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1. (WO1997036883) 1,3,4-OXADIAZINE DERIVATIVES AND THEIR USE AS PESTICIDES
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/1997/036883    International Application No.:    PCT/EP1997/001325
Publication Date: 09.10.1997 International Filing Date: 17.03.1997
Chapter 2 Demand Filed:    17.07.1997    
IPC:
A01N 43/88 (2006.01), B27K 3/34 (2006.01), C07C 281/02 (2006.01), C07D 209/14 (2006.01), C07D 273/04 (2006.01), C07D 317/28 (2006.01), C07D 333/20 (2006.01), C07D 413/06 (2006.01)
Applicants: BAYER AKTIENGESELLSCHAFT [DE/DE]; D-51368 Leverkusen (DE) (For All Designated States Except US).
DYKER, Hubert [DE/DE]; (DE) (For US Only).
PLANT, Andrew [GB/DE]; (DE) (For US Only).
SCHERKENBECK, Jürgen [DE/DE]; (DE) (For US Only).
ERDELEN, Christoph [DE/DE]; (DE) (For US Only).
HARDER, Achim [DE/DE]; (DE) (For US Only)
Inventors: DYKER, Hubert; (DE).
PLANT, Andrew; (DE).
SCHERKENBECK, Jürgen; (DE).
ERDELEN, Christoph; (DE).
HARDER, Achim; (DE)
Common
Representative:
BAYER AKTIENGESELLSCHAFT; D-51368 Leverkusen (DE)
Priority Data:
196 12 644.4 29.03.1996 DE
Title (DE) 1,3,4-OXADIAZIN-DERIVATE UND IHRE VERWENDUNG ALS SCHÄDLINGSBEKÄMPFUNGSMITTEL
(EN) 1,3,4-OXADIAZINE DERIVATIVES AND THEIR USE AS PESTICIDES
(FR) DERIVES DE 1,3,4-OXADIAZINE ET LEUR UTILISATION COMME PESTICIDES
Abstract: front page image
(DE)Die Erfindung betrifft neue (1,3,4)-Oxadiazin-Derivat der Formel (I), in welcher R?1¿ und R?2¿ unabhängig voneinander für Wasserstoff, jeweils gegebenenfalls durch Halogen substituiertes Alkyl, Hydroxyalkyl, Alkanoyloxyalkyl, Alkoxyalkyl, Arylalkoxyalkyl, Mercaptoalkyl, Alkylthioalkyl, Alkylsulfinylalkyl, Alkylsulfonylalkyl, Carboxyalkyl, Alkoxycarbonylalkyl, Aryloxycarbonylalkyl, Arylalkyloxycarbonylalkyl, Carbamoylalkyl, Aminoalkyl, Alkylaminoalkyl, Dialkylaminoalkyl, Alkoxycarbonylaminoalkyl, Alkylcarbonyl, Cycloalkylcarbonyl oder für jeweils gegebenenfalls substituiertes Cycloalkyl, Cycloalkylalkyl, Aryl, Arylalkyl, Arylcarbonyl, Heterocyclylalkyl, Hetaryl oder Hetarylalkyl stehen oder R?1¿, R?2¿ und die beiden Stickstoffatome, an die sie gebunden sind, für einen gegebenenfalls substituierten heterocyclischen Ring stehen, R?3¿ und R?4¿ unabhängig voneinander für Wasserstoff, jeweils gegebenenfalls durch Halogen substituiertes Alkyl, Alkenyl, Hydroxyalkyl, Alkanoyloxyalkyl, Alkoxyalkyl, Arylalkoxyalkyl, Mercaptoalkyl, Alkylthioalkyl, Alkylsufinylalkyl, Alkylsulfonylalkyl, Alkoxycarbonylalkyl, Aryloxycarbonylalkyl, Arylalkyloxycarbonylalkyl, Carbamoylalkyl, Aminoalkyl, Alkylaminoalkyl, Dialkylaminoalkyl, Alkylcarbonyl, Cycloalkylcarbonyl oder für jeweils gegebenenfalls subsituiertes Cycloalkyl, Cycloalkylalkyl, Aryl, Arylalkyl, Hetaryl oder Hetarylalkyl stehen oder R?3¿ und R?4¿ gemeinsam für Alkylen oder den Rest (a) stehen, worin R?5¿ und R?6¿ unabhängig voneinander für