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Machine translation
1. (WO1998030549) PROCESS FOR PREPARING SUBSTITUTED PYRIMIDINE DERIVATIVES
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/1998/030549    International Application No.:    PCT/EP1998/000074
Publication Date: 16.07.1998 International Filing Date: 08.01.1998
Chapter 2 Demand Filed:    20.07.1998    
IPC:
C07D 239/36 (2006.01), C07D 239/40 (2006.01)
Applicants: LONZA AG [CH/CH]; CH-3945 Gampel (CH) (For All Designated States Except US).
SCHMIDT, Beat [CH/CH]; (CH) (For US Only).
STUCKY, Gerhard [CH/CH]; (CH) (For US Only)
Inventors: SCHMIDT, Beat; (CH).
STUCKY, Gerhard; (CH)
Agent: WEINHOLD, Peter; Alois-Steinecker-Strasse 22, D-85354 Freising (DE)
Priority Data:
55/97 13.01.1997 CH
Title (DE) VERFAHREN ZUR HERSTELLUNG VON SUBSTITUIERTEN PYRIMIDINDERIVATEN
(EN) PROCESS FOR PREPARING SUBSTITUTED PYRIMIDINE DERIVATIVES
(FR) PROCEDE DE PREPARATION DE DERIVES DE PYRIMIDINE SUBSTITUES
Abstract: front page image
(DE)Es wird ein neues Verfahren zur Herstellung von substituierten Pyrimidinderivaten der allgemeinen Formel (I) beschrieben, worin ein [3-(Dimethylamino)-2-azaprop-2-en-1-yliden]dimethylammoniumhalogenid mit einem substituierten Acetamid umgesetzt wird. Die Verbindungen der allgemeinen Formel (I) sind bedeutende Zwischenprodukte für pharmazeutische oder agrochemische Wirkstoffe.
(EN)The invention concerns a novel process for preparing substituted pyrimidine derivatives of general formula (I) in which a [3-(dimethylamino)-2-azaprop-2-en-1-ylidene]dimethylammonium halide is reacted with a substituted acetamide. The compounds of general formula (I) are important intermediate products for pharmaceutical or agrochemical active substances.
(FR)L'invention concerne un nouveau procédé de préparation de dérivés de pyrimidine substitués de la formule générale (I) dans laquelle un [3-(diméthylamino)-2-azaprop-2-ène-1-ylidène]halogénure de diméthylammonium est mis à réagir avec un acétamide substitué. Les composés de la formule générale (I) sont des produits intermédiaires significatifs pour des principes actifs pharmaceutiques ou agrochimiques.
Designated States: AL, AM, AT, AU, AZ, BA, BB, BG, BR, BY, CA, CH, CN, CU, CZ, DE, DK, EE, ES, FI, GB, GE, GH, GM, GW, HU, ID, IL, IS, JP, KE, KG, KP, KR, KZ, LC, LK, LR, LS, LT, LU, LV, MD, MG, MK, MN, MW, MX, NO, NZ, PL, PT, RO, RU, SD, SE, SG, SI, SK, SL, TJ, TM, TR, TT, UA, UG, US, UZ, VN, YU, ZW.
African Regional Intellectual Property Organization (GH, GM, KE, LS, MW, SD, SZ, UG, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, CH, DE, DK, ES, FI, FR, GB, GR, IE, IT, LU, MC, NL, PT, SE)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, ML, MR, NE, SN, TD, TG).
Publication Language: German (DE)
Filing Language: German (DE)