, LS, LT, LU, LV, MC, MD, MG, MK, ML, MN, MR, MW, MX, NE, NL, NO, NZ, PL, PT, RO, RU, SD, SE, SG, SI, SK, SL, SN, SZ, TD, TG, TJ, TM, TR, TT, UA, UG, UZ, VN, YU, ZW)
NOVARTIS PHARMACEUTICALS UK LIMITED[GB/GB]; Calverley Lane Horsforth Leeds LS18 4RP, GB (GB)
Inventors: WALPOLE, Christopher, Simon, John; CA
PRASHAD, Mahavir; US
HAR, Denis; US
Agent: ROTH, Bernhard, M.; Novartis AG Patent- und Markenabteilung Lichtstrasse 35 CH-4002 Basel, CH
Priority Data:
9700597.914.01.1997GB
Title (EN) TACHYKININ ANTAGONISTS
(FR) ANTAGONISTES DE TACHYKININE
Abstract:
(EN) Compounds of formula (I) wherein X is -CH2-, -CO- or direct linkage, Y is -O-, -S- or -NH-, R1 is phenyl, R2=H or phenyl and R3 is H or -CH3- and their pharmaceutically acceptable salts have tachykinin antagonist activity and are useful as pharmaceuticals e.g. for the treatment of pain and migraine.
(FR) Composés représentés par la formule (I) dans laquelle X représente -CH2-, -CO- ou une liaison directe, Y représente -O-, -S- ou -NH-, R1 représente phényle, R2 représente H ou phényle et R3 représente H ou -CH3-, ainsi que leurs sels acceptables sur le plan pharmaceutique, actifs en tant qu'antagonistes de tachykinine et utiles en tant que remèdes pharmaceutiques, afin de traiter, par exemple, la douleur et la migraine.
Designated States: AL, AM, AT, AU, AZ, BA, BB, BG, BR, BY, CA, CH, CN, CU, CZ, DE, DK, EE, ES, FI, GB, GE, GH, GM, GW, HU, ID, IL, IS, JP, KE, KG, KP, KR, KZ, LC, LK, LR, LS, LT, LU, LV, MD, MG, MK, MN, MW, MX, NO, NZ, PL, PT, RO, RU, SD, SE, SG, SI, SK, SL, TJ, TM, TR, TT, UA, UG, US, UZ, VN, YU, ZW
African Regional Intellectual Property Organization (ARIPO) (GH, GM, KE, LS, MW, SD, SZ, UG, ZW)
Eurasian Patent Office (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (EPO) (AT, BE, CH, DE, DK, ES, FI, FR, GB, GR, IE, IT, LU, MC, NL, PT, SE)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, ML, MR, NE, SN, TD, TG)
Publication Language: English (EN)
Filing Language: English (EN)