Wasserstoff, jeweils gegebenenfalls durch Halogen subsituiertes Alkyl, Alkenyl, Hydroxyalkyl, Alkanoyloxyalkyl, Alkoxyalkyl, Arylalkoxyalkyl, Mercaptoalkyl, Alkylthioalkyl, Alkylsufinylalkyl, Alkylsulfonylalkyl, Alkoxycarbonylalkyl, Aryloxycarbonylalkyl, Aminoalkyl, Alkylaminoalkyl, Dialkylaminoalkyl, Alkylcarbonyl oder für jeweils gegebenenfalls subsituiertes Cycloalkyl, Cycloalkylalkyl, Aryl, Arylalkyl, Hetaryl oder Hetarylalkyl stehen und Q?1¿ und Q?2¿ unabhängig voneinander für Sauerstoff oder Schwefel stehen, wobei 6,6-Diphenyl-(1,3,4)-oxadiazinan-2,5-dion ausgenommen ist, Verfahren zu ihrer Herstellung und ihre Verwendung als Schädlingsbekämfungsmittel und Endoparasiten.
(EN)The invention concerns novel (1,3,4)-oxadiazine derivatives of formula (I) in which: R?1¿ and R?2¿, independently of each other, stand for hydrogen, or for alkyl, hydroxylalkyl, alkanoyloxyalkyl, alkoxyalkyl, arylalkoxyalkyl, mercaptoalkyl, alkylthioalkyl, alkylsulphinylalkyl, alkylsulphonylalkyl, carboxyalkyl, alkoxycarbonylalkyl, aryloxycarbonylalkyl, arylalkyloxycarbonylalkyl, carbamoylalkyl, aminoalkyl, alkylaminoalkyl, dialkylaminoalkyl, alkoxycarbonylaminoalkyl, alkylcarbonyl, cycloalkylcarbonyl in each case optionally substituted by halogen, or for in each case optionally substituted cycloalkyl, cycloalkylalkyl, aryl, arylalkyl, arylcarbonyl, heterocyclylalkyl, hetaryl or hetarylalkyl; or R?1¿, R?2¿ and the two nitrogen atoms to which they are bonded stand for an optionally substituted heterocyclic ring; R?3¿ and R?4¿, independently of each other, stand for hydrogen, or for alkyl, alkenyl, hydroxyalkyl, alkanoyloxyalkyl, alkoxyalkyl, arylalkoxyalkyl, mercaptoalkyl, alkylthioalkyl, alkylsulphinylalkyl, alkylsulphonylalkyl, alkoxycarbonylalkyl, aryloxycarbonylalkyl, arylalkyloxycarbonylalkyl, carbamoylalkyl, aminoalkyl, alkylaminoalkyl, dialkylaminoalkyl, alkylcarbonyl, cycloalkylcarbonyl in each case optionally substituted by halogen, or for in each case optionally substituted cycloalkyl, cycloalkylalkyl, aryl, arylalkyl, hetaryl or hetarylalkyl; or R?3¿ and R?4¿ jointly stand for alkylene or the group (a), in which R?5¿ and R?6¿, independently of each other, stand for hydrogen, or for alkyl, alkenyl, hydroxyalkyl, alkanoyloxyalkyl, alkoxyalkyl, arylalkoxyalkyl, mercaptoalkyl, alkylthioalkyl, alkylsulphinylalkyl, alkylsulphonylalkyl, alkoxycarbonylalkyl, aryloxycarbonylalkyl, aminoalkyl, alkylaminoalkyl, dialkylaminoalkyl, alkylcarbonyl in each case optionally substituted by halogen, or for in each case optionally substituted cycloalkyl, cycloalkylalkyl, aryl, arylalkyl, hetaryl or hetarylalkyl; and Q?1¿ and Q?2¿, independently of each other, stand for oxygen or sulphur, 6,6-diphenyl-(1,3,4)-oxadiazinane-2,5-dione being excluded. The invention also concerns a process for preparing these substances and their use as pesticides and endoparasites.
