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Machine translation
1. (WO1997022594) COMBINATORIAL LIBRARIES
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/1997/022594    International Application No.:    PCT/DK1996/000534
Publication Date: 26.06.1997 International Filing Date: 16.12.1996
Chapter 2 Demand Filed:    24.05.1997    
IPC:
C07B 61/00 (2006.01), C07D 237/32 (2006.01)
Applicants: PHYTERA SYMBION APS [DK/DK]; Forskerbyen Symbion, Fruebjergvej 3, DK-2100 Copenhagen Ø (DK) (For All Designated States Except US).
NIELSEN, John [DK/DK]; (DK) (For US Only)
Inventors: NIELSEN, John; (DK)
Agent: PLOUGMANN, VINGTOFT & PARTNERS; Sankt Annæ Plads 11, P.O. Box 3007, DK-1021 Copenhagen K (DK)
Priority Data:
1419/95 15.12.1995 DK
Title (EN) COMBINATORIAL LIBRARIES
(FR) BANQUES COMBINATOIRES
Abstract: front page image
(EN)The invention provides a method for the production of a combinatorial library of compound of general formula (I) using solid phase methodologies. The cleavage of the array of immobilised compounds of the phthalimido type from the solid support matrix is accomplished by using an array of dinucleophiles, e.g. hydrazines (hydrazinolysis) or N-hydroxylamines, whereby a combinatorial dimension is introduced in the cleavage step. The invention also provides a compound library.
(FR)Procédé de production d'une banque combinatoire de composés répondant à la formule générale (I), à l'aide de méthodes du type en phase solide. On effectue le clivage de l'ensemble de composés immobilisés du type phtalimido à partir de la matrice support solide, en faisant intervenir un ensemble de dinucléophiles, par exemple des hydrazines (hydrazinolyse) ou des N-hydroxylamines, de manière à apporter à l'étape de clivage une dimension combinatoire. On décrit également une banque de composés.
Designated States: AL, AM, AT, AU, AZ, BA, BB, BG, BR, BY, CA, CH, CN, CU, CZ, DE, DK, EE, ES, FI, GB, GE, HU, IL, IS, JP, KE, KG, KP, KR, KZ, LC, LK, LR, LS, LT, LU, LV, MD, MG, MK, MN, MW, MX, NO, NZ, PL, PT, RO, RU, SD, SE, SG, SI, SK, TJ, TM, TR, TT, UA, UG, US, UZ, VN.
African Regional Intellectual Property Organization (KE, LS, MW, SD, SZ, UG)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, CH, DE, DK, ES, FI, FR, GB, GR, IE, IT, LU, MC, NL, PT, SE)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, ML, MR, NE, SN, TD, TG).
Publication Language: English (EN)
Filing Language: English (EN)