(FR)L'invention concerne de nouveaux dérivés de (1,3,4)-oxadiazine de la formule (I), dans laquelle R?1¿ et R?2¿, indépendamment l'un de l'autre, représentent hydrogène, ou bien alkyle, hydroxyalkyle, alcanoyloxyalkyle, alcoxyalkyle, arylalcoxyalkyle, mercaptoalkyle, alkylthioalkyle, alkylsulfinylalkyle, alkylsulfonylalkyle, carboxyalkyle, alcoxycarbonylalkyle, aryloxycarbonylalkyle, arylalkyloxycarbonylalkyle, carbamoyalkyle, aminoalkyle, alkylaminoalkyle, dialkylaminoalkyle, alcoxycarbonylaminoalkyle, alkylcarbonyle, cycloalkylcarbonyle, chacun de ces groupes pouvant être substitué par halogène, ou bien cycloalkyle, cycloalkylalkyle, aryle, arylalkyle, arylcarbonyle, hétérocyclylalkyle, hétaryle ou hétarylalkyle, chacun de ces groupes pouvant aussi être substitué; ou R?1¿, R?2¿ et les deux atomes d'azote auxquels ils sont liés représentent un noyau hétérocyclique éventuellement substitué; R?3¿ et R?4¿, indépendamment l'un de l'autre, représentent hydrogène, ou bien alkyle, alcényle, hydroxyalkyle, alcanoyloxyalkyle, alcoxyalkyle, arylalcoxyalkyle, mercaptoalkyle, alkylthioalkyle, alkylsulfinylalkyle, alkylsulfonylalkyle, alcoxycarbonylalkyle, aryloxycarbonylalkyle, arylalkyloxycarbonylalkyle, carbamoylalkyle, aminoalkyle, alkylaminoalkyle, dialkylaminoalkyle, alkylcarbonyle, cycloalkylcarbonyle, chacun de ces groupes pouvant être substitué par halogène, ou bien représente cycloalkyle, cycloalkylalkyle, aryle, arylalkyle, hétaryle ou hétarylalkyle, chacun de ces groupes pouvant aussi être substitué; ou bien R?3¿ et R?4¿ représentent ensemble alkylène ou le groupe (a), dans lequel R?5¿ et R?6¿, indépendamment l'un de l'autre, représentent hydrogène ou bien alkylalcényle, hydroxyalkyle, alcanoyloxyalkyle, alcoxyalkyle, arylalcoxyalkyle, mercaptoalkyle, alkylthioalkyle, alkylsulfinylalkyle, alkylsulfonylalkyle, alcoxycarbonylalkyle, aryloxycarbonylalkyle, aminoalkyle, alkylaminoalkyle, dialkylaminoalkyle, alkylcarbonyle, chacun de ces groupes pouvant être substitué par halogène, ou bien représente cycloalkyle, cycloalkylalkyle, aryle, arylalkyle, hétaryle ou hétarylalkyle, chacun de ces groupes pouvant également être substitué; et Q?1¿ et Q?2¿, indépendamment l'un de l'autre, représentent oxygène ou soufre, la 6,6-diphényle-(1,3,4)-oxadiazinan-2,5-dione étant exclue. L'invention concerne également un procédé de production de ces dérivés et leur utilisation comme pesticides et endoparasites.
Designated States: AU, BB, BG, BR, BY, CA, CN, CZ, HU, IL, JP, KR, KZ, LK, MX, NO, NZ, PL, RO, RU, SK, TR, UA, US.
European Patent Office (AT, BE, CH, DE, DK, ES, FI, FR, GB, GR, IE, IT, LU, MC, NL, PT, SE)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, ML, MR, NE, SN, TD, TG).
Publication Language: German (DE)
Filing Language: German (DE)